ATE465999T1 - Verfahren zur herstellung substituierter pyrimidine - Google Patents

Verfahren zur herstellung substituierter pyrimidine

Info

Publication number
ATE465999T1
ATE465999T1 AT06759727T AT06759727T ATE465999T1 AT E465999 T1 ATE465999 T1 AT E465999T1 AT 06759727 T AT06759727 T AT 06759727T AT 06759727 T AT06759727 T AT 06759727T AT E465999 T1 ATE465999 T1 AT E465999T1
Authority
AT
Austria
Prior art keywords
formula
compound
substituted pyrimidines
producing substituted
bromophenyl
Prior art date
Application number
AT06759727T
Other languages
English (en)
Inventor
Gary Annis
Original Assignee
Du Pont
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont filed Critical Du Pont
Application granted granted Critical
Publication of ATE465999T1 publication Critical patent/ATE465999T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C07D239/36—One oxygen atom as doubly bound oxygen atom or as unsubstituted hydroxy radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT06759727T 2005-05-16 2006-05-12 Verfahren zur herstellung substituierter pyrimidine ATE465999T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68129805P 2005-05-16 2005-05-16
PCT/US2006/018522 WO2006124657A1 (en) 2005-05-16 2006-05-12 Method for preparing substituted pyrimidines

Publications (1)

Publication Number Publication Date
ATE465999T1 true ATE465999T1 (de) 2010-05-15

Family

ID=36867439

Family Applications (1)

Application Number Title Priority Date Filing Date
AT06759727T ATE465999T1 (de) 2005-05-16 2006-05-12 Verfahren zur herstellung substituierter pyrimidine

Country Status (13)

Country Link
US (1) US8013155B2 (de)
EP (1) EP1888536B1 (de)
JP (1) JP5069677B2 (de)
KR (1) KR101348458B1 (de)
CN (1) CN101175730B (de)
AT (1) ATE465999T1 (de)
AU (1) AU2006247581B2 (de)
BR (1) BRPI0612414A2 (de)
DE (1) DE602006013970D1 (de)
IL (1) IL185884A (de)
PL (1) PL1888536T3 (de)
WO (1) WO2006124657A1 (de)
ZA (1) ZA200707974B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ME00498B (me) * 2005-05-06 2011-10-10 Du Pont Postupak za dobijanje opciono 2-supstituisanih 1,6-dihidr0-6-0ks0-4- pirimidinkarboksilnih kiselina
WO2007120706A2 (en) * 2006-04-10 2007-10-25 E. I. Du Pont De Nemours And Company Herbicidal mixtures
WO2013124246A1 (de) 2012-02-22 2013-08-29 Bayer Intellectual Property Gmbh Herbizid wirksame 4-dialkoxymethyl-2-phenylpyrimidine
CN102977050B (zh) * 2012-11-20 2015-04-22 浙江工业大学 一种2-苯并噻唑二甲缩醛和2-苯并噻唑甲醛的合成方法
CN116063179A (zh) * 2023-02-20 2023-05-05 南京杰运医药科技有限公司 一种4-甲氧基乙酰乙酸甲酯的合成方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA207185A (en) 1921-01-04 C. Wagner Virgil Warming plate
GB2095240A (en) * 1981-03-05 1982-09-29 Fujisawa Pharmaceutical Co Dihydropyrimidine derivatives, processes for preparation thereof and pharmaceutical composition comprising the same
JPS57158779A (en) * 1981-03-05 1982-09-30 Fujisawa Pharmaceut Co Ltd Dihydropyrimidine derivative and its salt, their preparation and antiallergic containing the same
DE3935277A1 (de) 1989-10-24 1991-05-02 Hoechst Ag Sulfonierte heterocyclische carboxamide, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als herbizide oder wachstumsregulatoren
CN1071049A (zh) * 1991-10-09 1993-04-21 纳幕尔杜邦公司 用于稻中杂草防治的除草剂
ATE245641T1 (de) * 1998-02-17 2003-08-15 Tularik Inc Antivirale pyrimidinderivate
ES2240093T3 (es) 1999-04-15 2005-10-16 Basf Aktiengesellschaft Procedimiento para la preparacion de pirimidinas substituidas.
US20030130264A1 (en) 2001-02-16 2003-07-10 Tularik Inc. Methods of using pyrimidine-based antiviral agents
ATE440825T1 (de) * 2003-06-06 2009-09-15 Vertex Pharma Pyrimidin-derivate zur verwendung als modulatoren von atp-bindende kassette transportern
TWI355894B (en) * 2003-12-19 2012-01-11 Du Pont Herbicidal pyrimidines
ME00498B (me) * 2005-05-06 2011-10-10 Du Pont Postupak za dobijanje opciono 2-supstituisanih 1,6-dihidr0-6-0ks0-4- pirimidinkarboksilnih kiselina

Also Published As

Publication number Publication date
US20090054647A1 (en) 2009-02-26
AU2006247581A1 (en) 2006-11-23
JP2008540655A (ja) 2008-11-20
IL185884A0 (en) 2008-01-06
BRPI0612414A2 (pt) 2010-11-09
PL1888536T3 (pl) 2010-09-30
US8013155B2 (en) 2011-09-06
KR20080016640A (ko) 2008-02-21
EP1888536A1 (de) 2008-02-20
DE602006013970D1 (de) 2010-06-10
KR101348458B1 (ko) 2014-01-07
WO2006124657A1 (en) 2006-11-23
AU2006247581B2 (en) 2011-10-20
EP1888536B1 (de) 2010-04-28
CN101175730B (zh) 2011-05-25
JP5069677B2 (ja) 2012-11-07
ZA200707974B (en) 2008-11-26
CN101175730A (zh) 2008-05-07
IL185884A (en) 2012-03-29

Similar Documents

Publication Publication Date Title
ATE371657T1 (de) Verfahren zur herstellung kondensierter oxazinone aus einer aromatischen ortho-aminocarbonsäure und einer carbonsäure in gegenwart eines sulfonylchlorids und pyridin
ATE506352T1 (de) Verfahren zur herstellung von optional 2- substituierten 1,6-dihydro-6-oxo-4- pyrimidincarboxylsäuren
ATE530531T1 (de) Verfahren zur herstellung von bosentan
UA101482C2 (ru) Способ получения 2'-дезокси-5-азацитидина (децитабина)
ATE465999T1 (de) Verfahren zur herstellung substituierter pyrimidine
ATE552230T1 (de) Verfahren zur herstellung von derivaten aus 1-(2- halobiphenyl-4-yl)-cyclopropancarboxylsäure
WO2008117733A1 (ja) リン含有α－ケト酸の製造法
ATE447567T1 (de) Verfahren zur herstellung von tryptase- inhibitoren
ATE461924T1 (de) Verfahren zur herstellung von rosuvastatin und intermediate
WO2006066044A3 (en) Processes for producing 4-aminoquinazolines
ATE526312T1 (de) Verfahren zur herstellung von reinen 4- pyrrolidinophenylbenzyletherderivaten als maob- inhibitoren
MX2010013758A (es) Procedimiento para elaborar 2-amino-tiazolonas sustituidas.
ATE423764T1 (de) Verfahren zur herstellung von hydrazon-derivaten
ATE423096T1 (de) Verfahren zur herstellung von 2- azabicycloä3.3.0üoctan-3-carbonsäurederivaten
ATE532516T1 (de) Verfahren zur synthese von glyt-1-hemmern
DE602007005077D1 (de) Verfahren zur Herstellung von Pyridinmethylsulphinylverbindungen
RS20060157A (en) Method for the manufacture of thip
ATE555093T1 (de) Verfahren zur herstellung einer (s)-1-alkyl-2i,6i-pipecoloxylididverbindung
ATE519739T1 (de) Neuartiges verfahren zur herstellung von sulphonylpyrrolen als hdac-hemmer
ATE353877T1 (de) Verfahren zur herstellung von monoifluorierten pyridinyl- und pyrimidinyl-beta-ketoestern
ATE469141T1 (de) Verfahren zur herstellung von substituierten thiophensulfonylisocyanaten
ATE517890T1 (de) Verfahren zur herstellung von reinem irbesartan
ATE380183T1 (de) Verfahren zur herstellung von phenyltetrazolderivaten
DE50304869D1 (de) Verfahren zur herstellung einer spezifischen kristallmodifikation von 2-(2-chlor-4-mesyl-benzoyl)-cyclohexan-1,3-dion
MXPA05007217A (es) Proceso para la preparacion de derivados de imidazol sustituidos y los productos intermedios usados en este proceso.

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties