ATE243211T1 - Verfahren zur herstellung von dihalogenazolopyrimidinen - Google Patents

Verfahren zur herstellung von dihalogenazolopyrimidinen

Info

Publication number: ATE243211T1
Authority: AT; Austria
Prior art keywords: dihalogenazolopyrimidines; producing; producing dihalogenazolopyrimidines
Prior art date: 1995-10-27

Application number

AT96307528T

Other languages

English (en)

Inventor

Guenther Krummel

Karl-Otto Stumm

Klaus-Juergen Pees

Peter Heinz Rudi Liers

Original Assignee

Basf Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-10-27

Filing date

1996-10-16

Publication date

2003-07-15

1996-10-16 Application filed by Basf Ag filed Critical Basf Ag

2003-07-15 Application granted granted Critical

2003-07-15 Publication of ATE243211T1 publication Critical patent/ATE243211T1/de

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AT96307528T 1995-10-27 1996-10-16 Verfahren zur herstellung von dihalogenazolopyrimidinen ATE243211T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US802295P	1995-10-27	1995-10-27

Publications (1)

Publication Number	Publication Date
ATE243211T1 true ATE243211T1 (de)	2003-07-15

Family

ID=21729405

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT96307528T ATE243211T1 (de)	1995-10-27	1996-10-16	Verfahren zur herstellung von dihalogenazolopyrimidinen

Country Status (22)

Country	Link
US (1)	US5808066A (de)
EP (1)	EP0770615B1 (de)
JP (1)	JP4018182B2 (de)
KR (1)	KR100443182B1 (de)
AR (1)	AR004122A1 (de)
AT (1)	ATE243211T1 (de)
BR (1)	BR9605258A (de)
CA (1)	CA2188905C (de)
DE (1)	DE69628712T2 (de)
DK (1)	DK0770615T3 (de)
ES (1)	ES2202419T3 (de)
HU (1)	HU217773B (de)
IL (1)	IL119496A (de)
MX (1)	MX9604882A (de)
PT (1)	PT770615E (de)
RU (1)	RU2147584C1 (de)
SG (1)	SG55239A1 (de)
SI (1)	SI0770615T1 (de)
SK (1)	SK284071B6 (de)
TR (1)	TR199600792A2 (de)
UA (1)	UA48132C2 (de)
ZA (1)	ZA968957B (de)

Families Citing this family (40)

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US6117876A (en) *	1997-04-14	2000-09-12	American Cyanamid Company	Fungicidal trifluorophenyl-triazolopyrimidines
DK1054888T3 (da) *	1998-02-11	2004-04-05	Basf Ag	Fungicide 7-alkyl-triazolpyrimidiner
US6117865A (en) *	1998-09-10	2000-09-12	American Cyanamid Company	Fungicidal trifluorophenyl-triazolopyrimidines
US6380202B1 (en) *	1998-09-25	2002-04-30	Basf Aktiengesellschaft	Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines
US6156925A (en) *	1998-09-25	2000-12-05	American Cyanamid Company	Process for the preparation of halogenated phenylmaloates
US6242451B1 (en) *	1998-09-25	2001-06-05	Klaus-Juergen Pees	Fungicidal trihalophenyl-triazolopyrimidines
US6559151B2 (en)	2000-05-08	2003-05-06	Basf Aktiengesellschaft	6-(2-trifluoromethyl-phenyl)-triazolopyrimidines
US6756379B2 (en) *	2001-07-26	2004-06-29	Taro Pharmaceutical Industries Ltd.	Non-sedating barbiturate compounds as neuroprotective agents
US7683071B2 (en) *	2000-07-26	2010-03-23	Taro Pharmaceuticals Industries Ltd.	Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
US6939873B2 (en) *	2000-07-26	2005-09-06	Taro Pharmaceuticals Industries Limited	Non-sedating barbituric acid derivatives
DE10063115A1 (de) *	2000-12-18	2002-06-27	Bayer Ag	Triazolopyrimidine
JP2002249492A (ja) *	2000-12-22	2002-09-06	Nippon Bayer Agrochem Co Ltd	トリアゾロピリミジン類
DE10121101A1 (de) *	2001-04-27	2002-10-31	Bayer Ag	Triazolopyrimidine
WO2003004465A2 (de)	2001-07-05	2003-01-16	Basf Aktiengesellschaft	Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
EP1412356A1 (de)	2001-07-18	2004-04-28	Basf Aktiengesellschaft	Substituierte 6-(2-methoxyphenyl)triazolopyrimidine als fungizide
EA006133B1 (ru)	2001-07-26	2005-10-27	Басф Акциенгезельшафт	7-аминотриазолопиримидины, способ и промежуточные продукты для их получения, содержащие их средства, а также их применение для борьбы с фитопатогенными грибами
ES2287312T3 (es)	2001-09-04	2007-12-16	Sumitomo Chemical Company, Limited	Imidazo(1,2-a)pirimidinas y composiciones fungicidas que las contienen.
US7148227B2 (en)	2002-03-21	2006-12-12	Basf Aktiengesellschaft	Fungicidal triazolopyrimidines, methods for producing the same, use thereof for combating harmful fungi and agents containing said substances
JP4739760B2 (ja) *	2002-12-11	2011-08-03	タロー・ファーマシューティカル・インダストリーズ・リミテッド	バルビツール酸誘導体を使用する運動障害の治療方法
US7419982B2 (en) *	2003-09-24	2008-09-02	Wyeth Holdings Corporation	Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
KR20060098368A (ko) *	2003-09-24	2006-09-18	와이어쓰 홀딩스 코포레이션	항암제로서의 6-[(치환된)페닐]트리아졸로피리미딘
AU2004275728A1 (en) *	2003-09-24	2005-04-07	Wyeth Holdings Corporation	6-aryl-7-halo-imidazo[1,2-a]pyrimidines as anticancer agent
MY179926A (en) *	2003-12-08	2020-11-19	Wyeth Corp	Process for the preparation of tubulin inhibitors
TW200533670A (en) *	2003-12-19	2005-10-16	Basf Ag	6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
DE102004007076A1 (de) *	2004-02-13	2005-08-25	Bayer Cropscience Ag	Imidazolopyrimidine
CA2557781C (en)	2004-03-10	2012-01-10	Basf Aktiengesellschaft	5,6-dialkyl-7-amino-triazolopyrimidines, method for their production, their use for controlling pathogenic fungi and agents containing said compounds
BRPI0508337A (pt) *	2004-03-10	2007-07-24	Basf Ag	compostos, processos para a preparação dos mesmos, agente fungicida, semente, e, processo para o combate de fungos nocivos fitopatogênicos
PE20060020A1 (es) *	2004-03-30	2006-03-10	Basf Ag	5-6-cicloalquil-7-amino-triazolopirimidinas para combatir hongos fitopatogenos y procedimientos para su obtencion
EP1781624A4 (de) *	2004-07-02	2010-06-23	Taro Pharma Ind	Verfahren zur herstellung von 1-methoxymethyl-5,5-diphenylbarbitursäure
US20080188493A1 (en) *	2005-03-01	2008-08-07	Basf Aktiengesellschaft	5,6-Dialkyl-7-Aminoazolopyrimidines, Their Preparation and Their Use For Controlling Harmful Fungi, and Compositions Comprising These Compounds
TW200640928A (en) *	2005-03-01	2006-12-01	Basf Ag	5,6-Dialkyl-7-aminoazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
TW200640927A (en) *	2005-03-01	2006-12-01	Basf Ag	5,6-Dialkyl-7-aminoazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
TW200643022A (en) *	2005-03-02	2006-12-16	Basf Ag	2-substituted 7-aminoazolopyrimidines, processes for their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
JP2008532979A (ja) *	2005-03-10	2008-08-21	ビーエーエスエフソシエタス・ヨーロピア	有害菌類を防除するための４−アミノピリミジン類の使用、新規の４−アミノピリミジン類、それらを調製する方法およびそれらを含む組成物
EP1863752A1 (de) *	2005-03-18	2007-12-12	Basf Aktiengesellschaft	Verfahren zur herstellung von 5-halo-2,4,6-trifluorisophthalsäure
CN101208289A (zh) *	2005-06-27	2008-06-25	巴斯福股份公司	生产取代的苯基丙二酸酯中间体化合物的方法及其在生产5,7-二羟基-6-(2,4,6-三氟苯基)[1,2,4]***并[1,5-a]嘧啶中的用途
US20080200675A1 (en) *	2005-06-27	2008-08-21	Basf Aktiengesellschaft	Method for Production of Substituted Phenylmalonate Esters, Novel Phenylmalonate Esters and Use Thereof
EP2081576A4 (de) *	2006-11-14	2010-06-30	Taro Pharmaceuticals North Ame	Verfahren zur verbesserung der bioverfügbarkeit für nichtsedierende barbiturate
CN101583613A (zh) *	2007-01-11	2009-11-18	巴斯夫欧洲公司	生产芳基取代的稠合嘧啶的方法
WO2011082271A2 (en) *	2009-12-30	2011-07-07	Arqule, Inc.	Substituted triazolo-pyrimidine compounds

Family Cites Families (10)

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US3907799A (en) *	1971-08-16	1975-09-23	Icn Pharmaceuticals	Xanthine oxidase inhibitors
JPS5962593A (ja) *	1982-09-30	1984-04-10	Ss Pharmaceut Co Ltd	３―置換―５，７―ジクロルトリアゾロピリミジン誘導体
DE3522463A1 (de) *	1985-06-22	1987-01-02	Bayer Ag	Herbizide mittel
US4910306A (en) *	1987-11-09	1990-03-20	The Dow Chemical Company	Preparation of substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
US4892945A (en) *	1987-12-21	1990-01-09	Ciba-Geigy Corporation	Isoindoline pigments containing at least one triazolopyrimidone radical
US5006656A (en) *	1990-02-26	1991-04-09	Dowelanco	Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
US5177206A (en) *	1991-10-08	1993-01-05	Dowelanco	Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides
TW224044B (de) *	1991-12-30	1994-05-21	Shell Internat Res Schappej B V
IL108731A (en) *	1993-03-04	1997-03-18	Shell Int Research	6, N-DISUBSTITUTED-£1, 2, 4\| TRIAZOLO-£1, 5-a\| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
EP0724586B1 (de) *	1993-10-18	2002-01-23	Dow AgroSciences LLC	Verfahren zur herstellung von n-(2,6-dichloro-3-methylphenyl)-5-7-dihalo[1,2,4]triazolo[1,5a]pyrimidin-2-sulfonamid durch cyclisierung und halo-dehydroxylierung

1996
- 1996-09-30 RU RU96120421A patent/RU2147584C1/ru not_active IP Right Cessation
- 1996-10-03 TR TR96/00792A patent/TR199600792A2/xx unknown
- 1996-10-15 US US08/729,204 patent/US5808066A/en not_active Expired - Lifetime
- 1996-10-16 DE DE69628712T patent/DE69628712T2/de not_active Expired - Lifetime
- 1996-10-16 SI SI9630630T patent/SI0770615T1/xx unknown
- 1996-10-16 EP EP96307528A patent/EP0770615B1/de not_active Expired - Lifetime
- 1996-10-16 PT PT96307528T patent/PT770615E/pt unknown
- 1996-10-16 ES ES96307528T patent/ES2202419T3/es not_active Expired - Lifetime
- 1996-10-16 DK DK96307528T patent/DK0770615T3/da active
- 1996-10-16 AT AT96307528T patent/ATE243211T1/de not_active IP Right Cessation
- 1996-10-16 MX MX9604882A patent/MX9604882A/es not_active IP Right Cessation
- 1996-10-18 SG SG1996010896A patent/SG55239A1/en unknown
- 1996-10-23 UA UA96104029A patent/UA48132C2/uk unknown
- 1996-10-23 JP JP29790396A patent/JP4018182B2/ja not_active Expired - Fee Related
- 1996-10-24 ZA ZA9608957A patent/ZA968957B/xx unknown
- 1996-10-25 BR BR9605258A patent/BR9605258A/pt not_active IP Right Cessation
- 1996-10-25 SK SK1377-96A patent/SK284071B6/sk unknown
- 1996-10-25 AR ARP960104928A patent/AR004122A1/es active IP Right Grant
- 1996-10-25 CA CA002188905A patent/CA2188905C/en not_active Expired - Fee Related
- 1996-10-25 HU HU9602957A patent/HU217773B/hu not_active IP Right Cessation
- 1996-10-26 KR KR1019960048877A patent/KR100443182B1/ko not_active IP Right Cessation
- 1996-10-27 IL IL11949696A patent/IL119496A/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
IL119496A0 (en)	1997-01-10
UA48132C2 (uk)	2002-08-15
KR100443182B1 (ko)	2005-04-19
MX9604882A (es)	1997-04-30
PT770615E (pt)	2003-10-31
JPH09124651A (ja)	1997-05-13
ZA968957B (en)	1998-04-24
IL119496A (en)	2001-07-24
RU2147584C1 (ru)	2000-04-20
AR004122A1 (es)	1998-09-30
SG55239A1 (en)	1998-12-21
HU217773B (hu)	2000-04-28
TR199600792A2 (tr)	1997-05-21
SI0770615T1 (en)	2003-12-31
EP0770615B1 (de)	2003-06-18
DK0770615T3 (da)	2003-07-14
HUP9602957A3 (en)	1998-01-28
ES2202419T3 (es)	2004-04-01
CA2188905A1 (en)	1997-04-28
SK284071B6 (sk)	2004-09-08
CA2188905C (en)	2005-12-06
KR970021081A (ko)	1997-05-28
JP4018182B2 (ja)	2007-12-05
US5808066A (en)	1998-09-15
EP0770615A1 (de)	1997-05-02
HUP9602957A2 (en)	1997-06-30
DE69628712T2 (de)	2004-04-29
BR9605258A (pt)	1998-07-21
DE69628712D1 (de)	2003-07-24
HU9602957D0 (en)	1996-12-30
SK137796A3 (en)	1997-05-07

Legal Events

Date

Code

Title

Description

2004-01-15

UEP

Publication of translation of european patent specification

Ref document number: 0770615

Country of ref document: EP

2009-07-15

REN

Ceased due to non-payment of the annual fee

Publication	Publication Date	Title
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