ATE154347T1 - Benzisothiazolinon-1-dioxyde als elastase- inhibitoren - Google Patents

Benzisothiazolinon-1-dioxyde als elastase- inhibitoren

Info

Publication number: ATE154347T1
Authority: AT; Austria
Prior art keywords: benzisothiazolinone; compositions; dioxyde; chem; cosmetic
Prior art date: 1990-03-08

Application number

AT91301895T

Other languages

English (en)

Inventor

Ladislas Robert

Elemer Moczar

William Georges Hornebeck

Christiane Marie-Pierr Kerneur

Original Assignee

Unilever Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-03-08

Filing date

1991-03-07

Publication date

1997-06-15

1991-03-07 Application filed by Unilever Nv filed Critical Unilever Nv

1997-06-15 Application granted granted Critical

1997-06-15 Publication of ATE154347T1 publication Critical patent/ATE154347T1/de

Links

239000003602 elastase inhibitor Substances 0.000 title 1
239000000203 mixture Substances 0.000 abstract 3
102000016387 Pancreatic elastase Human genes 0.000 abstract 2
108010067372 Pancreatic elastase Proteins 0.000 abstract 2
239000002537 cosmetic Substances 0.000 abstract 2
239000004480 active ingredient Substances 0.000 abstract 1
125000001931 aliphatic group Chemical group 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
230000002209 hydrophobic effect Effects 0.000 abstract 1
230000001527 leucocytic effect Effects 0.000 abstract 1
229920006395 saturated elastomer Polymers 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
- C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
- A61K2800/74—Biological properties of particular ingredients
- A61K2800/78—Enzyme modulators, e.g. Enzyme agonists
- A61K2800/782—Enzyme inhibitors; Enzyme antagonists
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/08—Anti-ageing preparations
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q5/00—Preparations for care of the hair

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Dermatology (AREA)
Epidemiology (AREA)
Birds (AREA)
Chemical Kinetics & Catalysis (AREA)
Gerontology & Geriatric Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cosmetics (AREA)
Medicines Containing Plant Substances (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Enzymes And Modification Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Thiazole And Isothizaole Compounds (AREA)

AT91301895T 1990-03-08 1991-03-07 Benzisothiazolinon-1-dioxyde als elastase- inhibitoren ATE154347T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR9002951A FR2659327A1 (fr)	1990-03-08	1990-03-08	Derives du benzisothiazolinone-1-dioxyde, utilisables comme inhibiteurs des elastases.

Publications (1)

Publication Number	Publication Date
ATE154347T1 true ATE154347T1 (de)	1997-06-15

Family

ID=9394523

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT91301895T ATE154347T1 (de)	1990-03-08	1991-03-07	Benzisothiazolinon-1-dioxyde als elastase- inhibitoren

Country Status (16)

Country	Link
US (2)	US5338747A (de)
EP (1)	EP0446047B1 (de)
JP (1)	JPH04234863A (de)
KR (1)	KR960014782B1 (de)
AT (1)	ATE154347T1 (de)
AU (1)	AU636013B2 (de)
BR (1)	BR9100938A (de)
CA (1)	CA2037665A1 (de)
DE (1)	DE69126460T2 (de)
ES (1)	ES2102994T3 (de)
FR (1)	FR2659327A1 (de)
ID (1)	ID820B (de)
IN (1)	IN172035B (de)
MY (1)	MY106067A (de)
TW (1)	TW200472B (de)
ZA (1)	ZA911728B (de)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5512589A (en) *	1990-11-01	1996-04-30	Sterling Winthrop Inc.	2-saccharinylmethyl aryl carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof
US5306818A (en) *	1990-11-01	1994-04-26	Sterling Winthrop Inc.	Tetrahydro 2-saccharinylmerthyl aryl carboxylates
US5250696A (en) *	1990-11-01	1993-10-05	Sterling Winthrop Inc.	2-saccharinylmethyl aryl carboxylate
AU653279B2 (en) *	1991-12-30	1994-09-22	Sanofi	Novel 2-saccharinylmethyl heterocyclic carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof
TW226016B (de) *	1991-12-30	1994-07-01	Sterling Winthrop Inc
US6375948B1 (en) *	1999-07-12	2002-04-23	Kao Corporation	Treating method for suppressing hair growth
GB0129987D0 (en) *	2001-12-14	2002-02-06	Zylepsis Ltd	Skin compositions
US7361767B2 (en)	2003-11-14	2008-04-22	3M Innovative Properties Company	N-sulfonyldicarboximide containing tethering compounds
US7943388B2 (en)	2003-11-14	2011-05-17	3M Innovative Properties Company	Acoustic sensors and methods
US7169933B2 (en)	2003-11-14	2007-01-30	3M Innovative Properties Company	N-sulfonylaminocarbonyl containing compounds
US7423155B2 (en)	2003-11-14	2008-09-09	3M Innovative Properties Company	N-sulfonyldicarboximide containing tethering compounds
US7179923B2 (en)	2003-11-14	2007-02-20	3M Innovative Properties Company	N-sulfonylaminocarbonyl containing compounds
US7402678B2 (en)	2004-12-17	2008-07-22	3M Innovative Properties Company	Multifunctional amine capture agents
US7342082B2 (en)	2004-12-17	2008-03-11	3M Innovative Properties Company	Soluble polymers as amine capture agents and methods
EP1699768B1 (de) *	2003-12-30	2014-09-24	3M Innovative Properties Company	Multifunktionelle amin-capture-mittel
US7544754B2 (en) *	2005-09-30	2009-06-09	3M Innovative Properties Company	Crosslinked polymers with amine binding groups
US7544756B2 (en)	2005-09-30	2009-06-09	3M Innovative Properties Company	Crosslinked polymers with amine binding groups
US7544755B2 (en)	2005-09-30	2009-06-09	3M Innovative Properties Company	Crosslinked polymers with amine binding groups
US8034448B2 (en) *	2008-08-19	2011-10-11	Los Alamos National Security, Llc	Fibrous composites comprising carbon nanotubes and silica
ES2534193T3 (es)	2009-12-01	2015-04-20	Lubrizol Advanced Materials, Inc.	Polímeros hidrolíticamente estables para múltiples fines
EP3509588B1 (de)	2016-09-12	2023-06-07	Integral Health,Inc.	Bicyclische verbindungen verwendbar als gpr120-modulatoren
US10800773B2 (en)	2016-09-12	2020-10-13	Integral Health, Inc.	Monocyclic compounds useful as GPR120 modulators

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4195023A (en) *	1975-08-20	1980-03-25	Merck & Co., Inc.	2-(2-Furoyl)1,2-benzisothiazole-3-one, 2-(2-furoyl) saccharin, and 2-(2-thenoyl) saccharin
US4276298A (en) *	1978-03-24	1981-06-30	Merck & Co., Inc.	2-Aryl-1,2-benzisothiazolinone-1,1-dioxides and their use as selective protease inhibitors
FR2546164B1 (fr) *	1983-05-16	1987-07-17	Centre Nat Rech Scient	Nouveaux derives de peptides, leur preparation et leur application comme inhibiteurs de l'elastase

1990
- 1990-03-08 FR FR9002951A patent/FR2659327A1/fr active Pending
1991
- 1991-03-06 AU AU72635/91A patent/AU636013B2/en not_active Ceased
- 1991-03-06 CA CA002037665A patent/CA2037665A1/en not_active Abandoned
- 1991-03-07 AT AT91301895T patent/ATE154347T1/de not_active IP Right Cessation
- 1991-03-07 MY MYPI91000361A patent/MY106067A/en unknown
- 1991-03-07 ES ES91301895T patent/ES2102994T3/es not_active Expired - Lifetime
- 1991-03-07 DE DE69126460T patent/DE69126460T2/de not_active Expired - Fee Related
- 1991-03-07 EP EP91301895A patent/EP0446047B1/de not_active Expired - Lifetime
- 1991-03-07 US US07/666,093 patent/US5338747A/en not_active Expired - Fee Related
- 1991-03-08 KR KR91003708A patent/KR960014782B1/ko active IP Right Grant
- 1991-03-08 IN IN69/BOM/91A patent/IN172035B/en unknown
- 1991-03-08 BR BR919100938A patent/BR9100938A/pt not_active Application Discontinuation
- 1991-03-08 ZA ZA911728A patent/ZA911728B/xx unknown
- 1991-03-08 JP JP3125607A patent/JPH04234863A/ja active Pending
- 1991-04-13 TW TW080102851A patent/TW200472B/zh active
1992
- 1992-01-29 ID IDP185092A patent/ID820B/id unknown
1994
- 1994-04-19 US US08/230,048 patent/US5411978A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
DE69126460T2 (de)	1997-12-04
MY106067A (en)	1995-03-31
EP0446047B1 (de)	1997-06-11
JPH04234863A (ja)	1992-08-24
AU636013B2 (en)	1993-04-08
KR960014782B1 (en)	1996-10-19
FR2659327A1 (fr)	1991-09-13
US5338747A (en)	1994-08-16
DE69126460D1 (de)	1997-07-17
ZA911728B (en)	1992-11-25
US5411978A (en)	1995-05-02
KR910016330A (ko)	1991-11-05
BR9100938A (pt)	1991-11-05
IN172035B (de)	1993-03-20
EP0446047A1 (de)	1991-09-11
TW200472B (de)	1993-02-21
AU7263591A (en)	1991-09-12
ID820B (id)	1996-07-22
CA2037665A1 (en)	1991-09-09
ES2102994T3 (es)	1997-08-16

Legal Events

Date	Code	Title	Description
1997-12-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
DE69126460D1 (de)	1997-07-17	Benzisothiazolinon-1-dioxyde als Elastase-Inhibitoren
ATE164588T1 (de)	1998-04-15	Triterpenderivat
DE69212921D1 (de)	1996-09-26	Sonnenschutzmittel
FI932390A0 (fi)	1993-05-26	Nya hydroxiaminsyra- och N-hydroxiureaderivat samt deras anvaendning
SE8804036L (sv)	1989-05-10	Ny anvaendning av 11,28-dioxa-4-azatricklo (22.3.1.04.9)-oktakos-18-en-derivat och farmaceutiska kompositioner innehaallande desamma
ATE321543T1 (de)	2006-04-15	Pharmazeutische zusammensetzungen mit hydroximsäurederivaten
DE69716810T2 (de)	2003-02-27	2,3-Disubstituierte-(5,6)-heteroarylkondensierte-pyrimidin-4-one
FI920023A0 (fi)	1992-01-03	Heteroarylpiperazinfoereningar som antipsykotiska aemnen.
ATE251443T1 (de)	2003-10-15	Antimikrobielle kosmetische präparate
FI930974A0 (fi)	1993-03-04	Substituerade aminofosfonatderivat, foerfarande foer framstaellning av desamma och farmaceutiska kompositioner innehaollande desamma
YU48329B (sh)	1998-05-15	Antinflamatorne hidroksamske kiseline i n-hidroksikarbamidi
SE8404065D0 (sv)	1984-08-10	Novel biologically active compounds
SE8600658D0 (sv)	1986-02-14	Novel composition of matter
ES2075272T3 (es)	1995-10-01	Composicion dermatologica conteniendo acido cis-urocanico.
ATE110714T1 (de)	1994-09-15	Derivate von hydroxaminsäure die lipoxygenase hemmen.
MX9305523A (es)	1994-04-29	Composiciones quimoterapeuticas mejoradas frente a infecciones microbianas en peces, la reparacion y uso de las mismas.
ATE103890T1 (de)	1994-04-15	Neue acylaminosaeurederivate enthaltende arzneimittel und diaetetika.
DE68922596T2 (de)	1995-09-28	3-(3-Ethyl-1,2,4-oxadiazol-5-yl)-1-azabicycloheptan, Verfahren zu seiner Herstellung und dieses enthaltende pharmazeutische Zubereitungen.
SE9201188L (sv)	1993-10-15	Ny användning
PT986390E (pt)	2003-01-31	Composicoes farmaceuticas que contem cicloridrato de cinchonina