AR231636A1 - Procedimiento para la elaboracion de nuevos derivados de 5-alquilo-benzimidazol-2-sustituidos - Google Patents

Procedimiento para la elaboracion de nuevos derivados de 5-alquilo-benzimidazol-2-sustituidos

Info

Publication number: AR231636A1
Authority: AR; Argentina
Prior art keywords: elaboration; benzimidazole; substituted; alkyl; procedure
Prior art date: 1977-08-01

Application number

AR278849A

Other languages

English (en)

Original Assignee

Ciba Geigy Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-08-01

Filing date

1979-11-12

Publication date

1985-01-31

1977-08-01 Priority claimed from HU77CI1761A external-priority patent/HU180700B/hu

1979-11-12 Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag

1985-01-31 Application granted granted Critical

1985-01-31 Publication of AR231636A1 publication Critical patent/AR231636A1/es

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/45—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by at least one doubly—bound oxygen atom, not being part of a —CHO group
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
- C07C45/46—Friedel-Crafts reactions
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/12—Radicals substituted by oxygen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pulmonology (AREA)
Immunology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

AR278849A 1977-08-01 1979-11-12 Procedimiento para la elaboracion de nuevos derivados de 5-alquilo-benzimidazol-2-sustituidos AR231636A1 (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
HU77CI1761A HU180700B (en)	1976-08-27	1977-08-01	Process for producing acylized benzimidasole derivatives
CH209478		1978-02-27

Publications (1)

Publication Number	Publication Date
AR231636A1 true AR231636A1 (es)	1985-01-31

Family

ID=25689497

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
AR273145A AR227125A1 (es)	1977-08-01	1978-07-31	Procedimiento para la elaboracion de nuevos derivados de benzimidazol y sus sales
AR278851A AR228023A1 (es)	1977-08-01	1979-11-12	Procedimiento para la elaboracion de nuevos compuestos derivados del 5-alquil-2-carboxi o 2-hidroximetil-benzimidazol y sus sales
AR278853A AR223196A1 (es)	1977-08-01	1979-11-12	Procedimiento para la elaboracion de nuevos derivados de 2-hidroximetil-5,6-dialquil(c1-c4)-benzimidazol
AR278849A AR231636A1 (es)	1977-08-01	1979-11-12	Procedimiento para la elaboracion de nuevos derivados de 5-alquilo-benzimidazol-2-sustituidos

Family Applications Before (3)

Application Number	Title	Priority Date	Filing Date
AR273145A AR227125A1 (es)	1977-08-01	1978-07-31	Procedimiento para la elaboracion de nuevos derivados de benzimidazol y sus sales
AR278851A AR228023A1 (es)	1977-08-01	1979-11-12	Procedimiento para la elaboracion de nuevos compuestos derivados del 5-alquil-2-carboxi o 2-hidroximetil-benzimidazol y sus sales
AR278853A AR223196A1 (es)	1977-08-01	1979-11-12	Procedimiento para la elaboracion de nuevos derivados de 2-hidroximetil-5,6-dialquil(c1-c4)-benzimidazol

Country Status (19)

Country	Link
US (1)	US4323688A (es)
EP (1)	EP0000574B1 (es)
JP (1)	JPS5427565A (es)
AR (4)	AR227125A1 (es)
AT (1)	AT364830B (es)
AU (1)	AU523324B2 (es)
CA (1)	CA1109072A (es)
DD (1)	DD138318A5 (es)
DE (1)	DE2861987D1 (es)
DK (1)	DK339578A (es)
ES (1)	ES472208A1 (es)
FI (1)	FI68231C (es)
GR (1)	GR77614B (es)
IE (1)	IE47285B1 (es)
IL (1)	IL55253A (es)
NO (1)	NO150082C (es)
NZ (1)	NZ188006A (es)
PL (1)	PL208772A1 (es)
PT (1)	PT68365A (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0000574B1 (de) *	1977-08-01	1982-08-04	Ciba-Geigy Ag	Benzimidazol-2-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung zur Herstellung von Arzneimitteln
US4322431A (en) *	1979-02-09	1982-03-30	Ciba-Geigy Corporation	Pharmaceutical preparations containing benzimidazole 2-derivatives
US4368201A (en) *	1981-07-20	1983-01-11	Usv Pharmaceutical Corporation	Tetrahydronaphthoxazoles

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB243766A (en) *	1924-12-01	1926-07-29	Bayer Ag	Process for the manufacture of benzimidazoles
US2053822A (en) *	1933-12-15	1936-09-08	Soc Of Chemical Ind	Alkylated imidazoles of high molecular weight and process of making same
GB766749A (en)	1954-01-11	1957-01-23	Aschaffenburger Zellstoffwerke	Benzimidazole cobalamines and process for their preparation and separation
US2876233A (en) *	1956-10-29	1959-03-03	Gruenenthal Chemie	1-(p-halobenzyl)-2-methyl benzimidazoles and salts
CH356461A (de) *	1956-10-30	1961-08-31	Gruenenthal Chemie	Verfahren zur Herstellung von neuen Derivaten des Benzimidazols
CH356460A (de) *	1956-10-30	1961-08-31	Gruenenthal Chemie	Verfahren zur Herstellung von neuen Derivaten des Benzimidazols
CH362411A (de) *	1956-10-30	1962-06-15	Gruenenthal Chemie	Verfahren zur Herstellung von neuen Derivaten des Benzimidazols
US3325271A (en) *	1963-07-17	1967-06-13	United States Borax Chem	Herbicidal composition and method employing substituted benzimidazoles
US3318889A (en) *	1963-10-14	1967-05-09	S B Penick & Company	2-benzimidazole carbamates
DE2014293A1 (de) *	1969-03-29	1970-10-08	Fisons Ltd., Felixstowe, Suffolk (Grossbritannien)	Substituierte Benzimidazole und Verfahren zu ihrer Herstellung und Verwendung
CH528514A (de) *	1969-05-22	1972-09-30	Bayer Ag	Verfahren zur Herstellung von Acylimidazolen
US3661925A (en) *	1970-05-15	1972-05-09	American Home Prod	Process for the preparation of 2-benzimidazolecarboxamides
FR2115067B1 (es) *	1970-11-27	1974-03-22	Delalande Sa
EP0000574B1 (de) *	1977-08-01	1982-08-04	Ciba-Geigy Ag	Benzimidazol-2-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung zur Herstellung von Arzneimitteln

1978
- 1978-07-24 EP EP78100489A patent/EP0000574B1/de not_active Expired
- 1978-07-24 DE DE7878100489T patent/DE2861987D1/de not_active Expired
- 1978-07-27 US US05/928,632 patent/US4323688A/en not_active Expired - Lifetime
- 1978-07-27 GR GR56880A patent/GR77614B/el unknown
- 1978-07-28 DD DD78207009A patent/DD138318A5/xx unknown
- 1978-07-28 CA CA308,351A patent/CA1109072A/en not_active Expired
- 1978-07-28 FI FI782348A patent/FI68231C/fi not_active IP Right Cessation
- 1978-07-31 ES ES472208A patent/ES472208A1/es not_active Expired
- 1978-07-31 DK DK339578A patent/DK339578A/da not_active Application Discontinuation
- 1978-07-31 NZ NZ188006A patent/NZ188006A/xx unknown
- 1978-07-31 AU AU38478/78A patent/AU523324B2/en not_active Expired
- 1978-07-31 IL IL55253A patent/IL55253A/xx unknown
- 1978-07-31 NO NO782615A patent/NO150082C/no unknown
- 1978-07-31 PT PT68365A patent/PT68365A/pt unknown
- 1978-07-31 AR AR273145A patent/AR227125A1/es active
- 1978-07-31 IE IE1545/78A patent/IE47285B1/en unknown
- 1978-07-31 AT AT0553978A patent/AT364830B/de not_active IP Right Cessation
- 1978-08-01 PL PL20877278A patent/PL208772A1/xx unknown
- 1978-08-01 JP JP9322478A patent/JPS5427565A/ja active Pending
1979
- 1979-11-12 AR AR278851A patent/AR228023A1/es active
- 1979-11-12 AR AR278853A patent/AR223196A1/es active
- 1979-11-12 AR AR278849A patent/AR231636A1/es active

Also Published As

Publication number	Publication date
PT68365A (de)	1978-08-01
ATA553978A (de)	1981-04-15
IL55253A0 (en)	1978-09-29
IE781545L (en)	1979-02-01
AR223196A1 (es)	1981-07-31
DE2861987D1 (en)	1982-09-30
EP0000574B1 (de)	1982-08-04
AU3847878A (en)	1980-02-07
US4323688A (en)	1982-04-06
FI782348A (fi)	1979-02-02
DK339578A (da)	1979-02-02
EP0000574A1 (de)	1979-02-07
ES472208A1 (es)	1979-03-16
NO150082C (no)	1984-08-15
IL55253A (en)	1982-04-30
AR227125A1 (es)	1982-09-30
PL208772A1 (pl)	1979-06-04
DD138318A5 (de)	1979-10-24
NZ188006A (en)	1981-11-19
AU523324B2 (en)	1982-07-22
AT364830B (de)	1981-11-25
NO782615L (no)	1979-02-02
CA1109072A (en)	1981-09-15
FI68231C (fi)	1985-08-12
IE47285B1 (en)	1984-02-08
FI68231B (fi)	1985-04-30
JPS5427565A (en)	1979-03-01
NO150082B (no)	1984-05-07
AR228023A1 (es)	1983-01-14
GR77614B (es)	1984-09-25

Publication	Publication Date	Title
MX5950E (es)	1984-09-06	Procedimiento para la preparacion de derivados de la pirrolidin-2-ona
MX5527E (es)	1983-09-23	Procedimiento para la preparacion de derivados de carboestirilo
AR220704A1 (es)	1980-11-28	Procedimiento para la preparacion de derivados de indanil y tetrahidronaftil octatrieno
AR220216A1 (es)	1980-10-15	Procedimiento para la preparacion de 1-(2-hidroxi-3-amino-propil sustituido)-2-nitroimidazoles
MX4988E (es)	1983-01-31	Procedimiento para la preparacion de derivados pirrolidinicos
AR221851A1 (es)	1981-03-31	Procedimiento para la preparacion de derivados de 4-piperidino-6,7-dialcoxi-quinazolina
AR224110A1 (es)	1981-10-30	Procedimiento para la preparacion de derivados de 5(6)-benzimidazoles
MX5479E (es)	1983-08-19	Procedimiento para la preparacion de derivados de 1-oxadetiacefalosporinas
MX5215E (es)	1983-04-25	Procedimiento de preparacion de derivados de tienopiridina
AR218296A1 (es)	1980-05-30	Procedimiento para la preparacion de nuevos derivados de 14-beta-amino-morfina
AR223656A1 (es)	1981-09-15	Procedimiento para obtener derivados de 2-feniliminoimidazolidina
AR222844A1 (es)	1981-06-30	Procedimiento para la obtencion de nuevos derivados de n1-glucofuranosil-6-ilo-n3-nitroso-ureas
AR225889A1 (es)	1982-05-14	Procedimiento para la elaboracion de acidos heterociclilcarboxilicos acilados
AR227866A1 (es)	1982-12-30	Procedimiento para la elaboracion de compuestos de ditienilalquilaminas
AR220730A1 (es)	1980-11-28	Procedimiento para la preparacion de nuevos derivados de la i-((benzoxatiolil)-metil)-4-heterociclil-piperazina
MX4884E (es)	1982-12-02	Procedimiento para la preparacion de derivados de la tienopiridina
AR221215A1 (es)	1981-01-15	Procedimiento para la preparacion de cloroacetanilidas substituidas
AR223465A1 (es)	1981-08-31	Procedimiento para obtener derivados de 5-bencil-2,4-diamino-pirimidinas
AR223319A1 (es)	1981-08-14	Procedimiento para la elaboracion de compuestos de 6-amino-penam
AR218933A1 (es)	1980-07-15	Procedimiento para obtener derivados de oxazolidona-2
MX147497A (es)	1982-12-10	Procedimiento para la elaboracion de hojas combinadas
AR230835A1 (es)	1984-07-31	Procedimiento para la obtencion de derivados de 2,1,3-tiadiazin-4-ona-2,2-dioxido
AR231636A1 (es)	1985-01-31	Procedimiento para la elaboracion de nuevos derivados de 5-alquilo-benzimidazol-2-sustituidos
AR222011A1 (es)	1981-04-15	Procedimiento para la preparacion de compuestos de 2-hidroxibenzotiazol
ES487954A0 (es)	1980-12-16	Procedimiento para la obtencion de derivados de la rifamici-na-s