AR228621A1 - Procedimiento de preparacion de derivados de acido n-(mercapto o carboxialquilamino)-azabiclico-octano-3-carboxilico - Google Patents

Procedimiento de preparacion de derivados de acido n-(mercapto o carboxialquilamino)-azabiclico-octano-3-carboxilico

Info

Publication number: AR228621A1
Authority: AR; Argentina
Prior art keywords: carboxialquilamino; azabiclico; carboxilico; octano; mercapto
Prior art date: 1980-10-21

Application number

AR287128A

Other languages

English (en)

Original Assignee

Science Union & Cie

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1980-10-21

Filing date

1981-10-19

Publication date

1983-03-30

1981-10-19 Application filed by Science Union & Cie filed Critical Science Union & Cie

1983-03-30 Application granted granted Critical

1983-03-30 Publication of AR228621A1 publication Critical patent/AR228621A1/es

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D223/32—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems containing carbocyclic rings other than six-membered
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/06—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing isoquinuclidine ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Biochemistry (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

AR287128A 1980-10-21 1981-10-19 Procedimiento de preparacion de derivados de acido n-(mercapto o carboxialquilamino)-azabiclico-octano-3-carboxilico AR228621A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR8022438A FR2492381A1 (fr)	1980-10-21	1980-10-21	Nouveaux acides aza bicyclo alcane carboxyliques substitues leurs procedes de preparation et leur emploi comme inhibiteur d'enzyme

Publications (1)

Publication Number	Publication Date
AR228621A1 true AR228621A1 (es)	1983-03-30

Family

ID=9247120

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AR287128A AR228621A1 (es)	1980-10-21	1981-10-19	Procedimiento de preparacion de derivados de acido n-(mercapto o carboxialquilamino)-azabiclico-octano-3-carboxilico

Country Status (29)

Country	Link
US (1)	US4397857A (es)
EP (1)	EP0051020B1 (es)
JP (2)	JPS5798281A (es)
KR (1)	KR860001877B1 (es)
AR (1)	AR228621A1 (es)
AT (1)	ATE8892T1 (es)
AU (1)	AU540609B2 (es)
CA (1)	CA1183140A (es)
DD (1)	DD201891A5 (es)
DE (1)	DE3165428D1 (es)
DK (1)	DK162444C (es)
EG (1)	EG15419A (es)
ES (1)	ES8301927A1 (es)
FI (1)	FI73678C (es)
FR (2)	FR2492381A1 (es)
GR (1)	GR75389B (es)
HU (1)	HU185058B (es)
IE (1)	IE51823B1 (es)
IL (1)	IL64075A0 (es)
MA (1)	MA19307A1 (es)
MX (1)	MX155032A (es)
NO (1)	NO155098C (es)
NZ (1)	NZ198701A (es)
OA (1)	OA06930A (es)
PH (1)	PH17338A (es)
PT (1)	PT73857B (es)
SU (1)	SU1138022A3 (es)
YU (1)	YU42587B (es)
ZA (1)	ZA817251B (es)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ATE20469T1 (de) *	1980-10-23	1986-07-15	Schering Corp	Carboxyalkyl-dipeptide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel.
IE54551B1 (en) *	1982-01-22	1989-11-22	Ici Plc	Amide derivatives
DE3227055A1 (de) *	1982-07-20	1984-01-26	Hoechst Ag, 6230 Frankfurt	Neue derivate der 2-aza-bicyclo(2.2.2)octan-3-carbonsaeure, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung sowie 2-aza-bicyclo(2.2.2)octan-3-carbonsaeure als zwischenstufe und verfahren zu deren herstellung
DE3246757A1 (de) *	1982-12-17	1984-06-20	Hoechst Ag, 6230 Frankfurt	Neue 2-azabicyclo(2.2.1)heptan-derivate, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung sowie 2-azabicyclo(2.2.1)heptan-derivate als zwischenprodukte und verfahren zu deren herstellung
DE3303344A1 (de)	1983-02-02	1984-08-02	Hoechst Ag, 6230 Frankfurt	Verfahren zur herstellung von n-alkylierten aminosaeuren und deren estern
US4693996A (en) *	1985-12-23	1987-09-15	Warner-Lambert Company	Method of treating heart failure and medicaments therefor
DE3707911C1 (de) *	1987-03-12	1988-03-31	Texaco Ag	Bicyclische Aminkatalysatoren
FR2619813B1 (fr) *	1987-08-28	1991-05-03	Adir	Nouveaux derives de l'acide aza - 2 bicyclooctane carboxylique - 3, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent
FR2635684A1 (fr) *	1988-08-24	1990-03-02	Adir	Utilisation de derives de l'acide aza - 2 bicyclooctane (2.2.2) carboxylique - 3 pour l'obtention de medicaments destines au traitement des maladies consecutives a l'alteration de la paroi vasculaire ainsi qu'aux troubles de la microcirculation
JPH0426348U (es) *	1990-06-25	1992-03-02
TW197945B (es) *	1990-11-27	1993-01-11	Hoechst Ag
LT3872B (en)	1993-12-06	1996-04-25	Hoechst Ag	Novel peptides and pharmaceutical compositions containing them
EP0796855B1 (de)	1996-03-20	2002-02-06	Hoechst Aktiengesellschaft	Inhibitoren der Knochenresorption und Vitronectinrezeptor-Antagonisten
FR2746394B1 (fr)	1996-03-20	1998-05-29	Roussel Uclaf	Nouveaux composes tricycliques, leur procede de preparation, et les intermediaires de ce procede, leur application a titre de medicaments et les compositions pharmaceutiques les renfermant
DE19653647A1 (de)	1996-12-20	1998-06-25	Hoechst Ag	Vitronectin - Rezeptorantagonisten, deren Herstellung sowie deren Verwendung
DE19821483A1 (de)	1998-05-14	1999-11-18	Hoechst Marion Roussel De Gmbh	Imidazolidinderivate, ihre Herstellung, ihre Verwendung und sie enthaltende pharmazeutische Präparate
US7001911B2 (en)	2000-06-28	2006-02-21	Bristol-Myers Squibb Company	Fused cyclic modulators of nuclear hormone receptor function
IL152719A0 (en) *	2000-06-28	2003-06-24	Bristol Myers Squibb Co	Selective androgen receptor modulators and methods for their identification
US20040077605A1 (en) *	2001-06-20	2004-04-22	Salvati Mark E.	Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
US6953679B2 (en)	2000-09-19	2005-10-11	Bristol-Myers Squibb Company	Method for the preparation of fused heterocyclic succinimide compounds and analogs thereof
EP1854798A3 (en) *	2000-09-19	2007-11-28	Bristol-Myers Squibb Company	Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
US20040087548A1 (en)	2001-02-27	2004-05-06	Salvati Mark E.	Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
AU2002364082A1 (en) *	2001-12-19	2003-07-09	Bristol-Myers Squibb Company	Fused heterocyclic compounds and analogs thereof: modulators of nuclear hormone receptor function

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE94175C (es) *
GB1095105A (en) *	1965-04-12	1967-12-13	Scherico Ltd	Novel n-(phenyl-sulfonyl)-isoquinuclidine-carboxamides
US3740408A (en) *	1967-09-11	1973-06-19	Upjohn Co	Oxygenated 3-aza bicyclo(3,3,1)nonanes
IE52663B1 (en) *	1980-04-02	1988-01-20	Warner Lambert Co	Substituted acyl derivatives of octahydro-1h-indole-2-carboxylic acids

1980
- 1980-10-21 FR FR8022438A patent/FR2492381A1/fr active Granted
1981
- 1981-10-06 MX MX8571A patent/MX155032A/es unknown
- 1981-10-13 YU YU2454/81A patent/YU42587B/xx unknown
- 1981-10-13 ES ES506222A patent/ES8301927A1/es not_active Expired
- 1981-10-19 IL IL64075A patent/IL64075A0/xx not_active IP Right Cessation
- 1981-10-19 AR AR287128A patent/AR228621A1/es active
- 1981-10-19 DK DK460181A patent/DK162444C/da not_active IP Right Cessation
- 1981-10-20 CA CA000388374A patent/CA1183140A/fr not_active Expired
- 1981-10-20 ZA ZA817251A patent/ZA817251B/xx unknown
- 1981-10-20 EG EG81609A patent/EG15419A/xx active
- 1981-10-20 AT AT81401642T patent/ATE8892T1/de active
- 1981-10-20 GR GR66308A patent/GR75389B/el unknown
- 1981-10-20 AU AU76624/81A patent/AU540609B2/en not_active Ceased
- 1981-10-20 SU SU813346599A patent/SU1138022A3/ru active
- 1981-10-20 NZ NZ198701A patent/NZ198701A/en unknown
- 1981-10-20 DD DD81234232A patent/DD201891A5/de not_active IP Right Cessation
- 1981-10-20 NO NO813541A patent/NO155098C/no unknown
- 1981-10-20 EP EP81401642A patent/EP0051020B1/fr not_active Expired
- 1981-10-20 PH PH26368A patent/PH17338A/en unknown
- 1981-10-20 PT PT73857A patent/PT73857B/pt not_active IP Right Cessation
- 1981-10-20 DE DE8181401642T patent/DE3165428D1/de not_active Expired
- 1981-10-20 IE IE2460/81A patent/IE51823B1/en not_active IP Right Cessation
- 1981-10-20 MA MA19509A patent/MA19307A1/fr unknown
- 1981-10-20 US US06/313,184 patent/US4397857A/en not_active Expired - Lifetime
- 1981-10-20 FI FI813279A patent/FI73678C/fi not_active IP Right Cessation
- 1981-10-21 JP JP56168516A patent/JPS5798281A/ja active Granted
- 1981-10-21 HU HU813066A patent/HU185058B/hu not_active IP Right Cessation
- 1981-10-21 KR KR1019810004015A patent/KR860001877B1/ko not_active IP Right Cessation
- 1981-10-21 OA OA57525A patent/OA06930A/xx unknown
1982
- 1982-04-22 FR FR8206899A patent/FR2525604B2/fr not_active Expired
1985
- 1985-11-12 JP JP60252137A patent/JPS61126025A/ja active Granted

Also Published As

Publication number	Publication date
DD201891A5 (de)	1983-08-17
MX155032A (es)	1988-01-21
US4397857A (en)	1983-08-09
DK460181A (da)	1982-04-22
IL64075A0 (en)	1982-01-31
NO155098C (no)	1987-02-11
ATE8892T1 (de)	1984-08-15
FR2525604A2 (fr)	1983-10-28
AU7662481A (en)	1982-04-29
HU185058B (en)	1984-11-28
DK162444B (da)	1991-10-28
FI813279L (fi)	1982-04-22
JPS6146453B2 (es)	1986-10-14
FR2525604B2 (fr)	1985-06-07
NO155098B (no)	1986-11-03
KR830007570A (ko)	1983-10-21
NO813541L (no)	1982-04-22
PH17338A (en)	1984-08-01
JPS61126025A (ja)	1986-06-13
KR860001877B1 (ko)	1986-10-24
EP0051020A1 (fr)	1982-05-05
YU245481A (en)	1984-04-30
PT73857B (fr)	1983-01-25
EP0051020B1 (fr)	1984-08-08
JPS6112911B2 (es)	1986-04-10
DE3165428D1 (en)	1984-09-13
GR75389B (es)	1984-07-13
EG15419A (en)	1986-03-31
PT73857A (fr)	1981-11-01
ES506222A0 (es)	1983-01-01
IE812460L (en)	1982-04-21
FI73678C (fi)	1987-11-09
CA1183140A (fr)	1985-02-26
IE51823B1 (en)	1987-04-01
FR2492381B1 (es)	1983-08-12
SU1138022A3 (ru)	1985-01-30
AU540609B2 (en)	1984-11-29
FI73678B (fi)	1987-07-31
OA06930A (fr)	1983-05-31
ZA817251B (en)	1982-09-29
DK162444C (da)	1992-03-23
JPS5798281A (en)	1982-06-18
YU42587B (en)	1988-10-31
MA19307A1 (fr)	1982-07-01
ES8301927A1 (es)	1983-01-01
NZ198701A (en)	1984-07-06
FR2492381A1 (fr)	1982-04-23

Publication	Publication Date	Title
AR228621A1 (es)	1983-03-30	Procedimiento de preparacion de derivados de acido n-(mercapto o carboxialquilamino)-azabiclico-octano-3-carboxilico
ES504955A0 (es)	1982-08-16	Procedimiento para la preparacion de derivados de aminoacidos
RO86825A (ro)	1985-05-20	Procedeu pentru prepararea unor acizi 7-amino-3-metil-substituit -dela 3-cefem-4-carbo0ilici
NO820287L (no)	1982-08-04	Fremgangsmaate for fremstilling av isocyanursyre-derivater
DK523579A (da)	1980-06-12	Fremgangsmaade til fremstilling af aminosyrederivater
DK372479A (da)	1980-03-08	Fremgangsmaade til fremstilling af aminosyrederivater
MX154685A (es)	1987-11-25	Procedimiento para la preparacion de derivados de urea
RO86213A (ro)	1985-03-15	Procedeu pentru prepararea izobutenei
ES498437A0 (es)	1981-11-01	Procedimiento para la preparacion de acido silicico de pre- cipitacion
AR225363A1 (es)	1982-03-15	Procedimiento para la preparacion de acido alfa-hidroxi-gamma-metilmercaptobutirico
MX7101E (es)	1987-06-24	Procedimiento para la preparacion de derivados de acido quinolin-carboxilico
DK536281A (da)	1982-07-11	Fremgangsmaade til fremstilling af carbonsyrederivater
ES495697A0 (es)	1981-12-16	Procedimiento para la obtencion de compuestos de acido di- glicidil-isocianurico n-sustituidos
DK34781A (da)	1981-07-29	Fremgangsmaade til fremstilling af phenylalkansyrederivater
AR231289A1 (es)	1984-10-31	Procedimiento para preparar derivados de quinolil-4-1-piperidilo-4-2-etanol o quinolil-4-1-piperidil-4-3-propanol
IT1150046B (it)	1986-12-10	Procedimento per la produzione di teatrafluoruro di zolfo
RO80112A (ro)	1982-10-26	Procedeu pentru prepararea de acid 1,1-dioxopenicilic
ES504753A0 (es)	1982-08-16	Procedimiento para la preparacion de imidas de acidos succi-nicos
ES522058A0 (es)	1984-12-01	Procedimiento de preparacion de derivados de acido carbacico.
MX6900E (es)	1986-10-10	Procedimiento para la preparacion de n-(halogenometil)acilamidas
NO802873L (no)	1981-10-09	Fremgangsmaate for fremstilling av en vandig opploesning av kalsiumnitritt
ES500959A0 (es)	1982-04-16	Procedimiento para la preparacion de derivados de cianoal- quil-fenilurea
AR229470A1 (es)	1983-08-31	Procedimiento de preparacion de piridilalquil tio-esteres de acido 1-p-clorobenzoil-5-metoxi-2-metil-indol-3-acetico
DK267880A (da)	1980-12-26	Fremgangsmaade til fremstilling af acylaminobenzoesyrederivater
ES504338A0 (es)	1982-06-01	Procedimiento de preparacion de derivados difeniletericos