AR061165A1 - Formulaciones de liberacion pulsada de fenilefrina y composiciones farmaceuticas - Google Patents

Formulaciones de liberacion pulsada de fenilefrina y composiciones farmaceuticas

Info

Publication number
AR061165A1
AR061165A1 ARP070102383A ARP070102383A AR061165A1 AR 061165 A1 AR061165 A1 AR 061165A1 AR P070102383 A ARP070102383 A AR P070102383A AR P070102383 A ARP070102383 A AR P070102383A AR 061165 A1 AR061165 A1 AR 061165A1
Authority
AR
Argentina
Prior art keywords
phenylephrine
component
pharmaceutical composition
phenylefrine
formulations
Prior art date
Application number
ARP070102383A
Other languages
English (en)
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38582318&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR061165(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Publication of AR061165A1 publication Critical patent/AR061165A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/14Decongestants or antiallergics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente describe una formulacion de liberacion pulsada o una composicion farmacéutica que comprende fenilefrina. La composicion farmacéutica comprende un componente de liberacion inmediata y un componente con recubrimiento entérico formulados conjuntamente ya sea en forma solida o en una suspension. El componente de la cubierta entérica comprende microcristales sembrados con fenilefrina como componente activo y recubierto con una cubierta sensible al pH para retardar la liberacion de la fenilefrina. La composicion farmacéutica puede comprender además por lo menos un componente activo seleccionado del grupo que consiste en un antihistamínico, un analgésico, un antipirético, un anti-inflamatorio no esteroide y mezclas de dos o más de dichos componentes activos. Reivindicacion 20: Un método de preparacion de una composicion de acuerdo con la reivindicacion 2, que comprende mezclar microcristales con cubierta entérica que contienen fenilefrina, fenilefrina a granel y un líquido.
ARP070102383A 2006-06-01 2007-06-01 Formulaciones de liberacion pulsada de fenilefrina y composiciones farmaceuticas AR061165A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US81001806P 2006-06-01 2006-06-01

Publications (1)

Publication Number Publication Date
AR061165A1 true AR061165A1 (es) 2008-08-06

Family

ID=38582318

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP070102383A AR061165A1 (es) 2006-06-01 2007-06-01 Formulaciones de liberacion pulsada de fenilefrina y composiciones farmaceuticas

Country Status (15)

Country Link
US (1) US20070281019A1 (es)
EP (1) EP2029105A1 (es)
JP (1) JP2009538919A (es)
KR (1) KR20090015103A (es)
CN (1) CN101472561A (es)
AR (1) AR061165A1 (es)
AU (1) AU2007254819A1 (es)
CA (1) CA2653950A1 (es)
MX (1) MX2008015357A (es)
NO (1) NO20085416L (es)
PE (1) PE20080313A1 (es)
RU (1) RU2008151945A (es)
TW (1) TW200808376A (es)
WO (1) WO2007143156A1 (es)
ZA (1) ZA200810162B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8940796B2 (en) 2006-02-21 2015-01-27 Wyeth Llc Phenylephrine liquid formulations
US9005652B2 (en) 2006-07-25 2015-04-14 Wyeth Chewable tablet containing phenylephrine
EP2385823A4 (en) * 2009-01-09 2014-02-12 Panacea Biotec Ltd DOUBLE RELEASE PHARMACEUTICAL SUSPENSION
MX2009001925A (es) * 2009-02-20 2010-08-20 Senosiain S A De C V Lab Composicion farmaceutica oral para uso en enfermedades respiratorias.
BR112017005574A2 (pt) * 2014-09-19 2017-12-12 Procter & Gamble formas de dosagem de liberação pulsada de fenilefrina
US10278930B2 (en) 2017-03-16 2019-05-07 The Procter & Gamble Company Method for relieving sinus congestion
CN109875966B (zh) * 2019-04-09 2021-03-26 海南普利制药股份有限公司 地氯雷他定干混悬剂

Family Cites Families (41)

* Cited by examiner, † Cited by third party
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US3558768A (en) * 1969-12-19 1971-01-26 Sterling Drug Inc Sustained release pharmaceutical compositions
US4291015A (en) * 1979-08-14 1981-09-22 Key Pharmaceuticals, Inc. Polymeric diffusion matrix containing a vasodilator
US5025019A (en) * 1984-04-09 1991-06-18 Analgesic Associates Cough/cold mixtures comprising non-steroidal anti-inflammatory drugs
US4764378A (en) * 1986-02-10 1988-08-16 Zetachron, Inc. Buccal drug dosage form
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US4990535A (en) * 1989-05-03 1991-02-05 Schering Corporation Pharmaceutical composition comprising loratadine, ibuprofen and pseudoephedrine
US5133974A (en) * 1989-05-05 1992-07-28 Kv Pharmaceutical Company Extended release pharmaceutical formulations
DE69107461T2 (de) * 1990-08-07 1995-06-22 Pfizer Verwendung von interfacial polymerisierten membranen in abgabevorrichtungen.
US5518730A (en) * 1992-06-03 1996-05-21 Fuisz Technologies Ltd. Biodegradable controlled release flash flow melt-spun delivery system
US5458879A (en) * 1994-03-03 1995-10-17 The Procter & Gamble Company Oral vehicle compositions
US6160020A (en) * 1996-12-20 2000-12-12 Mcneill-Ppc, Inc. Alkali metal and alkaline-earth metal salts of acetaminophen
MX9701946A (es) * 1997-03-14 1998-04-30 Arturo Jimenez Bayardo Solucion oftalmica transportadora.
EP1021204B1 (en) * 1997-09-26 2005-12-28 Noven Pharmaceuticals, Inc. Bioadhesive compositions and methods for topical administration of active agents
US6602521B1 (en) * 1998-09-29 2003-08-05 Impax Pharmaceuticals, Inc. Multiplex drug delivery system suitable for oral administration
US6521254B2 (en) * 1998-12-07 2003-02-18 J-Med Pharmaceuticals, Inc. Single-dose antihistamine/decongestant formulations for treating rhinitis
CN1161112C (zh) * 1999-02-23 2004-08-11 株式会社柳韩洋行 含氯雷他定和伪麻黄碱的药物胶囊组合物
US6267986B1 (en) * 1999-09-24 2001-07-31 Ranbaxy Laboratories Limited Process for the preparation of a controlled drug delivery system containing pseudoephedrine and a long acting antihistamine
US6114346A (en) * 1999-10-22 2000-09-05 Schering Corporation Treating sleep disorders using desloratadine
AU2276801A (en) * 1999-12-20 2001-07-03 Schering Corporation Extended release oral dosage composition
WO2001045668A2 (en) * 1999-12-20 2001-06-28 Schering Corporation Stable extended release oral dosage composition comprising pseudoephedrine and desloratadine
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US8940796B2 (en) * 2006-02-21 2015-01-27 Wyeth Llc Phenylephrine liquid formulations
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US9005652B2 (en) * 2006-07-25 2015-04-14 Wyeth Chewable tablet containing phenylephrine
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Also Published As

Publication number Publication date
NO20085416L (no) 2008-12-30
TW200808376A (en) 2008-02-16
US20070281019A1 (en) 2007-12-06
EP2029105A1 (en) 2009-03-04
AU2007254819A1 (en) 2007-12-13
PE20080313A1 (es) 2008-04-10
ZA200810162B (en) 2009-11-25
JP2009538919A (ja) 2009-11-12
MX2008015357A (es) 2009-03-06
CN101472561A (zh) 2009-07-01
KR20090015103A (ko) 2009-02-11
RU2008151945A (ru) 2010-07-20
CA2653950A1 (en) 2007-12-13
WO2007143156A1 (en) 2007-12-13

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