AR057331A1 - Serin- amidas sustituidas con heteroaroilo - Google Patents

Serin- amidas sustituidas con heteroaroilo

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Publication number
AR057331A1
AR057331A1 ARP060102179A ARP060102179A AR057331A1 AR 057331 A1 AR057331 A1 AR 057331A1 AR P060102179 A ARP060102179 A AR P060102179A AR P060102179 A ARP060102179 A AR P060102179A AR 057331 A1 AR057331 A1 AR 057331A1
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Argentina
Prior art keywords
alkyl
alkoxy
amino
phenyl
aminocarbonyl
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ARP060102179A
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English (en)
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Basf Ag
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Publication of AR057331A1 publication Critical patent/AR057331A1/es

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/68Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Furan Compounds (AREA)

Abstract

Procedimientos y productos intermediarios para su preparacion, así como el uso de esos compuestos o agentes que contienen estos compuestos, para el combate de plantas no deseadas. Reivindicacion 1: Serin-amidas sustituidas con heteroaroílo, caracterizadas porque tienen la formula en donde las variables tienen los siguientes significados: A es heteroarilo de 5 o 6 miembros con uno a cuatro átomos de N, o con uno a tres átomos de N y un átomo de O o S, o con un átomo de O o S, que puede estar parcial o totalmente halogenado y/o que puede llevar 1 a 3 radicales del grupo ciano, alquilo C1-6, cicloalquilo C3-6, halogenoalquilo C1-6, alcoxi C1-6, halogenoalcoxi C1-6 y alcoxi C1-6-alquilo C1-4; R1, R2 es H, hidroxi o alcoxi C1-6; R3 es alquilo C1-6, cianoalquilo C1-4 o halogenoalquilo C1-6; R4 es H, alquilo C1-6, cicloalquilo C3-6, alquenilo C3-6, alquinilo C3-6, halogenalquenilo C3-6, halogenalquinilo C3-6, formilo, alquil C1-6-carbonilo, cicloalquilcarbonilo C3-6, alquenilcarbonilo C2-6, alquinilcarbonilo C2-6, alcoxi C1-6-carbonilo, alqueniloxicarbonilo C3-6, alquinil C3-6-oxicarbonilo, alquil C1-6-aminocarbonilo, alquenilaminocarbonilo C3-6, alquinilaminocarbonilo C3-6, alquil C1-6-sulfonilaminocarbonilo, di(alquil C1-6)-aminocarbonilo, N-(alquenil C3-6)-N-(alquil C1-6)-aminocarbonilo, N-(alquinil C3-6)-N(alquilo C1-6)-aminocarbonilo, N-(alcoxi C1-6)-N-(alquil C1-6)-amino-carbonilo, N-(alquenil C3-6)-N-(alcoxi C1-6)-aminocarbonilo, N-(alquinil C3-6)- N-(alcoxi C1-6)-aminocarbonilo, di-(alquil C1-6)-aminotiocarbonilo, (alquil 1-6)cianoimino, (amino)cianoimino, [(alquil C1-6)amino]cianoimino, [di(alquil C1-6)amino]cianoimino, alquil C1-6-carbonil-alquilo C1-6, alcoxi C1-6-imino-alquilo C1-6, N- (alquil C1-6-amino)-imino-alquilo C1-6, N-(di-alquil C1-6-amino)-imino-alquilo C1-6, o tri-alquil C1-4-sililo, en donde los radicales alquilo, cicloalquilo y alcoxi mencionados pueden estar parcial o totalmente halogenados y/o pueden llevar 1 a 3 de los siguientes grupos: ciano, hidroxi, cicloalquilo C3-6, alcoxi C1-6-alquilo C1-4, alcoxi C1-4-alcoxi C1-4-alquilo C1-4, alcoxi C1-4, alquil C1-4-tio, di(alquil C1-4)-amino, alquilo C1-4-alcoxi C1-6-carbonilamino, alquil C1-4-carbonilo, hidroxicarbonilo, alcoxi C1-4-carbonilo, aminocarbonilo, alquil C1-4-aminocarbonilo, di(alquil C1-4)aminocarbonilo o alquil C1-4-carboniloxi; fenilo, fenil-alquilo C1-6, fenilcarbonilo, fenilcarbonil-alquilo C1-6, fenoxicarbonilo, fenilaminocarbonilo, fenilsulfonilaminocarbonilo, N-(alquilo C1-6)-N-(fenil)-aminocarbonilo, fenil-alquil C1-6-carbonilo, en donde el radical fenilo puede estar parcial o totalmente halogenado y/o puede llevar 1 a 3 de los siguientes grupos: nitro, ciano, alquilo C1-4, halogenalquilo C1-4, alcoxi C1-4 o halogenalcoxi C1-4, o SO2R7; R5 es H o alquilo C1-6; R6 es alquilo C1-6, alquenilo C2-6, alquinilo C2-6, halogenalquilo C1-6, halogenalquenilo C2-6, halogenalquinilo C2-6, cianoalquilo C1-6, cianoalquenilo C2-6, cianoalquinilo C2-6, hidroxialquilo C1-6, hidroxialquenilo C2-6, hidroxialquinilo C2-6, cicloalquilo C3-6, cicloalquenilo C3-6, heterociclilo de 3 a 6 miembros, heterociclil-alquilo C1-4 de 3 a 6 miembros, en donde los radicales cicloalquilo, cicloalquenilo o heterociclilo de 3 a 6 miembros antes mencionados peden estar parcial o totalmente halogenados y/o pueden llevar 1 a 3 radicales del grupo oxo, ciano, nitro, alquilo C1-6, halogenalquilo C1-6, hidroxi, alcoxi C1-6, halogenalcoxi C1-6, hidroxicarbonilo, alcoxi C1-6-carbonilo, hidroxicarbonil-alcoxi C1-6, alcoxi C1-6-carbonil-alcoxi C1-6, amino, alquil C1-6-amino, di(alquil C1-6)amino, alquil C1-6-sulfonilamino, halogenalquil C1-6-sulfonilamino, aminocarbonilamino, (alquil C1-6-amino)carbonilamino, di-(alquil C1-6)-aminocarbonilamino, arilo y aril(alquilo C1-6); alcoxi C1-6-alquilo C1-4, alquenil C2-6-oxi-alquilo C1-4, alquinil C2-6-oxi-alquilo C1-4, halogenalcoxi C1-6-alquilo C1-4, halogenalquenil C2-6-oxi-alquilo C1-4, halogenalquinil C2-6-oxi-alquilo C1-4, alcoxi C1-6-alcoxi C1-4-alquilo C1-4, alquil C1-6-tio-alquilo C1-4, alquenil C2-6-tio-alquilo C1-4, alquinil C2-6-tioalquilo C1-4, halogenalquil C1-6-tioalquilo C1-4, halogenalquenil C2-6-tioalquilo C1-4, halogenalquinil C2-6-tioalquilo C1-4, alquil C1-6-sulfinil-alquilo C1-4, halogenalquil C1-6-sulfinil-alquilo C1-4, alquil C1-4-sulfonil-alquilo C1-4, halogenalquil C1-6-sulfonil-alquilo C1-4, amino-alquilo C1-4, alquil C1-6-amino-alquilo C1-4, di-(alquil C1-6)amino-alquilo C1-4, alquil C1-6-sulfonilamino-alquilo C1-4, alquil C1-6-sulfonil-(alquil C1-6)-amino-alquilo C1-4, alquil C1-6-carbonilo, hidroxicarbonilo, alcoxi C1-6-carbonilo, aminocarbonilo, alquil C1-6-aminocarbonilo, di-(alquil C1-6)-aminocarbonilo, alquil C1-6-carbonil-alquilo C1-6, hidroxicarbonil-alquilo C1-4, alcoxi C1-6-carbonil-alquilo C1-4, halogenalcoxi C1-6-carbonil-alquilo C1-4, alquil C1-6-carboniloxi-alquilo C1-4, aminocarbonil- alquilo C1-4, alquil C1-6-aminocarbonil-alquilo C1-4, di(alquil C1-6)aminocarbonil-alquilo C1-4, formilamino-alquilo C1-4, alcoxi C1-6-carbonilamino-alquilo C1-4, alquil C1-6-carbonilamino-alquilo C1-4, alquil C1-6-carbonil-(alquil C1-6-amino)- alquilo C1-4, [(alquil C1-6)aminocarboniloxi]-alquilo C1-4, [di(-alquil C1-6)aminocarboniloxi]-alquilo C1-4, {di-[di-(alquil C1-6)amino]carboniloxi}-alquilo C1-4, [(alquil C1-6-amino)carbonilamino]-alquilo C1-4, [di-(alquil C1-6)aminocarbonilamino]- alquilo C1-4; fenil-alquilo C1-4, fenil-alquenilo C2-4, fenil-alquinilo C2-4, fenil-halogenalquilo C1-4, fenil-halogenalquenilo C2-4, fenil-halogenalquinilo C2-4, fenil-hidroxialquilo C1-4, fenil-hidroxialquenilo C2-4, fenil-hidroxialquinilo C2-4, fenilcarbonil-alquilo C1-4, fenilcarbonilamino-alquilo C1-4, fenilcarboniloxi-alquilo C1-4, fenilcarbonil-alquilo C1-4, feniloxi-alquilo C1-4, feniltio-alquilo C1-4, fenilsulfinil-alquilo C1-4, fenilsulfonil-alquilo C1-4, heteroaril-alquilo C1-4, heteroaril-alquenilo C2-4, heteroaril-alquinilo C2-4, heteroaril-halogenalquilo C1-4, heteroaril-halogenalquenilo C2-4, heteroaril-halogenalquinilo C2-4, heteroaril-hidroxialquilo C1-4, heteroaril-hidroxialquenilo C2-4, heteroaril-hidroxialquinilo C1-4, heteroarilcarbonil-alquilo C1-4, heteroarilcarboniloxi-alquilo C1-4, heteroariloxicarbonil-alquilo C1-4, heteroariloxi-alquilo C1-4, heteroariltio-alquilo C1-4, heteroarilsulfinil-alquilo C1-4, heteroarilsulfonil-alquilo C1-4, en donde los radicales fenilo y heteroarilo antes mencionados pueden estar parcial o totalmente halogenados y/o pueden llevar 1 a 3 radicales del grupo ciano, nitro, alquilo C1-6, halogenalquilo C1-6, hidroxi, alcoxi C1-6, halogenalcoxi C1-6, hidroxicarbonilo, alcoxi C1-6-carbonilo, hidroxicarbonil-alcoxi C1-6, alcoxi C1-6-carbonil-alcoxi C1-6, amino, alquil C1-6-amino, di-(alquil C1-6)amino, alquil C1-6-sulfonilamino, halogenalquil C1-6-sulfonilamino, (alquil C1-6-amino)carbonilamino, di-(alquil C1-6)- aminocarbonilamino, arilo y aril(alquilo C1-6); R7 alquilo C1-6, halogenalquilo C1-6 o fenilo; en donde el radical fenilo puede estar parcial o totalmente halogenado y/o puede llevar 1 a 3 de los siguientes grupos: alquilo C1-6, haloalquilo C1-6, o alcoxi C1-6; así como sus sales de utilidad en agricultura.
ARP060102179A 2005-05-25 2006-05-24 Serin- amidas sustituidas con heteroaroilo AR057331A1 (es)

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DE102005024599 2005-05-25

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US (1) US7879761B2 (es)
EP (1) EP1888532A1 (es)
JP (1) JP4981037B2 (es)
CN (1) CN101228133A (es)
AR (1) AR057331A1 (es)
AU (1) AU2006251302A1 (es)
BR (1) BRPI0611498B1 (es)
CA (1) CA2609243A1 (es)
EA (1) EA013636B1 (es)
IL (1) IL187502A0 (es)
MX (1) MX2007014490A (es)
PE (1) PE20070051A1 (es)
TW (1) TW200716558A (es)
UA (1) UA90720C2 (es)
UY (1) UY29565A1 (es)
WO (1) WO2006125687A1 (es)
ZA (1) ZA200711009B (es)

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BRPI0611498A2 (pt) 2011-02-22
PE20070051A1 (es) 2007-02-01
JP4981037B2 (ja) 2012-07-18
TW200716558A (en) 2007-05-01
WO2006125687A1 (de) 2006-11-30
BRPI0611498B1 (pt) 2015-10-13
ZA200711009B (en) 2009-11-25
EA013636B1 (ru) 2010-06-30
US20080200338A1 (en) 2008-08-21
JP2008542231A (ja) 2008-11-27
CA2609243A1 (en) 2006-11-30
EA200702443A1 (ru) 2008-06-30
UY29565A1 (es) 2006-12-29
AU2006251302A1 (en) 2006-11-30
US7879761B2 (en) 2011-02-01
EP1888532A1 (de) 2008-02-20
CN101228133A (zh) 2008-07-23

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