AR057331A1 - Serin- amidas sustituidas con heteroaroilo - Google Patents
Serin- amidas sustituidas con heteroaroiloInfo
- Publication number
- AR057331A1 AR057331A1 ARP060102179A ARP060102179A AR057331A1 AR 057331 A1 AR057331 A1 AR 057331A1 AR P060102179 A ARP060102179 A AR P060102179A AR P060102179 A ARP060102179 A AR P060102179A AR 057331 A1 AR057331 A1 AR 057331A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- alkoxy
- amino
- phenyl
- aminocarbonyl
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pyridine Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Furan Compounds (AREA)
Abstract
Procedimientos y productos intermediarios para su preparacion, así como el uso de esos compuestos o agentes que contienen estos compuestos, para el combate de plantas no deseadas. Reivindicacion 1: Serin-amidas sustituidas con heteroaroílo, caracterizadas porque tienen la formula en donde las variables tienen los siguientes significados: A es heteroarilo de 5 o 6 miembros con uno a cuatro átomos de N, o con uno a tres átomos de N y un átomo de O o S, o con un átomo de O o S, que puede estar parcial o totalmente halogenado y/o que puede llevar 1 a 3 radicales del grupo ciano, alquilo C1-6, cicloalquilo C3-6, halogenoalquilo C1-6, alcoxi C1-6, halogenoalcoxi C1-6 y alcoxi C1-6-alquilo C1-4; R1, R2 es H, hidroxi o alcoxi C1-6; R3 es alquilo C1-6, cianoalquilo C1-4 o halogenoalquilo C1-6; R4 es H, alquilo C1-6, cicloalquilo C3-6, alquenilo C3-6, alquinilo C3-6, halogenalquenilo C3-6, halogenalquinilo C3-6, formilo, alquil C1-6-carbonilo, cicloalquilcarbonilo C3-6, alquenilcarbonilo C2-6, alquinilcarbonilo C2-6, alcoxi C1-6-carbonilo, alqueniloxicarbonilo C3-6, alquinil C3-6-oxicarbonilo, alquil C1-6-aminocarbonilo, alquenilaminocarbonilo C3-6, alquinilaminocarbonilo C3-6, alquil C1-6-sulfonilaminocarbonilo, di(alquil C1-6)-aminocarbonilo, N-(alquenil C3-6)-N-(alquil C1-6)-aminocarbonilo, N-(alquinil C3-6)-N(alquilo C1-6)-aminocarbonilo, N-(alcoxi C1-6)-N-(alquil C1-6)-amino-carbonilo, N-(alquenil C3-6)-N-(alcoxi C1-6)-aminocarbonilo, N-(alquinil C3-6)- N-(alcoxi C1-6)-aminocarbonilo, di-(alquil C1-6)-aminotiocarbonilo, (alquil 1-6)cianoimino, (amino)cianoimino, [(alquil C1-6)amino]cianoimino, [di(alquil C1-6)amino]cianoimino, alquil C1-6-carbonil-alquilo C1-6, alcoxi C1-6-imino-alquilo C1-6, N- (alquil C1-6-amino)-imino-alquilo C1-6, N-(di-alquil C1-6-amino)-imino-alquilo C1-6, o tri-alquil C1-4-sililo, en donde los radicales alquilo, cicloalquilo y alcoxi mencionados pueden estar parcial o totalmente halogenados y/o pueden llevar 1 a 3 de los siguientes grupos: ciano, hidroxi, cicloalquilo C3-6, alcoxi C1-6-alquilo C1-4, alcoxi C1-4-alcoxi C1-4-alquilo C1-4, alcoxi C1-4, alquil C1-4-tio, di(alquil C1-4)-amino, alquilo C1-4-alcoxi C1-6-carbonilamino, alquil C1-4-carbonilo, hidroxicarbonilo, alcoxi C1-4-carbonilo, aminocarbonilo, alquil C1-4-aminocarbonilo, di(alquil C1-4)aminocarbonilo o alquil C1-4-carboniloxi; fenilo, fenil-alquilo C1-6, fenilcarbonilo, fenilcarbonil-alquilo C1-6, fenoxicarbonilo, fenilaminocarbonilo, fenilsulfonilaminocarbonilo, N-(alquilo C1-6)-N-(fenil)-aminocarbonilo, fenil-alquil C1-6-carbonilo, en donde el radical fenilo puede estar parcial o totalmente halogenado y/o puede llevar 1 a 3 de los siguientes grupos: nitro, ciano, alquilo C1-4, halogenalquilo C1-4, alcoxi C1-4 o halogenalcoxi C1-4, o SO2R7; R5 es H o alquilo C1-6; R6 es alquilo C1-6, alquenilo C2-6, alquinilo C2-6, halogenalquilo C1-6, halogenalquenilo C2-6, halogenalquinilo C2-6, cianoalquilo C1-6, cianoalquenilo C2-6, cianoalquinilo C2-6, hidroxialquilo C1-6, hidroxialquenilo C2-6, hidroxialquinilo C2-6, cicloalquilo C3-6, cicloalquenilo C3-6, heterociclilo de 3 a 6 miembros, heterociclil-alquilo C1-4 de 3 a 6 miembros, en donde los radicales cicloalquilo, cicloalquenilo o heterociclilo de 3 a 6 miembros antes mencionados peden estar parcial o totalmente halogenados y/o pueden llevar 1 a 3 radicales del grupo oxo, ciano, nitro, alquilo C1-6, halogenalquilo C1-6, hidroxi, alcoxi C1-6, halogenalcoxi C1-6, hidroxicarbonilo, alcoxi C1-6-carbonilo, hidroxicarbonil-alcoxi C1-6, alcoxi C1-6-carbonil-alcoxi C1-6, amino, alquil C1-6-amino, di(alquil C1-6)amino, alquil C1-6-sulfonilamino, halogenalquil C1-6-sulfonilamino, aminocarbonilamino, (alquil C1-6-amino)carbonilamino, di-(alquil C1-6)-aminocarbonilamino, arilo y aril(alquilo C1-6); alcoxi C1-6-alquilo C1-4, alquenil C2-6-oxi-alquilo C1-4, alquinil C2-6-oxi-alquilo C1-4, halogenalcoxi C1-6-alquilo C1-4, halogenalquenil C2-6-oxi-alquilo C1-4, halogenalquinil C2-6-oxi-alquilo C1-4, alcoxi C1-6-alcoxi C1-4-alquilo C1-4, alquil C1-6-tio-alquilo C1-4, alquenil C2-6-tio-alquilo C1-4, alquinil C2-6-tioalquilo C1-4, halogenalquil C1-6-tioalquilo C1-4, halogenalquenil C2-6-tioalquilo C1-4, halogenalquinil C2-6-tioalquilo C1-4, alquil C1-6-sulfinil-alquilo C1-4, halogenalquil C1-6-sulfinil-alquilo C1-4, alquil C1-4-sulfonil-alquilo C1-4, halogenalquil C1-6-sulfonil-alquilo C1-4, amino-alquilo C1-4, alquil C1-6-amino-alquilo C1-4, di-(alquil C1-6)amino-alquilo C1-4, alquil C1-6-sulfonilamino-alquilo C1-4, alquil C1-6-sulfonil-(alquil C1-6)-amino-alquilo C1-4, alquil C1-6-carbonilo, hidroxicarbonilo, alcoxi C1-6-carbonilo, aminocarbonilo, alquil C1-6-aminocarbonilo, di-(alquil C1-6)-aminocarbonilo, alquil C1-6-carbonil-alquilo C1-6, hidroxicarbonil-alquilo C1-4, alcoxi C1-6-carbonil-alquilo C1-4, halogenalcoxi C1-6-carbonil-alquilo C1-4, alquil C1-6-carboniloxi-alquilo C1-4, aminocarbonil- alquilo C1-4, alquil C1-6-aminocarbonil-alquilo C1-4, di(alquil C1-6)aminocarbonil-alquilo C1-4, formilamino-alquilo C1-4, alcoxi C1-6-carbonilamino-alquilo C1-4, alquil C1-6-carbonilamino-alquilo C1-4, alquil C1-6-carbonil-(alquil C1-6-amino)- alquilo C1-4, [(alquil C1-6)aminocarboniloxi]-alquilo C1-4, [di(-alquil C1-6)aminocarboniloxi]-alquilo C1-4, {di-[di-(alquil C1-6)amino]carboniloxi}-alquilo C1-4, [(alquil C1-6-amino)carbonilamino]-alquilo C1-4, [di-(alquil C1-6)aminocarbonilamino]- alquilo C1-4; fenil-alquilo C1-4, fenil-alquenilo C2-4, fenil-alquinilo C2-4, fenil-halogenalquilo C1-4, fenil-halogenalquenilo C2-4, fenil-halogenalquinilo C2-4, fenil-hidroxialquilo C1-4, fenil-hidroxialquenilo C2-4, fenil-hidroxialquinilo C2-4, fenilcarbonil-alquilo C1-4, fenilcarbonilamino-alquilo C1-4, fenilcarboniloxi-alquilo C1-4, fenilcarbonil-alquilo C1-4, feniloxi-alquilo C1-4, feniltio-alquilo C1-4, fenilsulfinil-alquilo C1-4, fenilsulfonil-alquilo C1-4, heteroaril-alquilo C1-4, heteroaril-alquenilo C2-4, heteroaril-alquinilo C2-4, heteroaril-halogenalquilo C1-4, heteroaril-halogenalquenilo C2-4, heteroaril-halogenalquinilo C2-4, heteroaril-hidroxialquilo C1-4, heteroaril-hidroxialquenilo C2-4, heteroaril-hidroxialquinilo C1-4, heteroarilcarbonil-alquilo C1-4, heteroarilcarboniloxi-alquilo C1-4, heteroariloxicarbonil-alquilo C1-4, heteroariloxi-alquilo C1-4, heteroariltio-alquilo C1-4, heteroarilsulfinil-alquilo C1-4, heteroarilsulfonil-alquilo C1-4, en donde los radicales fenilo y heteroarilo antes mencionados pueden estar parcial o totalmente halogenados y/o pueden llevar 1 a 3 radicales del grupo ciano, nitro, alquilo C1-6, halogenalquilo C1-6, hidroxi, alcoxi C1-6, halogenalcoxi C1-6, hidroxicarbonilo, alcoxi C1-6-carbonilo, hidroxicarbonil-alcoxi C1-6, alcoxi C1-6-carbonil-alcoxi C1-6, amino, alquil C1-6-amino, di-(alquil C1-6)amino, alquil C1-6-sulfonilamino, halogenalquil C1-6-sulfonilamino, (alquil C1-6-amino)carbonilamino, di-(alquil C1-6)- aminocarbonilamino, arilo y aril(alquilo C1-6); R7 alquilo C1-6, halogenalquilo C1-6 o fenilo; en donde el radical fenilo puede estar parcial o totalmente halogenado y/o puede llevar 1 a 3 de los siguientes grupos: alquilo C1-6, haloalquilo C1-6, o alcoxi C1-6; así como sus sales de utilidad en agricultura.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102005024599 | 2005-05-25 |
Publications (1)
Publication Number | Publication Date |
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AR057331A1 true AR057331A1 (es) | 2007-11-28 |
Family
ID=36702367
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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ARP060102179A AR057331A1 (es) | 2005-05-25 | 2006-05-24 | Serin- amidas sustituidas con heteroaroilo |
Country Status (17)
Country | Link |
---|---|
US (1) | US7879761B2 (es) |
EP (1) | EP1888532A1 (es) |
JP (1) | JP4981037B2 (es) |
CN (1) | CN101228133A (es) |
AR (1) | AR057331A1 (es) |
AU (1) | AU2006251302A1 (es) |
BR (1) | BRPI0611498B1 (es) |
CA (1) | CA2609243A1 (es) |
EA (1) | EA013636B1 (es) |
IL (1) | IL187502A0 (es) |
MX (1) | MX2007014490A (es) |
PE (1) | PE20070051A1 (es) |
TW (1) | TW200716558A (es) |
UA (1) | UA90720C2 (es) |
UY (1) | UY29565A1 (es) |
WO (1) | WO2006125687A1 (es) |
ZA (1) | ZA200711009B (es) |
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DE10204951A1 (de) | 2002-02-06 | 2003-08-14 | Basf Ag | Phenylalaninderivate als Herbizide |
AU2004303492A1 (en) | 2003-12-19 | 2005-07-07 | Basf Aktiengesellschaft | Benzoyl-substituted phenylalanine amides |
EA011928B1 (ru) * | 2003-12-19 | 2009-06-30 | Басф Акциенгезельшафт | Замещённые гетероароилом фенилаланин-амиды |
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CA2577181A1 (en) * | 2004-09-16 | 2006-03-23 | Basf Aktiengesellschaft | Heteroaroyl-substituted serine amides utilized as herbicides |
-
2006
- 2006-03-29 JP JP2008512789A patent/JP4981037B2/ja not_active Expired - Fee Related
- 2006-03-29 AU AU2006251302A patent/AU2006251302A1/en not_active Abandoned
- 2006-03-29 UA UAA200714187A patent/UA90720C2/ru unknown
- 2006-03-29 EA EA200702443A patent/EA013636B1/ru not_active IP Right Cessation
- 2006-03-29 WO PCT/EP2006/061128 patent/WO2006125687A1/de active Application Filing
- 2006-03-29 US US11/915,227 patent/US7879761B2/en not_active Expired - Fee Related
- 2006-03-29 CN CNA2006800271632A patent/CN101228133A/zh active Pending
- 2006-03-29 CA CA002609243A patent/CA2609243A1/en not_active Abandoned
- 2006-03-29 MX MX2007014490A patent/MX2007014490A/es not_active Application Discontinuation
- 2006-03-29 BR BRPI0611498A patent/BRPI0611498B1/pt not_active IP Right Cessation
- 2006-03-29 EP EP06725384A patent/EP1888532A1/de not_active Withdrawn
- 2006-04-14 TW TW095113549A patent/TW200716558A/zh unknown
- 2006-05-24 AR ARP060102179A patent/AR057331A1/es unknown
- 2006-05-24 PE PE2006000547A patent/PE20070051A1/es not_active Application Discontinuation
- 2006-05-25 UY UY29565A patent/UY29565A1/es unknown
-
2007
- 2007-11-20 IL IL187502A patent/IL187502A0/en unknown
- 2007-12-19 ZA ZA200711009A patent/ZA200711009B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
UA90720C2 (en) | 2010-05-25 |
IL187502A0 (en) | 2008-03-20 |
MX2007014490A (es) | 2008-02-11 |
BRPI0611498A2 (pt) | 2011-02-22 |
PE20070051A1 (es) | 2007-02-01 |
JP4981037B2 (ja) | 2012-07-18 |
TW200716558A (en) | 2007-05-01 |
WO2006125687A1 (de) | 2006-11-30 |
BRPI0611498B1 (pt) | 2015-10-13 |
ZA200711009B (en) | 2009-11-25 |
EA013636B1 (ru) | 2010-06-30 |
US20080200338A1 (en) | 2008-08-21 |
JP2008542231A (ja) | 2008-11-27 |
CA2609243A1 (en) | 2006-11-30 |
EA200702443A1 (ru) | 2008-06-30 |
UY29565A1 (es) | 2006-12-29 |
AU2006251302A1 (en) | 2006-11-30 |
US7879761B2 (en) | 2011-02-01 |
EP1888532A1 (de) | 2008-02-20 |
CN101228133A (zh) | 2008-07-23 |
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