AR044065A1 - Procedimiento para preparar nicotinaldehidos, sustancias de partida para dicho procedimiento y el uso de morfolinamidas del acido nicotinico para la preparacion de los nicotinaldehidos correspondientes - Google Patents
Procedimiento para preparar nicotinaldehidos, sustancias de partida para dicho procedimiento y el uso de morfolinamidas del acido nicotinico para la preparacion de los nicotinaldehidos correspondientesInfo
- Publication number
- AR044065A1 AR044065A1 ARP040101376A ARP040101376A AR044065A1 AR 044065 A1 AR044065 A1 AR 044065A1 AR P040101376 A ARP040101376 A AR P040101376A AR P040101376 A ARP040101376 A AR P040101376A AR 044065 A1 AR044065 A1 AR 044065A1
- Authority
- AR
- Argentina
- Prior art keywords
- nicotinic acid
- procedure
- nicotinaldehydes
- starting substances
- hal
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
- C07D213/46—Oxygen atoms
- C07D213/48—Aldehydo radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/56—Amides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
Se describe un procedimiento para la preparación reductiva de nicotinaldehídos que en calidad de sustancias de partida para la reducción emplea las correspondientes morfolinamidas del ácido nicotínico. Dichas morfolinamidas de ácido nicotínico responden preferentemente a la fórmula (1), en la que: R1', R1'' representan independientemente H, Hal, A, OA, CH2R2 o Ar; R2 representa OA o NA2; A representa alquilo de cadena recta o ramificada y de C1-10, en donde uno o dos grupos CH2 pueden estar reemplazados por átomos de O o S y/o por grupos -CH=CH y/o también 1 a 7 átomos de H pueden estar reemplazados por F; Ar representa un sistema homo o heterocíclico con los heteroátomos O, N, S, de uno o más núcleos, insaturado, parcialmente o totalmente saturado, no sustituido o mono o polisustituido con Hal A, OA, NA2, NO2, NASO2A, SO2NA, SO2A; y Hal representa F, Cl, Br o I. También se describen el uso de morfolinamidas del ácido nicotínico y las sustancias de partida para el procedimiento mencionado más arriba. Este procedimiento permite obtener aldehídos del ácido nicotínico con rendimientos casi cuantitativos por reducción en condiciones normales (temperatura ambiente y sin presión).
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10318690A DE10318690B3 (de) | 2003-04-24 | 2003-04-24 | Verfahren zur Herstellung von Nicotinaldehyden |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR044065A1 true AR044065A1 (es) | 2005-08-24 |
Family
ID=33154397
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP040101376A AR044065A1 (es) | 2003-04-24 | 2004-04-23 | Procedimiento para preparar nicotinaldehidos, sustancias de partida para dicho procedimiento y el uso de morfolinamidas del acido nicotinico para la preparacion de los nicotinaldehidos correspondientes |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US7528256B2 (es) |
| EP (1) | EP1615891B1 (es) |
| JP (1) | JP2006524196A (es) |
| KR (1) | KR101106621B1 (es) |
| CN (1) | CN100355730C (es) |
| AR (1) | AR044065A1 (es) |
| AU (1) | AU2004232454B2 (es) |
| BR (1) | BRPI0409644B1 (es) |
| CA (1) | CA2523190C (es) |
| DE (1) | DE10318690B3 (es) |
| ES (1) | ES2426412T3 (es) |
| HK (1) | HK1087111A1 (es) |
| MX (1) | MXPA05011253A (es) |
| RU (1) | RU2339619C2 (es) |
| WO (1) | WO2004094383A1 (es) |
| ZA (1) | ZA200509495B (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5807955B2 (ja) * | 2011-12-15 | 2015-11-10 | 国立大学法人横浜国立大学 | 植物用抵抗性誘導剤、植物の抵抗性誘導方法、及び植物病害の予防方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2994182B2 (ja) * | 1992-07-23 | 1999-12-27 | 石原産業株式会社 | アミド系化合物又はその塩、それらの製造方法及びそれらを含有する有害動物防除剤 |
| US6521618B2 (en) * | 2000-03-28 | 2003-02-18 | Wyeth | 3-cyanoquinolines, 3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors |
| AR035851A1 (es) * | 2000-03-28 | 2004-07-21 | Wyeth Corp | 3-cianoquinolinas, 3-ciano-1,6-naftiridinas y 3-ciano-1,7-naftiridinas como inhibidoras de proteina quinasas |
| SI1427724T1 (sl) * | 2001-09-19 | 2006-10-31 | Merck Patent Gmbh | Nova uporaba substituiranih aminometil-kromanov |
-
2003
- 2003-04-24 DE DE10318690A patent/DE10318690B3/de not_active Expired - Fee Related
-
2004
- 2004-03-27 WO PCT/EP2004/003272 patent/WO2004094383A1/de active Application Filing
- 2004-03-27 BR BRPI0409644A patent/BRPI0409644B1/pt not_active IP Right Cessation
- 2004-03-27 EP EP04723902.5A patent/EP1615891B1/de not_active Expired - Lifetime
- 2004-03-27 CN CNB2004800108542A patent/CN100355730C/zh not_active Expired - Fee Related
- 2004-03-27 ES ES04723902T patent/ES2426412T3/es not_active Expired - Lifetime
- 2004-03-27 AU AU2004232454A patent/AU2004232454B2/en not_active Ceased
- 2004-03-27 RU RU2005136382/04A patent/RU2339619C2/ru not_active IP Right Cessation
- 2004-03-27 JP JP2006504889A patent/JP2006524196A/ja active Pending
- 2004-03-27 KR KR1020057020088A patent/KR101106621B1/ko active IP Right Grant
- 2004-03-27 MX MXPA05011253A patent/MXPA05011253A/es active IP Right Grant
- 2004-03-27 US US10/554,061 patent/US7528256B2/en active Active
- 2004-03-27 CA CA2523190A patent/CA2523190C/en not_active Expired - Fee Related
- 2004-04-23 AR ARP040101376A patent/AR044065A1/es unknown
-
2005
- 2005-11-23 ZA ZA200509495A patent/ZA200509495B/xx unknown
-
2006
- 2006-06-28 HK HK06107301A patent/HK1087111A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200509495B (en) | 2009-03-25 |
| AU2004232454B2 (en) | 2010-02-25 |
| CA2523190A1 (en) | 2004-11-04 |
| AU2004232454A1 (en) | 2004-11-04 |
| EP1615891A1 (de) | 2006-01-18 |
| EP1615891B1 (de) | 2013-06-19 |
| KR101106621B1 (ko) | 2012-01-20 |
| CA2523190C (en) | 2012-01-24 |
| CN100355730C (zh) | 2007-12-19 |
| US20060199965A1 (en) | 2006-09-07 |
| KR20060006056A (ko) | 2006-01-18 |
| BRPI0409644B1 (pt) | 2019-01-22 |
| RU2339619C2 (ru) | 2008-11-27 |
| ES2426412T3 (es) | 2013-10-23 |
| JP2006524196A (ja) | 2006-10-26 |
| DE10318690B3 (de) | 2004-11-11 |
| RU2005136382A (ru) | 2006-06-10 |
| US7528256B2 (en) | 2009-05-05 |
| WO2004094383A1 (de) | 2004-11-04 |
| BRPI0409644A (pt) | 2006-04-25 |
| CN1777587A (zh) | 2006-05-24 |
| MXPA05011253A (es) | 2005-12-14 |
| HK1087111A1 (en) | 2006-10-06 |
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| FB | Suspension of granting procedure |