AR036631A1 - Pirazoles 3-substituidos insecticidas y acaricidas; metodo para el control de insectos o acaros; metodo para la proteccion de una planta; metodo para la proteccion de madera, productos de madera o estructuras de madera; composicion; y procedimiento para la preparacion de estos compuestos - Google Patents

Pirazoles 3-substituidos insecticidas y acaricidas; metodo para el control de insectos o acaros; metodo para la proteccion de una planta; metodo para la proteccion de madera, productos de madera o estructuras de madera; composicion; y procedimiento para la preparacion de estos compuestos

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Publication number
AR036631A1
AR036631A1 ARP020103615A ARP020103615A AR036631A1 AR 036631 A1 AR036631 A1 AR 036631A1 AR P020103615 A ARP020103615 A AR P020103615A AR P020103615 A ARP020103615 A AR P020103615A AR 036631 A1 AR036631 A1 AR 036631A1
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AR
Argentina
Prior art keywords
halogen
haloalkyl
alkyl
hydrogen
alkoxy
Prior art date
Application number
ARP020103615A
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English (en)
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of AR036631A1 publication Critical patent/AR036631A1/es

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/28—Two oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C07D231/40—Acylated on said nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

Pirazoles 3-substituidos que tienen la fórmula (1), en la cual las variables y el índice tienen los siguientes significados: R1 es hidrógeno, halógeno, alquilo C1-6, haloalquilo C1-6, alquenilo C2-6, haloalquenilo C2-6, alquiltio C1-6, alcoxi C1-6-alquilo C1-4, alquiltio C1-6-alquilo C1-4 o fenilo que no está sustituido o está sustituido con 1 a 3 grupos Ra; Ra es halógeno, nitro, ciano, alquilo C1-6, haloalquilo C1-6, alquiltio C1-6, haloalquiltio C1-6, alcoxi C1-6 o haloalcoxi C1-6; R2 es hidrógeno, halógeno, alquilo C1-6, haloalquilo C1-6, alquenilo C2-6, haloalquenilo C2-6 o fenilo que no está sustituido o está sustituido con 1 a 3 grupos Ra; A es hidrógeno, hidroxi, ciano, nitro, halógeno, ródano, alcoxi C1-6, haloalcoxi C1-6, alqueniloxi C2-6, alquiltio C1-6, haloalquiltio C1-6, alquilsulfinilo C1-6, alquilsulfonilo C1-6, aminotiocarbonilo, hidroxicarbonilo, alcoxicarbonilo C1-6 o aminocarbonilo; B es hidrógeno, hidroxi, amino, ciano, nitro o halógeno; alquilo C1-6 no sustituido o sustituido con 1 a 3 grupos seleccionados de halógeno y ciano; alcoxi C1-6 no sustituido o sustituido con 1 a 3 grupos seleccionados de halógeno, ciano, alquenilo C2-4 y alcoxicarbonilo C1-6-alquenilo C2-4; alquenilo C2-6 no sustituido o sustituido con 1 a 3 grupos seleccionados de halógeno y ciano; alqueniloxi C2-6, alquiltio C1-6, haloalquilo C1-6, alcoxitiocarboniltio C1-6, alcoxicarbonil C1-6-alcoxi C1-4, alcoxicarbonil C1-6-alquiltio C1-4, alquilsulfinilo C1-6, alquilsulfonilo C1-6, aminotiocarbonilo, NR3R4, N=CHOR5 o N=CHNR5; R3 y R4 son cada uno independientemente hidrógeno, alquilo C1-6, alcoxicarbonil C1-6-alquilo C1-4, [(alcoxicarbonil C1-6)(alquenil C2-4)]alquilo C1-4, alcoxicarbonilo C1-6-alquenilo C2-4, alquilcarbonilo C1-6, cicloalquilcarbonilo C3-7, alquilaminocarbonilo C1-6, di-(alquil C1-6)aminocarbonilo, alcoxicarbonilo C1-6, alcoxiaminosulfonilo C1-6 o di-(alcoxi C1-6)aminosulfonilo; R5 es alquilo C1-6, haloalquilo C1-6 o fenilalquilo C1-4; Q es hidrógeno, nitro, halógeno, haloalquilo C1-4, alquilamino C1-6, dialquilamino C1-6, alcoxi C1-6, haloalcoxi C1-6 o alqueniloxi C2-6; X es hidrógeno, halógeno, haloalquilo C1-6. alcoxi C1-6 o haloalcoxi C1-6; Y es hidrógeno, halógeno, haloalquilo C1-6, alcoxi C1-6 o haloalcoxi C1-6; Z es hidrógeno, halógeno, haloalquilo C1-6, alcoxi C1-6 o haloalcoxi C1-6; M es N ó CR6; R6 es hidrógeno, nitro, halógeno o haloalquilo C1-4; y n es 0, 1, 2, 3 ó 4; con la condición de que cuando R1 es hidrógeno, n no es 0; método para el control de insectos o acáridos; método para la protección de una planta; método para la protección de madera, productos de madera o estructuras de madera; composición; y procedimiento para la preparación de estos compuestos. Estos compuestos se usan también para tratar, controlar, prevenir y proteger contra infección causada por arácnidos y artrópodos endo y ectoparasíticos.El procedimiento de preparación de los compuestos de fórmula (2), en donde A es ciano y B es amino, consiste en que compuestos de fórmula (3) se hacen reaccionar con malononitrilo en presencia de una base, donde los valores de los sustituyentes son los mencionados arriba).
ARP020103615A 2001-09-25 2002-09-25 Pirazoles 3-substituidos insecticidas y acaricidas; metodo para el control de insectos o acaros; metodo para la proteccion de una planta; metodo para la proteccion de madera, productos de madera o estructuras de madera; composicion; y procedimiento para la preparacion de estos compuestos AR036631A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US32463301P 2001-09-25 2001-09-25

Publications (1)

Publication Number Publication Date
AR036631A1 true AR036631A1 (es) 2004-09-22

Family

ID=23264427

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP020103615A AR036631A1 (es) 2001-09-25 2002-09-25 Pirazoles 3-substituidos insecticidas y acaricidas; metodo para el control de insectos o acaros; metodo para la proteccion de una planta; metodo para la proteccion de madera, productos de madera o estructuras de madera; composicion; y procedimiento para la preparacion de estos compuestos

Country Status (16)

Country Link
US (1) US20040260097A1 (es)
EP (1) EP1432688A1 (es)
JP (1) JP2005512969A (es)
KR (1) KR20040035846A (es)
CN (1) CN1305857C (es)
AR (1) AR036631A1 (es)
BR (1) BR0212385A (es)
CA (1) CA2460906A1 (es)
EA (1) EA007969B1 (es)
HU (1) HUP0402238A3 (es)
IL (1) IL160444A0 (es)
MX (1) MXPA04002040A (es)
PL (1) PL370353A1 (es)
UA (1) UA79758C2 (es)
WO (1) WO2003029222A1 (es)
ZA (1) ZA200402932B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2004196795A (ja) * 2002-12-16 2004-07-15 Wyeth 外部寄生虫駆除剤としてのｎ−フェニル−３−シクロプロピルピラゾール−４−カルボニトリル
FR2848780B1 (fr) * 2002-12-19 2005-05-13 Solvay Utilisation d'une poudre acaricide
GB0905365D0 (en) 2009-03-27 2009-05-13 Norbrook Lab Ltd A topical parasiticide composition
RU2514004C1 (ru) * 2012-10-25 2014-04-27 Государственное научное учреждение Курский научно-исследовательский институт агропромышленного производства Россельхозакадемии Способ получения комплексного препарата с иммунометаболической и антгельминтной активностью
EP3068385A4 (en) * 2013-08-15 2017-08-02 Sylleta Inc. Compositions and methods for control of marine ectoparasites
EP3872068A1 (en) * 2015-12-16 2021-09-01 Nippon Soda Co., Ltd. Arylazole compound and pest control agent
WO2023174397A1 (en) * 2022-03-18 2023-09-21 Insilico Medicine Ip Limited Pyrazole membrane-associated tyrosine-and threonine-specific cdc2-inhibitory kinase (pkmyt1) inhibitors and uses thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3509567A1 (de) * 1985-03-16 1986-09-18 Bayer Ag, 5090 Leverkusen Herbizide und insektizide mittel auf basis von pyrazolderivaten
GB8531485D0 (en) * 1985-12-20 1986-02-05 May & Baker Ltd Compositions of matter
US5232940A (en) * 1985-12-20 1993-08-03 Hatton Leslie R Derivatives of N-phenylpyrazoles
AU6517196A (en) * 1995-07-13 1997-02-10 Knoll Aktiengesellschaft Piperazine derivatives as therapeutic agents
ES2191076T3 (es) * 1995-12-19 2003-09-01 Bayer Cropscience Sa Nuevos derivados de 1-aril-pirazol y su empleo como plaguicidas.
US6531477B1 (en) * 1998-10-13 2003-03-11 Dupont Pharmaceuticals Company 6-substituted pyrazolo [3,4-d] pyrimidin-4-ones useful as cyclin dependent kinase inhibitors

Also Published As

Publication number Publication date
EP1432688A1 (en) 2004-06-30
EA200400413A1 (ru) 2004-08-26
ZA200402932B (en) 2005-04-19
HUP0402238A2 (hu) 2005-02-28
JP2005512969A (ja) 2005-05-12
CN1558902A (zh) 2004-12-29
PL370353A1 (en) 2005-05-16
HUP0402238A3 (en) 2008-02-28
IL160444A0 (en) 2004-07-25
CN1305857C (zh) 2007-03-21
CA2460906A1 (en) 2003-04-10
US20040260097A1 (en) 2004-12-23
BR0212385A (pt) 2004-08-17
KR20040035846A (ko) 2004-04-29
WO2003029222A1 (en) 2003-04-10
UA79758C2 (en) 2007-07-25
MXPA04002040A (es) 2004-06-07
EA007969B1 (ru) 2007-02-27

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