AR033504A1 - Uso de 1-arilpirazoles para preparar una composicion para el control de parasitos en o sobre un animal; compuestos relacionados; y composicion que los contiene - Google Patents

Uso de 1-arilpirazoles para preparar una composicion para el control de parasitos en o sobre un animal; compuestos relacionados; y composicion que los contiene

Info

Publication number
AR033504A1
AR033504A1 ARP000106403A ARP000106403A AR033504A1 AR 033504 A1 AR033504 A1 AR 033504A1 AR P000106403 A ARP000106403 A AR P000106403A AR P000106403 A ARP000106403 A AR P000106403A AR 033504 A1 AR033504 A1 AR 033504A1
Authority
AR
Argentina
Prior art keywords
optionally substituted
alkyl
haloalkyl
composition
r205r206n
Prior art date
Application number
ARP000106403A
Other languages
English (en)
Original Assignee
Aventis Cropscience Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Cropscience Sa filed Critical Aventis Cropscience Sa
Publication of AR033504A1 publication Critical patent/AR033504A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/561,2-Diazoles; Hydrogenated 1,2-diazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/02Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/18Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, directly attached to a heterocyclic or cycloaliphatic ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/28Two oxygen or sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Uso de una cantidad efectiva parasiticida, sustancialmente no emética de un 1-arilpirazol de formula (1) en la cual R201 es ciano, C(O)alquilo, C(S)NH2, C(NH)OR203, C(NH)SR203, alquilo, C(=NOH)NH2, C(=NNH2)NH2, C(O)NH2, C(O)NHR205, C(O)NR205R206, haloalquilo o heterociclilo del grupo (2) opcionalmente sustituido con R203; R202 es S(O)hR203 alquenilo C2-6, haloalquenilo C2-6, cicloalquilo, halocicloalquilo, cicloalquilalquilo, alquinilo C2-6, nitro o imidazol-2-ilo opcionalmente sustituido con alquilo, alcoxi, haloalquilo, halogeno, ciano y/o nitro; R203 es alquilo o haloalquilo; R204 es ûOH, R205O-, HC(O)O-, R205C(O)O-, R205OC(O)O-, NH2C(O)O-, R205NHC(O)O-, R205R206NC(O)O-, R205S(O)nC(O)O-, R206SO2O-, aril-SO2O-, oxacicloalquiloxi (C4-7), R205R206N-C(NR205)-O-, R205R206N-C(NH)-O, R205NH-C(NR205)-O-, R205NH(NH)-O-, R205N=CH-O-, R205N=C(R206)-O-, R205NH-C(S)-O-, R205R206N-C(S)-O-; R205 es alquilo, haloalquilo, cicloalquilo, halocicloalquilo, alcoxialquilo, haloalcoxialquilo, adamantilo, aminoalquilo, alquilaminoalquilo, dialquilaminoalquilo, haloalquilaminoalquilo, di(haloalquilo)aminoalquilo, arilo opcionalmente sustituido, hetarilo, opcionalmente sustituido, arilalquilo opcionalmente sustituido, hetarilalquilo opcionalmente sustituido, alquenilo C2-6, alquinilo C2-6; R206 es alquilo, haloalquilo, cicloalquilo, halocicloalquilo, alcoxialquilo, haloalcoxialquilo, arilo, opcionalmente sustituido, hetarilo opcionalmente sustituido, arilaquilo opcionalmente sustituido hetarilalquilo opcionalmente sustituido; o R205 y R206 pueden formar junto con el nitrogeno al cual están unidos un anillo de 3 a 7 miembros el cual puede contener adicionalmente uno o más heteroátomos seleccionados entre nitrogeno, oxígeno y azufre; X1 se selecciona entre nitrogeno y C-R212; R211, R212 se seleccionan independientemente entre halogeno, hidrogeno, CN, alquilo C1-3 y NO2; R213 se selecciona entre halogeno, haloalquilo, haloalcoxi, -S(O)kCF3, y ûSF5 o forma un anillo con R214; R214 es hidrogeno o puede constituir junto con R213 un grupo de OCF2O, CF2OCF2, CF2OCF2O y CF2CF2O, el cual forma junto con los carbonos a los cuales están unidos un anillo de cinco a seis miembros; y h, k y n se seleccionan independientemente entre 0,1 y 2; y sus sales aceptables la veterinaria, que se usa para preparar una composicion para el control de parásitos en o sobre un animal; compuestos relacionados; y composicion que los contiene.
ARP000106403A 1999-12-02 2000-12-04 Uso de 1-arilpirazoles para preparar una composicion para el control de parasitos en o sobre un animal; compuestos relacionados; y composicion que los contiene AR033504A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US16865899P 1999-12-02 1999-12-02

Publications (1)

Publication Number Publication Date
AR033504A1 true AR033504A1 (es) 2003-12-26

Family

ID=22612402

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000106403A AR033504A1 (es) 1999-12-02 2000-12-04 Uso de 1-arilpirazoles para preparar una composicion para el control de parasitos en o sobre un animal; compuestos relacionados; y composicion que los contiene

Country Status (20)

Country Link
US (4) US6569886B2 (es)
EP (1) EP1237873B1 (es)
JP (1) JP2003516941A (es)
KR (1) KR100816914B1 (es)
CN (2) CN1939909A (es)
AR (1) AR033504A1 (es)
AU (1) AU784798B2 (es)
BR (1) BR0015945A (es)
CA (1) CA2393197C (es)
CO (1) CO5261614A1 (es)
CZ (1) CZ20021898A3 (es)
ES (1) ES2409630T3 (es)
HU (1) HUP0300357A3 (es)
IL (2) IL149856A0 (es)
MX (1) MXPA02005511A (es)
MY (1) MY129771A (es)
PL (1) PL364874A1 (es)
TW (1) TWI290137B (es)
WO (1) WO2001040195A2 (es)
ZA (1) ZA200204336B (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20060115904A (ko) 2003-12-24 2006-11-10 바이엘 크롭사이언스 게엠베하 식물 성장 조절
EA014881B1 (ru) 2004-03-05 2011-02-28 Ниссан Кемикал Индастриз, Лтд. Производные замещенного алкилбензола
US20050234119A1 (en) * 2004-04-16 2005-10-20 Soll Mark D Antiparasitical agents and methods for treating, preventing and controlling external parasites in animals
FR2869905B1 (fr) 2004-05-10 2008-09-05 Sanofi Synthelabo Procede de preparation d'ester de l'acide 1,5-diphenylpyrazole carboxylique.
GB0413970D0 (en) * 2004-06-22 2004-07-28 Syngenta Participations Ag Chemical compounds
UY28617A1 (es) * 2004-11-12 2006-06-30 Popley Pharma Ltda Nuevas composiciones
US7923465B2 (en) 2005-06-02 2011-04-12 Glenmark Pharmaceuticals S.A. Cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation
BRPI0810929B8 (pt) 2007-06-27 2022-12-06 Du Pont uso de um composto de fórmula 1
WO2010059529A2 (en) 2008-11-19 2010-05-27 Merial Limited Compositions comprising an aryl pyrazole and/or a formamidine, methods and uses thereof
US8642636B2 (en) * 2008-11-19 2014-02-04 Merial Limited Dimeric 1-arylpyrazole derivatives for use against ectoparasites, agricultural pests, and household pests
UA108641C2 (uk) 2010-04-02 2015-05-25 Паразитицидна композиція, яка містить чотири активних агенти, та спосіб її застосування
JP5743418B2 (ja) * 2010-04-09 2015-07-01 Oatアグリオ株式会社 新規なピラゾール化合物、その製造方法及び有害生物防除剤
CN104023720B (zh) 2011-11-17 2016-10-26 梅里亚有限公司 包含芳基吡唑和取代咪唑的组合物,其方法和用途
TWI579274B (zh) 2012-04-20 2017-04-21 龍馬躍公司 製備1-芳基-5-烷基吡唑化合物的改良方法
JP5943387B2 (ja) * 2012-10-25 2016-07-05 国立大学法人 名古屋工業大学 新規トリフロン誘導体及びその製造方法
NZ731446A (en) 2014-10-31 2018-09-28 Boehringer Ingelheim Animal Health Usa Inc Parasiticidal composition comprising fipronil
US10766866B2 (en) 2017-10-30 2020-09-08 University Of North Texas Health Science Center At Fort Worth Deterrents for arthropods and marine organisms

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8713768D0 (en) 1987-06-12 1987-07-15 May & Baker Ltd Compositions of matter
US5232940A (en) 1985-12-20 1993-08-03 Hatton Leslie R Derivatives of N-phenylpyrazoles
DE3617554A1 (de) * 1986-05-24 1987-11-26 Bayer Ag 5-oxy(thio)-pyrazol-derivate
DE3625686A1 (de) * 1986-07-30 1988-02-04 Bayer Ag 4-cyano(nitro)-5-oxy(thio)-pyrazol-derivate
CA2004776C (fr) 1988-12-13 2000-04-25 Claude Wakselman Procede de preparation de perfluoroalkylthioethers
US4918085A (en) * 1989-03-02 1990-04-17 Rhone-Poulenc Ag Company Pesticidal 3-cyano-5-alkoxy-1-arylpyrazoles, compositions and use
US5079370A (en) 1989-03-02 1992-01-07 Rhone-Poulenc Ag Company 1-arylpyrazoles
DE4023488A1 (de) 1990-07-24 1992-01-30 Bayer Ag 1-(pyri(mi)dyl-(2)) -5-hydroxy-pyrazol-mikrobizide
GB9306184D0 (en) 1993-03-25 1993-05-19 Zeneca Ltd Heteroaromatic compounds
GB9601128D0 (en) 1995-08-11 1996-03-20 Pfizer Ltd Parasiticidal compounds
FR2739255B1 (fr) 1995-09-29 1998-09-04 Rhone Merieux Composition antiparasitaire pour le traitement et la protection des animaux de compagnie
JPH10152476A (ja) 1996-01-30 1998-06-09 Takeda Chem Ind Ltd 1−アリールピラゾール誘導体、その製造法および用途
GB9625045D0 (en) 1996-11-30 1997-01-22 Pfizer Ltd Parasiticidal compounds
DE19650197A1 (de) 1996-12-04 1998-06-10 Bayer Ag 3-Thiocarbamoylpyrazol-Derivate
TW524667B (en) 1996-12-05 2003-03-21 Pfizer Parasiticidal pyrazoles
US6350771B1 (en) 1996-12-24 2002-02-26 Rhone-Poulenc, Inc. Pesticidal 1-arylpyrazoles
SK285866B6 (sk) 1996-12-24 2007-10-04 Rhone-Poulenc Agro 1-Arylpyrazolové zlúčeniny, pesticídne prostriedky obsahujúce tieto zlúčeniny ako účinné látky a spôsob ničenia škodcov
KR20000062318A (ko) 1996-12-24 2000-10-25 제닌 페트릭 살충성 1-아릴 및 피리딜피라졸 유도체
JPH11246555A (ja) * 1997-10-31 1999-09-14 Sumitomo Chem Co Ltd フッ素置換ベンゾヘテロ環化合物
JP2000169453A (ja) * 1998-09-30 2000-06-20 Mitsubishi Chemicals Corp 1―フェニルピラゾ―ル―3―カルボキサミド誘導体、その中間体およびこれを有効成分とする農薬

Also Published As

Publication number Publication date
US6992099B2 (en) 2006-01-31
US20060020013A1 (en) 2006-01-26
KR20030016204A (ko) 2003-02-26
IL149856A (en) 2009-02-11
JP2003516941A (ja) 2003-05-20
US20070078127A1 (en) 2007-04-05
KR100816914B1 (ko) 2008-03-26
TWI290137B (en) 2007-11-21
AU784798B2 (en) 2006-06-22
WO2001040195A2 (en) 2001-06-07
IL149856A0 (en) 2002-11-10
WO2001040195A3 (en) 2001-11-08
US20030176466A1 (en) 2003-09-18
HUP0300357A3 (en) 2009-01-28
ES2409630T3 (es) 2013-06-27
CA2393197C (en) 2009-03-03
CN1402713A (zh) 2003-03-12
CO5261614A1 (es) 2003-03-31
US6569886B2 (en) 2003-05-27
EP1237873B1 (en) 2013-04-03
HUP0300357A2 (hu) 2003-07-28
MXPA02005511A (es) 2004-09-10
PL364874A1 (en) 2004-12-27
US20020111352A1 (en) 2002-08-15
ZA200204336B (en) 2003-03-20
CZ20021898A3 (cs) 2003-04-16
MY129771A (en) 2007-04-30
BR0015945A (pt) 2002-11-12
US7468381B2 (en) 2008-12-23
AU2839301A (en) 2001-06-12
CN1939909A (zh) 2007-04-04
EP1237873A2 (en) 2002-09-11
CA2393197A1 (en) 2001-06-07

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