AR022470A1 - USE OF PIRAZOL-CARBOXAMIDS - Google Patents

USE OF PIRAZOL-CARBOXAMIDS

Info

Publication number
AR022470A1
AR022470A1 ARP000100428A ARP000100428A AR022470A1 AR 022470 A1 AR022470 A1 AR 022470A1 AR P000100428 A ARP000100428 A AR P000100428A AR P000100428 A ARP000100428 A AR P000100428A AR 022470 A1 AR022470 A1 AR 022470A1
Authority
AR
Argentina
Prior art keywords
carboxamids
pirazol
pyrazolcarboxamides
novel
pyrazolecarboxamides
Prior art date
Application number
ARP000100428A
Other languages
Spanish (es)
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of AR022470A1 publication Critical patent/AR022470A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06—Antianaemics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente invencion se refiere a pirazolcarboxamidas nuevas y conocidas de formulas generales (1) y (2). Además se describe la preparacion de laspirazolcarboxamidas o bien mediante química en fase solida o bien a través de lo nuevos ácidospirazolc arboxílicos. La pirazolcarboxamidas se utilizan comomedicamentos, en especial como medicamentos para el tratamiento de anemias.The present invention relates to novel and known pyrazolecarboxamides of general formulas (1) and (2). In addition, the preparation of pyrazolcarboxamides is described either by solid phase chemistry or through the novel pyroxy arboxylic acids. Pyrazolcarboxamides are used as medications, especially as medicines for the treatment of anemias.

ARP000100428A 1999-02-04 2000-02-01 USE OF PIRAZOL-CARBOXAMIDS AR022470A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19904397A DE19904397A1 (en) 1999-02-04 1999-02-04 Use of pyrazole carboxamides

Publications (1)

Publication Number Publication Date
AR022470A1 true AR022470A1 (en) 2002-09-04

Family

ID=7896339

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000100428A AR022470A1 (en) 1999-02-04 2000-02-01 USE OF PIRAZOL-CARBOXAMIDS

Country Status (8)

Country Link
EP (1) EP1148879A2 (en)
JP (1) JP2002536348A (en)
AR (1) AR022470A1 (en)
AU (1) AU3150300A (en)
CA (1) CA2361636A1 (en)
DE (1) DE19904397A1 (en)
GT (1) GT200000009A (en)
WO (1) WO2000045894A2 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6878729B2 (en) 2001-05-04 2005-04-12 The Procter & Gamble Company Medicinal uses of dihydropyrazoles
CA2579313A1 (en) * 2004-09-17 2006-03-30 Exelixis, Inc. Pyrazole kinase modulators and methods of use as c-kit or fit-3 kinase inhibitors
UY30892A1 (en) 2007-02-07 2008-09-02 Smithkline Beckman Corp AKT ACTIVITY INHIBITORS
UA106740C2 (en) 2009-01-30 2014-10-10 Глаксосмітклайн Ллс Crystalline n-{(1s)-2-amino-l-[(3-fluorophenyl)methyl]ethyl}-5-chloro-4-(4-chloro-l-methyl-1h-pyrazol-5-yl)-2-thiophenecarboxamide hydrochloride
EP4173485A1 (en) * 2021-10-27 2023-05-03 Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. Protein aggregation inhibiting compounds for plant disease control

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH27357A (en) * 1989-09-22 1993-06-21 Fujisawa Pharmaceutical Co Pyrazole derivatives and pharmaceutical compositions comprising the same
US5434178A (en) * 1993-11-30 1995-07-18 G.D. Searle & Co. 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation
WO1997019039A1 (en) * 1995-11-17 1997-05-29 Novartis Ag Solid phase synthesis of heterocyclic compounds and combinatorial compound library
DE19904406A1 (en) * 1999-02-04 2000-08-10 Bayer Ag Substituted pyrazole carboxylic acids
DE19904396A1 (en) * 1999-02-04 2000-08-10 Bayer Ag Substituted pyrazolbenzylamine derivatives

Also Published As

Publication number Publication date
CA2361636A1 (en) 2000-08-10
EP1148879A2 (en) 2001-10-31
AU3150300A (en) 2000-08-25
WO2000045894A3 (en) 2001-04-19
JP2002536348A (en) 2002-10-29
WO2000045894A2 (en) 2000-08-10
GT200000009A (en) 2001-07-27
DE19904397A1 (en) 2000-08-10

Similar Documents

Publication Publication Date Title
SE0001899D0 (en) New compounds
BR0108678A (en) New compounds
SV1999000049A (en) NEW DIETHYDROPYRIMIDINES 2 HETEROCICLICAMENTE SUBSTITUTED REF. READ 32793-SV
BR0113234A (en) Polymorphs of an epothilone analog
BR0213877A (en) Organic compounds
BR0017026A (en) Lipeptides as antibacterial agents
BR0112589A (en) Heteroaryl derivatives and their application as a medicine
BR0211801A (en) 7h-Pyrrolo [2,3-d] pyrimidine derivatives
BR0214469A (en) 17alpha-alkyl-17beta-oxystratrienes and intermediate products for their preparation, application of 17alpha-alkyl-17beta-oxystratrienes for the preparation of medicaments as well as pharmaceutical preparations
MEP39108A (en) Pharmaceutical composition
BRPI0409136A (en) pentacyclic heteroaromatic compound and medicinal use thereof
ATE361084T1 (en) TOPICAL PHARMACEUTICAL COMPOSITIONS CONTAINING PROANTHOCYANIDINS, GLYCYRRHETINIC ACID AND TELMESTEINS FOR THE TREATMENT OF DERMATITIS
BR0115605A (en) Naphthalene derivatives
BR0016467A (en) Lipopeptides as antibacterial agents
AR022469A1 (en) USE OF SUBSTITUTED AND DERIVATIVE ISOXAZOLCARBOXILIC ACIDS AND NEW SUBSTANCES
BR0208887A (en) Dihydro-benzo derivatives [b] [1,4] diazepin-2-one as mglur2 i antagonists
BRPI0414948A (en) pyrazolo-e-imidazo pyrimidine derivatives
BR9910573A (en) Antipicornoviral compounds, preparation and use thereof
BR0015147A (en) Cyclopropanes as cgrp-antagonists, drugs containing said compounds and process for their production
BR9916680A (en) Derivatives of 3,3-biarylpiperidine and 2,2-biarylmorpholine
AR022470A1 (en) USE OF PIRAZOL-CARBOXAMIDS
ATE284878T1 (en) PHARMACEUTICAL COMPOUNDS WITH SEROTONIN RECEPTOR ACTIVITY
MXPA04001655A (en) Ascorbic acid derivatives, methods of synthesis and pharmaceutical use thereof.
HUP0302970A2 (en) Use of amino acids for treating pain, process for their preparation and pharmaceutical compositions containing them
BRPI0412928A (en) dibenzo [b, f] oxepine-10-carboxamides and pharmaceutical uses thereof