AR012109A1 - DERIVATIVES OF BENZENOSULFONAMIDE, ITS PREPARATION, ITS APPLICATION IN THERAPEUTICS AND PHARMACEUTICAL COMPOSITION - Google Patents
DERIVATIVES OF BENZENOSULFONAMIDE, ITS PREPARATION, ITS APPLICATION IN THERAPEUTICS AND PHARMACEUTICAL COMPOSITIONInfo
- Publication number
- AR012109A1 AR012109A1 ARP980101236A ARP980101236A AR012109A1 AR 012109 A1 AR012109 A1 AR 012109A1 AR P980101236 A ARP980101236 A AR P980101236A AR P980101236 A ARP980101236 A AR P980101236A AR 012109 A1 AR012109 A1 AR 012109A1
- Authority
- AR
- Argentina
- Prior art keywords
- group
- benzenosulfonamide
- therapeutics
- derivatives
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/45—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups at least one of the singly-bound nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfonamides
- C07C311/47—Y being a hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D239/08—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
- C07D239/12—Nitrogen atoms not forming part of a nitro radical
- C07D239/14—Nitrogen atoms not forming part of a nitro radical with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to said nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Compuesto de la formula (I) en la cual: A representa un átomo de hidrogeno, un halogeno tal como el fluor, el coloro o el bromo, un grupo ciano, un grupoC1-4 alquilo o un grupo alcoxi; R1 y R2 idénticos o diferentes, repesentan cada uno un átomo de hidrogeno, un grupo C1-C6 alquilo, un grupo C2-6 alquenilo o R1y R2 forman juntos una cadena C2-6 alquileno o C2-6 alquenileno y R3 representa un átomo de hidrogeno o un grupo C1-4 alquilo con la exclusion del clorhidratode 3-bencenosulfonamidoguanidina. Aplicacion en terapéutica.Compound of formula (I) in which: A represents a hydrogen atom, a halogen such as fluorine, color or bromine, a cyano group, a C1-4alkyl group or an alkoxy group; R1 and R2 are identical or different, each representing a hydrogen atom, a C1-C6 alkyl group, a C2-6 alkenyl group or R1 and R2 together form a C2-6 alkylene or C2-6 alkenylene chain and R3 represents an atom of hydrogen or a C1-4 alkyl group with the exclusion of 3-benzenesulfonamidoguanidine hydrochloride. Therapeutic application.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9703394A FR2761061B1 (en) | 1997-03-20 | 1997-03-20 | BENZENESULFONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
Publications (1)
Publication Number | Publication Date |
---|---|
AR012109A1 true AR012109A1 (en) | 2000-09-27 |
Family
ID=9505005
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP980101236A AR012109A1 (en) | 1997-03-20 | 1998-03-19 | DERIVATIVES OF BENZENOSULFONAMIDE, ITS PREPARATION, ITS APPLICATION IN THERAPEUTICS AND PHARMACEUTICAL COMPOSITION |
Country Status (6)
Country | Link |
---|---|
EP (1) | EP0971900A1 (en) |
AR (1) | AR012109A1 (en) |
AU (1) | AU6924198A (en) |
FR (1) | FR2761061B1 (en) |
WO (1) | WO1998042679A1 (en) |
ZA (1) | ZA982358B (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6323231B1 (en) | 2000-02-17 | 2001-11-27 | Abbott Laboratories | Use of α1A adrenoceptor agonists with α1B and α1D antagonism for the treatment of stress urinary incontinence |
DE10106214A1 (en) * | 2001-02-10 | 2002-08-14 | Boehringer Ingelheim Pharma | New alkyl-phenylimino-imidazolidine derivatives for the treatment of urinary incontinence |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2456731A1 (en) * | 1979-05-16 | 1980-12-12 | Choay Sa | Guanidino and amino benzoate(s) and phenyl sulphonate(s) - and related cpds. inhibit protease(s) and have bacteriostatic and fungistatic activity |
FR2549049B1 (en) * | 1983-07-13 | 1986-06-20 | Chauvin Blache Lab | NEW AMIDINES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION |
US4788195A (en) * | 1986-01-13 | 1988-11-29 | American Cyanamid Company | 4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines |
FR2737494B1 (en) * | 1995-08-04 | 1997-08-29 | Synthelabo | BENZENESULFONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
-
1997
- 1997-03-20 FR FR9703394A patent/FR2761061B1/en not_active Expired - Fee Related
-
1998
- 1998-03-17 EP EP98914930A patent/EP0971900A1/en not_active Ceased
- 1998-03-17 WO PCT/FR1998/000530 patent/WO1998042679A1/en not_active Application Discontinuation
- 1998-03-17 AU AU69241/98A patent/AU6924198A/en not_active Abandoned
- 1998-03-19 AR ARP980101236A patent/AR012109A1/en unknown
- 1998-03-19 ZA ZA982358A patent/ZA982358B/en unknown
Also Published As
Publication number | Publication date |
---|---|
ZA982358B (en) | 1998-09-22 |
AU6924198A (en) | 1998-10-20 |
WO1998042679A1 (en) | 1998-10-01 |
EP0971900A1 (en) | 2000-01-19 |
FR2761061B1 (en) | 1999-04-23 |
FR2761061A1 (en) | 1998-09-25 |
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