AP2012006216A0 - Benzimidazole-imidazole derivatives. - Google Patents

Benzimidazole-imidazole derivatives.

Info

Publication number
AP2012006216A0
AP2012006216A0 AP2012006216A AP2012006216A AP2012006216A0 AP 2012006216 A0 AP2012006216 A0 AP 2012006216A0 AP 2012006216 A AP2012006216 A AP 2012006216A AP 2012006216 A AP2012006216 A AP 2012006216A AP 2012006216 A0 AP2012006216 A0 AP 2012006216A0
Authority
AP
ARIPO
Prior art keywords
benzimidazole
imidazole derivatives
imidazole
derivatives
Prior art date
Application number
AP2012006216A
Other languages
English (en)
Inventor
Piere Jean-Marie Raboisson
Stefaan Julien Last
Koen Vandyck
Original Assignee
Janssen R & D Ireland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen R & D Ireland filed Critical Janssen R & D Ireland
Publication of AP2012006216A0 publication Critical patent/AP2012006216A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AP2012006216A 2009-11-04 2010-11-03 Benzimidazole-imidazole derivatives. AP2012006216A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09175015 2009-11-04
EP10154583 2010-02-24
PCT/EP2010/066668 WO2011054834A1 (en) 2009-11-04 2010-11-03 Benzimidazole-imidazole derivatives

Publications (1)

Publication Number Publication Date
AP2012006216A0 true AP2012006216A0 (en) 2012-04-30

Family

ID=43266424

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2012006216A AP2012006216A0 (en) 2009-11-04 2010-11-03 Benzimidazole-imidazole derivatives.

Country Status (22)

Country Link
US (3) US9427428B2 (pt)
EP (1) EP2496572A1 (pt)
JP (1) JP6005515B2 (pt)
KR (1) KR20120091292A (pt)
CN (1) CN102741241B (pt)
AP (1) AP2012006216A0 (pt)
AR (1) AR078888A1 (pt)
AU (1) AU2010317085A1 (pt)
BR (1) BR112012010502A2 (pt)
CA (1) CA2780034C (pt)
CL (1) CL2012001176A1 (pt)
CO (1) CO6531445A2 (pt)
CR (1) CR20120302A (pt)
EA (1) EA022839B1 (pt)
EC (1) ECSP12011867A (pt)
IL (1) IL219087A0 (pt)
MX (1) MX2012005178A (pt)
TW (1) TW201127378A (pt)
UA (1) UA108211C2 (pt)
UY (1) UY32997A (pt)
WO (1) WO2011054834A1 (pt)
ZA (1) ZA201203205B (pt)

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Also Published As

Publication number Publication date
JP2013510119A (ja) 2013-03-21
WO2011054834A1 (en) 2011-05-12
KR20120091292A (ko) 2012-08-17
ECSP12011867A (es) 2012-10-30
JP6005515B2 (ja) 2016-10-12
US20120219594A1 (en) 2012-08-30
US20140107172A1 (en) 2014-04-17
US9433609B2 (en) 2016-09-06
BR112012010502A2 (pt) 2016-03-15
CA2780034C (en) 2018-04-10
CR20120302A (es) 2012-10-25
CO6531445A2 (es) 2012-09-28
US20160340344A1 (en) 2016-11-24
US9427428B2 (en) 2016-08-30
CL2012001176A1 (es) 2012-08-31
AR078888A1 (es) 2011-12-07
UY32997A (es) 2011-05-31
AU2010317085A1 (en) 2012-05-10
CN102741241A (zh) 2012-10-17
EA022839B1 (ru) 2016-03-31
TW201127378A (en) 2011-08-16
UA108211C2 (uk) 2015-04-10
IL219087A0 (en) 2012-06-28
CN102741241B (zh) 2015-05-20
EP2496572A1 (en) 2012-09-12
EA201290260A1 (ru) 2013-12-30
ZA201203205B (en) 2014-10-29
MX2012005178A (es) 2012-06-08
CA2780034A1 (en) 2011-05-12

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