ZA827055B - Substituted ethylamines,processes for their preparation,and pharmaceutical compositions thereof - Google Patents

Substituted ethylamines,processes for their preparation,and pharmaceutical compositions thereof

Info

Publication number: ZA827055B
Authority: ZA; South Africa
Prior art keywords: processes; preparation; pharmaceutical compositions; substituted ethylamines; ethylamines
Prior art date: 1981-09-28

Application number

ZA827055A

Other languages

English (en)

Inventor

Claus Schneider

Gerhard Walther

Karl-Heinz Weber

Wolf Dietrich Bechtel

Karin Boeke-Kuhn

Original Assignee

Boehringer Ingelheim Int

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-09-28

Filing date

1982-09-27

Publication date

1984-05-30

1982-09-27 Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int

1984-05-30 Publication of ZA827055B publication Critical patent/ZA827055B/xx

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, ***e
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/65—One oxygen atom attached in position 3 or 5
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/68—One oxygen atom attached in position 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/70—Sulfur atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Psychiatry (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Biomedical Technology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

ZA827055A 1981-09-28 1982-09-27 Substituted ethylamines,processes for their preparation,and pharmaceutical compositions thereof ZA827055B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19813138550 DE3138550A1 (de)	1981-09-28	1981-09-28	Substituierte 2-phenyl-2-(pyridyloxy)-ethylamine und isostere verbindungen, verfahren zu ihrer herstellung und verwendung

Publications (1)

Publication Number	Publication Date
ZA827055B true ZA827055B (en)	1984-05-30

Family

ID=6142812

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA827055A ZA827055B (en)	1981-09-28	1982-09-27	Substituted ethylamines,processes for their preparation,and pharmaceutical compositions thereof

Country Status (21)

Country	Link
US (1)	US4666910A (xx)
EP (1)	EP0075752B1 (xx)
JP (1)	JPS5869865A (xx)
KR (1)	KR880002705B1 (xx)
AR (1)	AR231534A1 (xx)
AT (1)	ATE18551T1 (xx)
AU (1)	AU550614B2 (xx)
CA (1)	CA1171086A (xx)
DE (2)	DE3138550A1 (xx)
DK (1)	DK156718C (xx)
ES (1)	ES515972A0 (xx)
FI (1)	FI78074C (xx)
GB (1)	GB2106902B (xx)
GR (1)	GR77657B (xx)
IE (1)	IE53959B1 (xx)
IL (1)	IL66870A (xx)
NO (1)	NO159999C (xx)
NZ (1)	NZ202015A (xx)
PH (1)	PH23219A (xx)
PT (1)	PT75611B (xx)
ZA (1)	ZA827055B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8320699D0 (en) *	1983-08-01	1983-09-01	Wellcome Found	Ethylenediamines
GB0004153D0 (en) *	2000-02-23	2000-04-12	Astrazeneca Uk Ltd	Novel use
GB0004152D0 (en)	2000-02-23	2000-04-12	Astrazeneca Uk Ltd	Novel compounds
GB0004151D0 (en) *	2000-02-23	2000-04-12	Astrazeneca Uk Ltd	Novel use
AR035700A1 (es) *	2001-05-08	2004-06-23	Astrazeneca Ab	Derivados de arilheteroalquilamina, composicion farmaceutica, usos de estos derivados para la fabricacion de medicamentos, metodos de tratamiento, y proceso para la preparacion de estos derivados
SE0102641D0 (sv) *	2001-07-31	2001-07-31	Astrazeneca Ab	Novel compounds
SE0102640D0 (sv) *	2001-07-31	2001-07-31	Astrazeneca Ab	Novel compounds
SE0102639D0 (sv) *	2001-07-31	2001-07-31	Astrazeneca Ab	Novel compounds
GB0219154D0 (en) *	2002-08-16	2002-09-25	Pfizer Ltd	Diaryl compounds
US6800652B2 (en)	2002-08-16	2004-10-05	Pfizer Inc.	Diaryl compounds
SE0203304D0 (sv) *	2002-11-07	2002-11-07	Astrazeneca Ab	Novel Coumpounds
KR20060110288A (ko) *	2003-10-09	2006-10-24	밀레니엄 파머슈티컬스 인코퍼레이티드	인자 ｘａ 의 저해제로서의 티오에테르-치환 벤즈아미드

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2734846A (en) *		1956-02-14		Aqueous suspension of procaine penicil-
US2734845A (en) *		1956-02-14		Aqueous suspension of procaine penicil-
FR1511398A (fr) *	1966-02-16	1968-01-26	Takeda Chemical Industries Ltd	Procédé de préparation de nouveaux dérivés de picoline
BE790592A (xx) *	1971-10-28	1973-04-26	Oreal
US4011324A (en) *	1976-01-20	1977-03-08	Pfizer Inc.	Esters and amides of pyrimido[4,5-b]quinolin-4(3H)-one-2-carboxylic acids as antiulcer agents
JPS53141271A (en) *	1977-05-13	1978-12-08	Yamanouchi Pharmaceut Co Ltd	Heterocyclic compounds and process for their preparation

1981
- 1981-09-28 DE DE19813138550 patent/DE3138550A1/de not_active Withdrawn
1982
- 1982-09-06 DE DE8282108196T patent/DE3269839D1/de not_active Expired
- 1982-09-06 EP EP82108196A patent/EP0075752B1/de not_active Expired
- 1982-09-06 AT AT82108196T patent/ATE18551T1/de not_active IP Right Cessation
- 1982-09-22 FI FI823246A patent/FI78074C/fi not_active IP Right Cessation
- 1982-09-24 AR AR290759A patent/AR231534A1/es active
- 1982-09-24 IL IL66870A patent/IL66870A/xx unknown
- 1982-09-27 AU AU88738/82A patent/AU550614B2/en not_active Ceased
- 1982-09-27 NZ NZ202015A patent/NZ202015A/en unknown
- 1982-09-27 ZA ZA827055A patent/ZA827055B/xx unknown
- 1982-09-27 ES ES515972A patent/ES515972A0/es active Granted
- 1982-09-27 JP JP57168221A patent/JPS5869865A/ja active Granted
- 1982-09-27 PT PT75611A patent/PT75611B/pt not_active IP Right Cessation
- 1982-09-27 KR KR8204342A patent/KR880002705B1/ko active
- 1982-09-27 CA CA000412268A patent/CA1171086A/en not_active Expired
- 1982-09-27 DK DK428582A patent/DK156718C/da not_active IP Right Cessation
- 1982-09-27 GB GB08227449A patent/GB2106902B/en not_active Expired
- 1982-09-27 IE IE2330/82A patent/IE53959B1/en not_active IP Right Cessation
- 1982-09-27 NO NO823253A patent/NO159999C/no unknown
- 1982-09-28 GR GR69383A patent/GR77657B/el unknown
1984
- 1984-08-28 US US06/645,007 patent/US4666910A/en not_active Expired - Fee Related
1985
- 1985-03-07 PH PH31952A patent/PH23219A/en unknown

Also Published As

Publication number	Publication date
EP0075752A2 (de)	1983-04-06
IL66870A (en)	1986-02-28
DK428582A (da)	1983-03-29
FI823246A0 (fi)	1982-09-22
JPS5869865A (ja)	1983-04-26
DK156718C (da)	1990-03-05
US4666910A (en)	1987-05-19
NO159999B (no)	1988-11-21
AR231534A1 (es)	1984-12-28
GB2106902A (en)	1983-04-20
ES8308543A1 (es)	1983-09-16
DE3269839D1 (en)	1986-04-17
NZ202015A (en)	1985-11-08
KR840001555A (ko)	1984-05-07
EP0075752A3 (en)	1984-03-21
PH23219A (en)	1989-06-06
PT75611A (de)	1982-10-01
IE822330L (en)	1983-03-28
DE3138550A1 (de)	1983-04-07
FI78074B (fi)	1989-02-28
AU8873882A (en)	1983-04-14
FI823246L (fi)	1983-03-29
AU550614B2 (en)	1986-03-27
NO159999C (no)	1989-03-01
CA1171086A (en)	1984-07-17
JPH0316952B2 (xx)	1991-03-06
EP0075752B1 (de)	1986-03-12
FI78074C (fi)	1989-06-12
ATE18551T1 (de)	1986-03-15
NO823253L (no)	1983-03-29
PT75611B (de)	1985-12-09
GR77657B (xx)	1984-09-25
IE53959B1 (en)	1989-04-26
IL66870A0 (en)	1982-12-31
DK156718B (da)	1989-09-25
ES515972A0 (es)	1983-09-16
GB2106902B (en)	1985-08-07
KR880002705B1 (ko)	1988-12-26

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IL75400A0 (en)	1985-10-31	Dialkoxypyridines,processes for the preparation thereof and pharmaceutical compositions containing the same
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IL72085A0 (en)	1984-10-31	13alpha-alkylylgonanes,processes for their preparation and pharmaceutical compositions containing the same
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DE3275296D1 (en)	1987-03-05	Azabicyclo-(3,3,1)-nonylbenzamide derivatives, processes for their preparation, and pharmaceutical compositions containing them
ZM9283A1 (en)	1984-06-21	Substituted phenylsulfonyloxybenzimidazolecarbamates,processes for their preparation and pharmaceutical compositions containing the same
ZA827055B (en)	1984-05-30	Substituted ethylamines,processes for their preparation,and pharmaceutical compositions thereof
DE3260490D1 (en)	1984-09-06	Secondary amines, their preparation, pharmaceutical compositions containing them and their use
ZA822388B (en)	1983-02-23	Secondary amines, processes for their preparation, and pharmaceutical compositions containing them
DE3273629D1 (en)	1986-11-13	New ribofuranuronic acid derivatives, processes for preparation thereof and pharmaceutical compositions thereof
IL70488A0 (en)	1984-03-30	Fluoromethylthiooxacephalosporins,processes for the preparation thereof and pharmaceutical and veterinary compositions containing the same
IL66227A0 (en)	1982-11-30	Amidobenzamides and their salts,their preparation and pharmaceutical compositions containing them
IL64880A0 (en)	1982-03-31	Imidazoline derivatives,processes for the preparation thereof and pharmaceutical compositions containing them
ZA825275B (en)	1984-03-28	Benzotriazoles,processes for their preparation,and pharmaceutical compositions thereof
ZA823919B (en)	1984-02-29	Diazepin-10-ones,processes for their preparation,and pharmaceutical compositions thereof
IL65177A0 (en)	1982-05-31	Fluoroprostacylins,their preparation and pharmaceutical compositions containing them
DE3060079D1 (en)	1982-01-21	Spiro-quinolylhydantoins, process for their preparation and pharmaceutical compositions thereof
ZA824437B (en)	1984-02-29	Substituted pyrimidines,processes for their preparation and pharmaceutical compositions thereof
EP0018077A3 (en)	1980-11-26	Phenylmorphans, processes for their preparation, pharmaceutical compositions containing them, and 4-phenyl-tetrahydro-pyridines
DE3067174D1 (en)	1984-04-26	Tetrahydro-fluorene compounds, processes for their preparation and pharmaceutical compositions thereof