ZA813255B - Triazoloquinoxalin-4-ones - Google Patents
Triazoloquinoxalin-4-onesInfo
- Publication number
- ZA813255B ZA813255B ZA00813255A ZA813255A ZA813255B ZA 813255 B ZA813255 B ZA 813255B ZA 00813255 A ZA00813255 A ZA 00813255A ZA 813255 A ZA813255 A ZA 813255A ZA 813255 B ZA813255 B ZA 813255B
- Authority
- ZA
- South Africa
- Prior art keywords
- triazoloquinoxalin
- ones
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
- C07D241/38—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
- C07D241/40—Benzopyrazines
- C07D241/44—Benzopyrazines with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/151,220 US4354027A (en) | 1980-05-19 | 1980-05-19 | Triazoloquinoxalin-4-ones |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA813255B true ZA813255B (en) | 1982-06-30 |
Family
ID=22537818
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA00813255A ZA813255B (en) | 1980-05-19 | 1981-05-15 | Triazoloquinoxalin-4-ones |
Country Status (12)
Country | Link |
---|---|
US (1) | US4354027A (fi) |
EP (1) | EP0040401B1 (fi) |
JP (1) | JPS5718681A (fi) |
AU (1) | AU538782B2 (fi) |
CA (1) | CA1176634A (fi) |
DE (1) | DE3162761D1 (fi) |
DK (1) | DK214981A (fi) |
ES (1) | ES502747A0 (fi) |
FI (1) | FI71148C (fi) |
NO (1) | NO811646L (fi) |
NZ (1) | NZ197101A (fi) |
ZA (1) | ZA813255B (fi) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3141304A (en) * | 1960-11-14 | 1964-07-21 | Jefferson Chem Co Inc | Soil stabilization by atactic polypropylene coating |
US4507300A (en) * | 1980-05-09 | 1985-03-26 | Usv Pharmaceutical Corporation | Pyridotriazolopyrazine-diones for treating allergy |
US4400382A (en) * | 1980-05-09 | 1983-08-23 | Usv Pharmaceutical Corporation | Thiazoloquinoxalin-1,4-diones for treating allergy |
US5153196A (en) * | 1991-06-05 | 1992-10-06 | Eli Lilly And Company | Excitatory amino acid receptor antagonists and methods for the use thereof |
US5196421A (en) * | 1991-06-05 | 1993-03-23 | Eli Lilly And Company | Excitatory amino acid receptor antagonists in methods for the use thereof |
DK162491D0 (da) * | 1991-09-20 | 1991-09-20 | Novo Nordisk As | Heterocycliske forbindelser, deres fremstilling og farmaceutiske praeparater indeholdende forbindelserne |
FR2696466B1 (fr) * | 1992-10-02 | 1994-11-25 | Rhone Poulenc Rorer Sa | Dérivés de 5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, leur préparation et les médicaments les contenant. |
DK31093D0 (fi) * | 1993-03-19 | 1993-03-19 | Novo Nordisk As | |
FR2717814B1 (fr) * | 1994-03-28 | 1996-04-26 | Rhone Poulenc Rorer Sa | Dérivés de 1,2,4-triazolo(4,3-a)pyrazine-4-one, leur préparation et les médicaments les contenant. |
FR2717813B1 (fr) * | 1994-03-28 | 1996-05-10 | Rhone Poulenc Rorer Sa | Dérivés d'imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, leur préparation et les médicaments les contenant . |
FR2717812B1 (fr) * | 1994-03-28 | 1996-05-10 | Rhone Poulenc Rorer Sa | Indeno[1,2-e]pyrazine-4-ones, leur préparation et les médicaments les contenant. |
FR2717805B1 (fr) * | 1994-03-28 | 1996-05-10 | Rhone Poulenc Rorer Sa | Dérivés de 5H-indeno[1,2-b]pyrazine-2,3-dione, leur préparation et les médicaments les contenant . |
DK0781282T3 (da) * | 1994-09-16 | 2000-02-28 | Novo Nordisk As | [1,2]triazolo[4,3-a]quinoxalinonderivater, deres fremstilling og anvendelse |
HUT76810A (en) * | 1994-09-16 | 1997-11-28 | Novo Nordisk As | [1,2,4]triazolo[4,3-a]quinoxalinone derivatives, process for their preparation and pharmaceutical compositions containing them |
FR2726275B1 (fr) * | 1994-11-02 | 1996-12-06 | Rhone Poulenc Rorer Sa | Spiro heterocycle-imidazo(1,2-a)indeno(1,2-e)pyrazine)-4'- ones, leur preparation et les medicaments les contenants |
US5679680A (en) * | 1995-02-16 | 1997-10-21 | Warner-Lambert Company | α-substituted hydrazides having calpain inhibitory activity |
CN101553491B (zh) * | 2006-12-13 | 2013-05-29 | Aska制药株式会社 | 喹喔啉衍生物 |
AR107456A1 (es) | 2016-02-12 | 2018-05-02 | Lilly Co Eli | Inhibidor de pde1 |
JOP20170164A1 (ar) | 2016-08-25 | 2019-01-30 | Lilly Co Eli | مشتق ترايازولو بيرازينون مفيد كمثبط لـ pde1 بشري |
AR112457A1 (es) | 2017-08-02 | 2019-10-30 | Lilly Co Eli | Derivados de [1,2,4]triazolo[4,3-a]pirazin-6(5h)-ona |
AR112346A1 (es) | 2017-08-10 | 2019-10-16 | Lilly Co Eli | Derivados de [1,2,4]triazolo |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1301228A (fi) * | 1971-03-04 | 1972-12-29 | Ici Ltd | |
JPS50116498A (fi) * | 1974-02-27 | 1975-09-11 | ||
US3979387A (en) * | 1975-06-10 | 1976-09-07 | Eli Lilly And Company | 4,5-Dihydrotetrazolo(1,5-A)quinoxalines |
-
1980
- 1980-05-19 US US06/151,220 patent/US4354027A/en not_active Expired - Lifetime
-
1981
- 1981-05-12 CA CA000377439A patent/CA1176634A/en not_active Expired
- 1981-05-13 AU AU70544/81A patent/AU538782B2/en not_active Ceased
- 1981-05-13 EP EP81103695A patent/EP0040401B1/en not_active Expired
- 1981-05-13 DE DE8181103695T patent/DE3162761D1/de not_active Expired
- 1981-05-14 NZ NZ197101A patent/NZ197101A/en unknown
- 1981-05-14 DK DK214981A patent/DK214981A/da not_active Application Discontinuation
- 1981-05-14 NO NO811646A patent/NO811646L/no unknown
- 1981-05-14 ES ES502747A patent/ES502747A0/es active Granted
- 1981-05-15 JP JP7239281A patent/JPS5718681A/ja active Pending
- 1981-05-15 ZA ZA00813255A patent/ZA813255B/xx unknown
- 1981-05-15 FI FI811504A patent/FI71148C/fi not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
DE3162761D1 (en) | 1984-04-26 |
NZ197101A (en) | 1984-03-16 |
ES8203375A1 (es) | 1982-04-01 |
EP0040401A1 (en) | 1981-11-25 |
NO811646L (no) | 1981-11-20 |
DK214981A (da) | 1981-11-20 |
AU7054481A (en) | 1981-11-19 |
US4354027A (en) | 1982-10-12 |
AU538782B2 (en) | 1984-08-30 |
CA1176634A (en) | 1984-10-23 |
FI71148C (fi) | 1986-11-24 |
FI811504L (fi) | 1981-11-20 |
EP0040401B1 (en) | 1984-03-21 |
ES502747A0 (es) | 1982-04-01 |
JPS5718681A (en) | 1982-01-30 |
FI71148B (fi) | 1986-08-14 |
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