ZA79778B - New propanone derivatives,process for producing thereof and pharmaceutical composition containing this derivative as active ingredient - Google Patents
New propanone derivatives,process for producing thereof and pharmaceutical composition containing this derivative as active ingredientInfo
- Publication number
- ZA79778B ZA79778B ZA79778A ZA79778A ZA79778B ZA 79778 B ZA79778 B ZA 79778B ZA 79778 A ZA79778 A ZA 79778A ZA 79778 A ZA79778 A ZA 79778A ZA 79778 B ZA79778 B ZA 79778B
- Authority
- ZA
- South Africa
- Prior art keywords
- derivative
- producing
- new
- pharmaceutical composition
- active ingredient
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/10—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms
- C07D295/104—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/108—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/10—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms
- C07D295/104—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/58—Radicals substituted by nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP1930378A JPS54125630A (en) | 1978-02-22 | 1978-02-22 | Novel propanone derivative*its manufacture and medical composition containing it as active component |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA79778B true ZA79778B (en) | 1980-03-26 |
Family
ID=11995644
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA79778A ZA79778B (en) | 1978-02-22 | 1979-02-20 | New propanone derivatives,process for producing thereof and pharmaceutical composition containing this derivative as active ingredient |
Country Status (17)
Country | Link |
---|---|
US (2) | US4277474A (xx) |
EP (1) | EP0004000B2 (xx) |
JP (1) | JPS54125630A (xx) |
AR (1) | AR221080A1 (xx) |
AT (1) | AT372086B (xx) |
AU (1) | AU530412B2 (xx) |
BR (1) | BR7901124A (xx) |
CA (1) | CA1120487A (xx) |
DE (1) | DE2967306D1 (xx) |
DK (1) | DK77679A (xx) |
ES (1) | ES477882A1 (xx) |
IL (1) | IL56664A (xx) |
MX (1) | MX5399E (xx) |
NZ (1) | NZ189721A (xx) |
PH (1) | PH15114A (xx) |
SU (1) | SU873873A3 (xx) |
ZA (1) | ZA79778B (xx) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CS184021B1 (en) * | 1973-07-19 | 1978-07-31 | Jan Drkal | Rolling machine for cross tapered rolling |
DE3019497A1 (de) * | 1980-05-22 | 1981-11-26 | Bayer Ag, 5090 Leverkusen | Aminopropiophenon-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide |
JPS5944371A (ja) * | 1982-09-07 | 1984-03-12 | Dainippon Pharmaceut Co Ltd | 1―フエニル―2―メチル―3―(1―ピロリジニル)―1―プロパノン誘導体 |
JPS59190981A (ja) * | 1983-04-15 | 1984-10-29 | Hokuriku Seiyaku Co Ltd | 3−ピロリジノ置換プロピオフエノン誘導体 |
JPS59190980A (ja) * | 1983-04-15 | 1984-10-29 | Hokuriku Seiyaku Co Ltd | 2’−クロロ−3−アミノ−2−メチル置換プロピオフエノン誘導体 |
HU33131A (xx) * | 1984-01-26 | 1984-10-29 | ||
NL8400508A (nl) * | 1984-02-17 | 1985-09-16 | Philips Nv | Audiotransmissiecircuit met als lijnspanningsstabilisator uitgevoerde zendversterker. |
DE3436450A1 (de) * | 1984-10-05 | 1986-04-10 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von p-aminoethylketonen |
US5057535A (en) * | 1985-04-11 | 1991-10-15 | Nippon Kayaku Kabushiki Kaisha | Derivatives of an aminoketone |
DE3688917T2 (de) * | 1985-04-11 | 1994-02-10 | Nippon Kayaku Kk | Derivate eines Aminoketons. |
US5103022A (en) * | 1985-04-11 | 1992-04-07 | Nippon Kayaku Kabushiki Kaisha | Process for producing an optically active aminoketone derivative |
US4650692A (en) * | 1985-11-01 | 1987-03-17 | Ashland Oil, Inc. | Metal-sulfonate/piperidine derivative combination protective coatings |
JPH03115267A (ja) * | 1989-09-28 | 1991-05-16 | Maruho Kk | プロピオフエノン誘導体、その製造方法、それを含む中枢性筋弛緩剤および抗痙攣剤 |
WO1999003835A1 (fr) * | 1997-07-18 | 1999-01-28 | Nippon Kayaku Kabushiki Kaisha | Derives cetoniques aromatiques et leurs utilisations |
WO1999045914A1 (fr) * | 1998-03-13 | 1999-09-16 | Maruho Kabushikikaisha | Derive alkylamine et agent anesthesique utilisant ce derive |
GB9808447D0 (en) | 1998-04-18 | 1998-06-17 | Zeneca Ltd | Process |
CN1869002A (zh) * | 2005-05-27 | 2006-11-29 | 中国科学院上海药物研究所 | 一类非甾体雄激素受体调节剂、其制备方法和用途 |
WO2007136790A2 (en) | 2006-05-18 | 2007-11-29 | Mannkind Corporation | Intracellular kinase inhibitors |
JP4827986B2 (ja) | 2007-06-08 | 2011-11-30 | マンカインド コーポレ−ション | IRE−1αインヒビター |
WO2018013213A1 (en) * | 2016-05-13 | 2018-01-18 | The Trustees Of Columbia University In The City Of New York | Compounds for reducing c-myc in c-myc overexpressing cancers |
IT201600098338A1 (it) * | 2016-09-30 | 2018-03-30 | Univ Degli Studi Padova | Composti 1-fenilpropanone e loro impiego |
Family Cites Families (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2282907A (en) * | 1941-05-01 | 1942-05-12 | Us Rubber Co | Parasiticide |
US2771391A (en) * | 1953-08-20 | 1956-11-20 | Allied Lab Inc | Physiologically active p-alkoxy-beta-piperidinopropiophenones causing cns depressantand anesthetic effects in animals |
BE623404A (xx) * | 1960-04-26 | |||
FR1301863A (fr) * | 1961-06-29 | 1962-08-24 | Science Union & Cie | Aminocétones substituées et leurs procédés de préparation |
US3151124A (en) * | 1961-11-20 | 1964-09-29 | Ciba Geigy Corp | Alpha oxy-beta alkyl-gamma tertiary amino-alpha phenyl propanes |
GB1142474A (en) * | 1965-03-24 | 1969-02-05 | Ferrosan Ab | Production of piperidino-butyrophenones |
GB1115992A (en) * | 1965-03-26 | 1968-06-06 | Lafon Labor | Improvements in or relating to n-piperidino-alkoxyacetophenones |
US3417087A (en) * | 1965-12-27 | 1968-12-17 | Research Corp | 3(aminopropionyl)benzothiophenes |
US3903092A (en) * | 1966-03-02 | 1975-09-02 | Aspro Nicholas Ltd | 2-Tertiaryamino-1-(benzo{8 b{9 thienyl)ethanols |
US3495015A (en) * | 1967-11-17 | 1970-02-10 | American Cyanamid Co | Treatment of depression with 3-substituted amino-2-phenylpropiophenones |
GB1213963A (en) * | 1968-03-28 | 1970-11-25 | Richter Gedeon Vegyeszet | Aromatic amino ketones |
US3637712A (en) * | 1970-01-26 | 1972-01-25 | Bristol Myers Co | Piperidylpropanol compounds |
FR2138488A1 (en) * | 1971-05-27 | 1973-01-05 | Lipha | 1-(5-indanyl)-omega-aminoalkanes - with tranquillizing activity |
FR2150594A1 (en) * | 1971-08-27 | 1973-04-13 | Delalande Sa | Omega-amino-1,2-diphenyl-1-alkanones - with analgesic antiinflammatory anti-ulcer,bronchodilator,spasmolytic and hypotensive |
HU166289B (xx) * | 1973-01-15 | 1975-02-28 | ||
US3995047A (en) * | 1973-12-14 | 1976-11-30 | Eisai Co., Ltd. | Propiophenone derivatives in the treatment of pathological muscular conditions |
JPS5527914B2 (xx) * | 1973-12-14 | 1980-07-24 | ||
FR2305981A1 (fr) * | 1975-04-03 | 1976-10-29 | Innothera Lab Sa | Nouvelles benzothienyl aminoethyl cetones, leur procede de preparation et leur application en therapeutique |
DD124521A1 (xx) * | 1976-03-16 | 1977-03-02 |
-
1978
- 1978-02-22 JP JP1930378A patent/JPS54125630A/ja active Granted
-
1979
- 1979-02-14 IL IL56664A patent/IL56664A/xx unknown
- 1979-02-20 ZA ZA79778A patent/ZA79778B/xx unknown
- 1979-02-20 ES ES477882A patent/ES477882A1/es not_active Expired
- 1979-02-21 NZ NZ189721A patent/NZ189721A/xx unknown
- 1979-02-21 CA CA000322031A patent/CA1120487A/en not_active Expired
- 1979-02-21 BR BR7901124A patent/BR7901124A/pt unknown
- 1979-02-21 PH PH22223A patent/PH15114A/en unknown
- 1979-02-21 MX MX797729U patent/MX5399E/es unknown
- 1979-02-21 AT AT0133279A patent/AT372086B/de not_active IP Right Cessation
- 1979-02-22 AU AU44517/79A patent/AU530412B2/en not_active Ceased
- 1979-02-22 SU SU792732452A patent/SU873873A3/ru active
- 1979-02-22 EP EP79100528A patent/EP0004000B2/en not_active Expired
- 1979-02-22 AR AR275590A patent/AR221080A1/es active
- 1979-02-22 DK DK77679A patent/DK77679A/da not_active Application Discontinuation
- 1979-02-22 DE DE7979100528T patent/DE2967306D1/de not_active Expired
- 1979-09-27 US US06/079,460 patent/US4277474A/en not_active Expired - Lifetime
-
1985
- 1985-01-24 US US06/693,838 patent/US4563454A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
SU873873A3 (ru) | 1981-10-15 |
NZ189721A (en) | 1981-11-19 |
DE2967306D1 (en) | 1985-01-10 |
AU530412B2 (en) | 1983-07-14 |
MX5399E (es) | 1983-07-12 |
EP0004000A1 (en) | 1979-09-19 |
AU4451779A (en) | 1979-08-30 |
US4563454A (en) | 1986-01-07 |
ES477882A1 (es) | 1979-10-16 |
US4277474A (en) | 1981-07-07 |
IL56664A0 (en) | 1979-05-31 |
JPS6256143B2 (xx) | 1987-11-24 |
AR221080A1 (es) | 1980-12-30 |
ATA133279A (de) | 1983-01-15 |
EP0004000B2 (en) | 1988-06-15 |
JPS54125630A (en) | 1979-09-29 |
EP0004000B1 (en) | 1984-11-28 |
CA1120487A (en) | 1982-03-23 |
DK77679A (da) | 1979-08-23 |
BR7901124A (pt) | 1979-09-11 |
IL56664A (en) | 1984-01-31 |
AT372086B (de) | 1983-08-25 |
PH15114A (en) | 1982-08-10 |
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