ZA722260B - 1-substituted-6-phenyl-4h-s-triazolo(3,4-a)(1,4)-benzodiazepines and process - Google Patents

1-substituted-6-phenyl-4h-s-triazolo(3,4-a)(1,4)-benzodiazepines and process

Info

Publication number
ZA722260B
ZA722260B ZA722260A ZA722260A ZA722260B ZA 722260 B ZA722260 B ZA 722260B ZA 722260 A ZA722260 A ZA 722260A ZA 722260 A ZA722260 A ZA 722260A ZA 722260 B ZA722260 B ZA 722260B
Authority
ZA
South Africa
Prior art keywords
benzodiazepines
triazolo
phenyl
substituted
Prior art date
Application number
ZA722260A
Other languages
English (en)
Inventor
J Hester
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of ZA722260B publication Critical patent/ZA722260B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ZA722260A 1971-04-28 1972-04-04 1-substituted-6-phenyl-4h-s-triazolo(3,4-a)(1,4)-benzodiazepines and process ZA722260B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/138,288 US4141902A (en) 1971-04-28 1971-04-28 1-Halomethyl-6-phenyl-4H-s-[4,3-a][1,4]benzodiazepines

Publications (1)

Publication Number Publication Date
ZA722260B true ZA722260B (en) 1973-02-28

Family

ID=22481351

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA722260A ZA722260B (en) 1971-04-28 1972-04-04 1-substituted-6-phenyl-4h-s-triazolo(3,4-a)(1,4)-benzodiazepines and process

Country Status (10)

Country Link
US (1) US4141902A (de)
JP (1) JPS5521751B1 (de)
AU (1) AU456549B2 (de)
BE (1) BE782848A (de)
CH (1) CH581655A5 (de)
DE (1) DE2220612A1 (de)
FR (1) FR2134586B1 (de)
GB (1) GB1331917A (de)
NL (1) NL7205783A (de)
ZA (1) ZA722260B (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4902794A (en) * 1971-04-28 1990-02-20 The Upjohn Company Triazolo-benzodiazepines
US3892763A (en) * 1974-03-21 1975-07-01 Upjohn Co 1-Propynylaminomethyl-6-phenyl-4H-s-triazolo{8 4,3-a{9 {8 1,4{9 benzodiazepines
US3910946A (en) * 1974-09-12 1975-10-07 Upjohn Co 4H-Imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines
US4021441A (en) 1975-04-07 1977-05-03 The Upjohn Company 1-[(Allylamino)-methyl]-6-phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines
US4455307A (en) * 1982-01-04 1984-06-19 The Upjohn Company Antihypertensive use of triazolobenzodiazepines
US4663454A (en) * 1985-04-17 1987-05-05 The Upjohn Company Process to prepare α-chloroalprazolam

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1955349U (de) 1966-09-22 1967-02-09 Adelbert Stephan Grossmengenduese.
PH9315A (en) * 1968-11-05 1975-08-22 K Meguro Triazolo(4,3-a)(1,4)benzodiazepine derivatives
US3987052A (en) 1969-03-17 1976-10-19 The Upjohn Company 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines
FR2022598A1 (en) * 1969-11-04 1970-07-31 Pakeda Chemical Ind Sedative chloro-phenyl-triazolobenzodiazepines
JPS4932874B1 (de) * 1970-12-11 1974-09-03

Also Published As

Publication number Publication date
CH581655A5 (de) 1976-11-15
NL7205783A (de) 1972-10-31
DE2220612A1 (de) 1972-11-09
FR2134586B1 (de) 1975-10-17
FR2134586A1 (de) 1972-12-08
BE782848A (fr) 1972-10-30
GB1331917A (en) 1973-09-26
US4141902A (en) 1979-02-27
JPS5521751B1 (de) 1980-06-12
AU456549B2 (en) 1974-12-04
AU4101572A (en) 1973-10-18

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