ZA201005318B - Macrocyclic serine protease inhibitors - Google Patents

Macrocyclic serine protease inhibitors

Info

Publication number
ZA201005318B
ZA201005318B ZA2010/05318A ZA201005318A ZA201005318B ZA 201005318 B ZA201005318 B ZA 201005318B ZA 2010/05318 A ZA2010/05318 A ZA 2010/05318A ZA 201005318 A ZA201005318 A ZA 201005318A ZA 201005318 B ZA201005318 B ZA 201005318B
Authority
ZA
South Africa
Prior art keywords
protease inhibitors
serine protease
macrocyclic serine
macrocyclic
inhibitors
Prior art date
Application number
ZA2010/05318A
Inventor
Christophe Claude Parsy
Francois-Rene Alexandre
Dominique Surleraux
Michel Derock
Frederic Leroy
Original Assignee
Idenix Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idenix Pharmaceuticals Inc filed Critical Idenix Pharmaceuticals Inc
Publication of ZA201005318B publication Critical patent/ZA201005318B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
ZA2010/05318A 2008-02-04 2010-07-26 Macrocyclic serine protease inhibitors ZA201005318B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US2608608P 2008-02-04 2008-02-04
US8386708P 2008-07-25 2008-07-25
PCT/US2009/000688 WO2009099596A2 (en) 2008-02-04 2009-02-03 Macrocyclic serine protease inhibitors

Publications (1)

Publication Number Publication Date
ZA201005318B true ZA201005318B (en) 2011-10-26

Family

ID=40568607

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA2010/05318A ZA201005318B (en) 2008-02-04 2010-07-26 Macrocyclic serine protease inhibitors

Country Status (22)

Country Link
US (2) US8003659B2 (en)
EP (1) EP2250174B1 (en)
JP (1) JP5574982B2 (en)
KR (1) KR20100118991A (en)
CN (1) CN101977915B (en)
AR (1) AR070413A1 (en)
AU (1) AU2009210789B2 (en)
BR (1) BRPI0908021A2 (en)
CA (1) CA2712971A1 (en)
CO (1) CO6501153A2 (en)
CR (1) CR11618A (en)
EC (1) ECSP10010413A (en)
ES (1) ES2437147T3 (en)
HK (1) HK1144198A1 (en)
IL (1) IL207333A0 (en)
MX (1) MX2010008523A (en)
NI (1) NI201000136A (en)
NZ (1) NZ587133A (en)
RU (1) RU2490272C2 (en)
TW (1) TW200936131A (en)
WO (1) WO2009099596A2 (en)
ZA (1) ZA201005318B (en)

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