ZA200805028B - Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor Xla inhibitors - Google Patents
Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor Xla inhibitorsInfo
- Publication number
- ZA200805028B ZA200805028B ZA200805028A ZA200805028A ZA200805028B ZA 200805028 B ZA200805028 B ZA 200805028B ZA 200805028 A ZA200805028 A ZA 200805028A ZA 200805028 A ZA200805028 A ZA 200805028A ZA 200805028 B ZA200805028 B ZA 200805028B
- Authority
- ZA
- South Africa
- Prior art keywords
- arylpropynamide
- arylmethylurea
- arylpropionamide
- arylacrylamide
- analogs
- Prior art date
Links
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US75013005P | 2005-12-14 | 2005-12-14 |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA200805028B true ZA200805028B (en) | 2009-12-30 |
Family
ID=40214768
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA200805028A ZA200805028B (en) | 2005-12-14 | 2008-06-09 | Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor Xla inhibitors |
Country Status (3)
Country | Link |
---|---|
CN (1) | CN101341129B (en) |
ES (1) | ES2365815T3 (en) |
ZA (1) | ZA200805028B (en) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20110097666A1 (en) * | 2009-10-27 | 2011-04-28 | Celin Savariar-Hauck | Lithographic printing plate precursors |
WO2011100402A1 (en) | 2010-02-11 | 2011-08-18 | Bristol-Myers Squibb Company | Macrocycles as factor xia inhibitors |
GB2494851A (en) * | 2011-07-07 | 2013-03-27 | Kalvista Pharmaceuticals Ltd | Plasma kallikrein inhibitors |
TWI613199B (en) * | 2011-12-21 | 2018-02-01 | 小野藥品工業股份有限公司 | Compounds |
US9475809B2 (en) * | 2013-07-23 | 2016-10-25 | Bayer Pharma Aktiengesellschaft | Substituted oxopyridine derivatives and use thereof as factor xia/plasma |
CN112028877B (en) * | 2019-06-04 | 2021-11-26 | 江西济民可信集团有限公司 | Alkoxy pyridone compound and preparation method and application thereof |
WO2022122035A1 (en) * | 2020-12-11 | 2022-06-16 | 上海领泰生物医药科技有限公司 | Coagulation factor xia inhibitor, preparation method therefor and use thereof |
CN115461330A (en) * | 2021-03-18 | 2022-12-09 | 深圳信立泰药业股份有限公司 | FXIa inhibitor compound impurity and preparation method and application thereof |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU746963B2 (en) * | 1998-06-12 | 2002-05-09 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) | Imidazolyl derivatives |
RU2242481C2 (en) * | 1998-06-16 | 2004-12-20 | Сосьете Де Консей Де Решерш Э Д'Аппликасьон Сьентифик Сас | Analogs of cyclic somatostatin |
ATE377017T1 (en) * | 2002-01-31 | 2007-11-15 | Morphochem Ag Komb Chemie | COMPOUNDS THAT INHIBIT FACTOR XA-ACTIVE T |
US7371743B2 (en) * | 2004-02-28 | 2008-05-13 | Boehringer Ingelheim International Gmbh | Carboxylic acid amides, the preparation thereof and their use as medicaments |
US7417063B2 (en) * | 2004-04-13 | 2008-08-26 | Bristol-Myers Squibb Company | Bicyclic heterocycles useful as serine protease inhibitors |
-
2006
- 2006-12-13 CN CN2006800472472A patent/CN101341129B/en not_active Expired - Fee Related
- 2006-12-13 ES ES06846594T patent/ES2365815T3/en active Active
-
2008
- 2008-06-09 ZA ZA200805028A patent/ZA200805028B/en unknown
Also Published As
Publication number | Publication date |
---|---|
CN101341129A (en) | 2009-01-07 |
ES2365815T3 (en) | 2011-10-11 |
CN101341129B (en) | 2011-12-14 |
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