ZA200503040B - Pharmaceutical compositions having a modified vehicle - Google Patents

Pharmaceutical compositions having a modified vehicle Download PDF

Info

Publication number: ZA200503040B
Authority: ZA; South Africa
Prior art keywords: oil; modified; composition; vehicle; composition according
Prior art date: 2002-11-19

Application number

ZA200503040A

Other languages

English (en)

Inventor

Ondrej Hendl

Susan Marie Machkovech

Niki Ann Waldron

Nancy Jean Britten

Dannette Marie Shaw

Alanta Lea Lary

Thomas Joseph Yellig

Original Assignee

Pharmacia & Upjohn Co Llc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-11-19

Filing date

2005-04-14

Publication date

2006-09-27

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32326579&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200503040(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2005-04-14 Application filed by Pharmacia & Upjohn Co Llc filed Critical Pharmacia & Upjohn Co Llc

2006-09-27 Publication of ZA200503040B publication Critical patent/ZA200503040B/en

Links

239000008194 pharmaceutical composition Substances 0.000 title claims description 11
239000000203 mixture Substances 0.000 claims description 92
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239000003921 oil Substances 0.000 claims description 41
235000019198 oils Nutrition 0.000 claims description 41
239000007788 liquid Substances 0.000 claims description 39
238000013268 sustained release Methods 0.000 claims description 36
239000012730 sustained-release form Substances 0.000 claims description 36
235000012343 cottonseed oil Nutrition 0.000 claims description 30
239000002385 cottonseed oil Substances 0.000 claims description 30
238000000034 method Methods 0.000 claims description 25
239000000126 substance Substances 0.000 claims description 23
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ZBHXIWJRIFEVQY-IHMPYVIRSA-N ceftiofur Chemical compound S([C@@H]1[C@@H](C(N1C=1C(O)=O)=O)NC(=O)\C(=N/OC)C=2N=C(N)SC=2)CC=1CSC(=O)C1=CC=CO1 ZBHXIWJRIFEVQY-IHMPYVIRSA-N 0.000 claims description 21
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DOZKMFVMCATMEH-ZCXUNETKSA-N 1-oleoyl-2-palmitoylglycerol Chemical compound CCCCCCCCCCCCCCCC(=O)OC(CO)COC(=O)CCCCCCC\C=C/CCCCCCCC DOZKMFVMCATMEH-ZCXUNETKSA-N 0.000 description 2
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RCINICONZNJXQF-MZXODVADSA-N taxol Chemical compound O([C@@H]1[C@@]2(C[C@@H](C(C)=C(C2(C)C)[C@H](C([C@]2(C)[C@@H](O)C[C@H]3OC[C@]3([C@H]21)OC(C)=O)=O)OC(=O)C)OC(=O)[C@H](O)[C@@H](NC(=O)C=1C=CC=CC=1)C=1C=CC=CC=1)O)C(=O)C1=CC=CC=C1 RCINICONZNJXQF-MZXODVADSA-N 0.000 description 1
YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 description 1
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LADGBHLMCUINGV-UHFFFAOYSA-N tricaprin Chemical compound CCCCCCCCCC(=O)OCC(OC(=O)CCCCCCCCC)COC(=O)CCCCCCCCC LADGBHLMCUINGV-UHFFFAOYSA-N 0.000 description 1
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/44—Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
- A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Epidemiology (AREA)
Oil, Petroleum & Natural Gas (AREA)
Dermatology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Cephalosporin Compounds (AREA)

ZA200503040A 2002-11-19 2005-04-14 Pharmaceutical compositions having a modified vehicle ZA200503040B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US42768002P	2002-11-19	2002-11-19

Publications (1)

Publication Number	Publication Date
ZA200503040B true ZA200503040B (en)	2006-09-27

Family

ID=32326579

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200503040A ZA200503040B (en)	2002-11-19	2005-04-14	Pharmaceutical compositions having a modified vehicle

Country Status (18)

Country	Link
US (1)	US7659061B2 (no)
EP (1)	EP1569693B1 (no)
JP (1)	JP4656945B2 (no)
KR (1)	KR20050085037A (no)
CN (2)	CN1713923A (no)
AR (1)	AR042193A1 (no)
AU (1)	AU2003276594B2 (no)
BR (1)	BR0316310A (no)
CA (1)	CA2502025C (no)
IL (1)	IL168183A (no)
MX (1)	MXPA05005319A (no)
NO (1)	NO20051688L (no)
NZ (1)	NZ539923A (no)
PL (1)	PL377740A1 (no)
RU (1)	RU2401127C2 (no)
TW (1)	TWI267379B (no)
WO (1)	WO2004045646A1 (no)
ZA (1)	ZA200503040B (no)

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US8975310B2 (en)	2011-07-20	2015-03-10	Brigham Young University	Hydrophobic ceragenin compounds and devices incorporating same
CA2852989C (en)	2011-09-13	2021-06-29	Brigham Young University	Compositions for treating bone diseases and broken bones
MX369385B (es)	2011-09-13	2019-11-07	Univ Brigham Young	Productos para cicatrizar heridas tisulares.
US9694019B2 (en)	2011-09-13	2017-07-04	Brigham Young University	Compositions and methods for treating bone diseases and broken bones
US9603859B2 (en)	2011-09-13	2017-03-28	Brigham Young University	Methods and products for increasing the rate of healing of tissue wounds
JP6051230B2 (ja)	2011-12-21	2016-12-27	ブリガムヤングユニバーシティ	口腔ケア組成物
US9533063B1 (en)	2012-03-01	2017-01-03	Brigham Young University	Aerosols incorporating ceragenin compounds and methods of use thereof
EP3225113B1 (en)	2012-05-02	2020-09-02	Brigham Young University	Methods for making ceragenin particulate materials
WO2014062960A1 (en)	2012-10-17	2014-04-24	Brigham Young University	Treatment and prevention of mastitis
CA2897150C (en)	2013-01-07	2021-07-13	Brigham Young University	Methods for reducing cellular proliferation and treating certain diseases
RU2669800C2 (ru)	2013-03-15	2018-10-16	Брихэм Янг Юниверсити	Способы лечения воспаления, аутоиммунных расстройств и боли
US10568893B2 (en)	2013-03-15	2020-02-25	Brigham Young University	Methods for treating inflammation, autoimmune disorders and pain
US11524015B2 (en)	2013-03-15	2022-12-13	Brigham Young University	Methods for treating inflammation, autoimmune disorders and pain
US9387215B2 (en)	2013-04-22	2016-07-12	Brigham Young University	Animal feed including cationic cholesterol additive and related methods
US11690855B2 (en)	2013-10-17	2023-07-04	Brigham Young University	Methods for treating lung infections and inflammation
US20150203527A1 (en)	2014-01-23	2015-07-23	Brigham Young University	Cationic steroidal antimicrobials
CA2844321C (en)	2014-02-27	2021-03-16	Brigham Young University	Cationic steroidal antimicrobial compounds
US9867836B2 (en)	2014-03-13	2018-01-16	Brigham Young University	Lavage and/or infusion using CSA compounds for increasing fertility in a mammal
US10220045B2 (en)	2014-03-13	2019-03-05	Brigham Young University	Compositions and methods for forming stabilized compositions with reduced CSA agglomeration
US9931350B2 (en)	2014-03-14	2018-04-03	Brigham Young University	Anti-infective and osteogenic compositions and methods of use
EP3131532A1 (de)	2014-04-16	2017-02-22	Veyx-Pharma GmbH	Veterinärpharmazeutische zusammensetzung und deren verwendung
US9686966B2 (en)	2014-04-30	2017-06-27	Brigham Young University	Methods and apparatus for cleaning or disinfecting a water delivery system
US10238665B2 (en)	2014-06-26	2019-03-26	Brigham Young University	Methods for treating fungal infections
US10441595B2 (en)	2014-06-26	2019-10-15	Brigham Young University	Methods for treating fungal infections
US10227376B2 (en)	2014-08-22	2019-03-12	Brigham Young University	Radiolabeled cationic steroid antimicrobials and diagnostic methods
US10155788B2 (en)	2014-10-07	2018-12-18	Brigham Young University	Cationic steroidal antimicrobial prodrug compositions and uses thereof
US9527883B2 (en)	2015-04-22	2016-12-27	Brigham Young University	Methods for the synthesis of ceragenins
WO2016172543A1 (en)	2015-04-22	2016-10-27	Savage Paul B	Methods for the synthesis of ceragenins
US9434759B1 (en)	2015-05-18	2016-09-06	Brigham Young University	Cationic steroidal antimicrobial compounds and methods of manufacturing such compounds
US10226550B2 (en)	2016-03-11	2019-03-12	Brigham Young University	Cationic steroidal antimicrobial compositions for the treatment of dermal tissue
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2003
- 2003-11-12 US US10/706,255 patent/US7659061B2/en active Active
- 2003-11-17 EP EP03811460.9A patent/EP1569693B1/en not_active Expired - Lifetime
- 2003-11-17 WO PCT/IB2003/005234 patent/WO2004045646A1/en active Application Filing
- 2003-11-17 CA CA2502025A patent/CA2502025C/en not_active Expired - Lifetime
- 2003-11-17 AR ARP030104227A patent/AR042193A1/es not_active Application Discontinuation
- 2003-11-17 JP JP2004553024A patent/JP4656945B2/ja not_active Expired - Lifetime
- 2003-11-17 PL PL377740A patent/PL377740A1/pl unknown
- 2003-11-17 AU AU2003276594A patent/AU2003276594B2/en not_active Ceased
- 2003-11-17 CN CNA2003801036161A patent/CN1713923A/zh active Pending
- 2003-11-17 CN CN2013101785052A patent/CN103272243A/zh active Pending
- 2003-11-17 NZ NZ539923A patent/NZ539923A/en not_active IP Right Cessation
- 2003-11-17 MX MXPA05005319A patent/MXPA05005319A/es active IP Right Grant
- 2003-11-17 RU RU2005115131/15A patent/RU2401127C2/ru active
- 2003-11-17 KR KR1020057008917A patent/KR20050085037A/ko not_active Application Discontinuation
- 2003-11-17 BR BR0316310-5A patent/BR0316310A/pt not_active Application Discontinuation
- 2003-11-18 TW TW092132304A patent/TWI267379B/zh not_active IP Right Cessation
2005
- 2005-04-05 NO NO20051688A patent/NO20051688L/no not_active Application Discontinuation
- 2005-04-14 ZA ZA200503040A patent/ZA200503040B/en unknown
- 2005-04-21 IL IL168183A patent/IL168183A/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
KR20050085037A (ko)	2005-08-29
CN103272243A (zh)	2013-09-04
NO20051688L (no)	2005-08-02
AR042193A1 (es)	2005-06-15
IL168183A (en)	2010-04-29
CA2502025A1 (en)	2004-06-03
BR0316310A (pt)	2005-09-27
JP2006514629A (ja)	2006-05-11
JP4656945B2 (ja)	2011-03-23
AU2003276594B2 (en)	2009-01-08
RU2005115131A (ru)	2005-10-27
PL377740A1 (pl)	2006-02-20
RU2401127C2 (ru)	2010-10-10
CN1713923A (zh)	2005-12-28
EP1569693B1 (en)	2016-12-28
CA2502025C (en)	2013-07-02
TW200427466A (en)	2004-12-16
MXPA05005319A (es)	2005-07-25
US20040170650A1 (en)	2004-09-02
NZ539923A (en)	2007-02-23
US7659061B2 (en)	2010-02-09
AU2003276594A1 (en)	2004-06-15
WO2004045646A1 (en)	2004-06-03
EP1569693A1 (en)	2005-09-07
NO20051688D0 (no)	2005-04-05
TWI267379B (en)	2006-12-01

Publication	Publication Date	Title
AU2003276594B2 (en)	2009-01-08	Pharmaceutical compositions having a modified vehicle
EP1575618B1 (en)	2006-08-16	Dispersible pharmaceutical compositions
CA2416566C (en)	2011-05-31	Depot formulation comprising ceftiofur and peroxidized natural oil
AU2001288323A1 (en)	2002-06-13	Pharmaceutical composition having modified carrier
US20020068065A1 (en)	2002-06-06	Pharmaceutical composition having specific water activity
DK1569693T3 (en)	2017-02-27	Pharmaceutical compositions with a modified vehicle
US7829100B2 (en)	2010-11-09	Pharmaceutical composition having modified carrier