WO2009156090A3 - Insecticidal sulfur-derivatized 1-azinylpyrazoles - Google Patents

Insecticidal sulfur-derivatized 1-azinylpyrazoles Download PDF

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Publication number
WO2009156090A3
WO2009156090A3 PCT/EP2009/004391 EP2009004391W WO2009156090A3 WO 2009156090 A3 WO2009156090 A3 WO 2009156090A3 EP 2009004391 W EP2009004391 W EP 2009004391W WO 2009156090 A3 WO2009156090 A3 WO 2009156090A3
Authority
WO
WIPO (PCT)
Prior art keywords
azinylpyrazoles
derivatized
sulfur
insecticidal
present
Prior art date
Application number
PCT/EP2009/004391
Other languages
German (de)
French (fr)
Other versions
WO2009156090A2 (en
Inventor
Hans-Georg Schwarz
Thomas Schenke
Achim Hense
Robert Velten
Simon MAECHLING
Stefan Werner
Eva-Maria Franken
Ulrich Görgens
Peter Lümmen
Ulrich Ebbinghaus-Kintscher
Arnd Voerste
Original Assignee
Bayer Cropscience Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Aktiengesellschaft filed Critical Bayer Cropscience Aktiengesellschaft
Publication of WO2009156090A2 publication Critical patent/WO2009156090A2/en
Publication of WO2009156090A3 publication Critical patent/WO2009156090A3/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/561,2-Diazoles; Hydrogenated 1,2-diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/44Oxygen and nitrogen or sulfur and nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

The present invention relates to sulfur-derivatized 1-azinylpyrazoles, the use thereof as insecticides and / or parasiticides and processes for the preparation thereof.  Further objects of the present invention are various intermediates of the production of the sulfur-derivatized 1-azinylpyrazoles of the invention.  Further objects of the present invention finally are materials, which contain such azinylpyrazoles.
PCT/EP2009/004391 2008-06-26 2009-06-18 Insecticidal sulfur-derivatized 1-azinylpyrazoles WO2009156090A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08159069 2008-06-26
EP08159069.7 2008-06-26

Publications (2)

Publication Number Publication Date
WO2009156090A2 WO2009156090A2 (en) 2009-12-30
WO2009156090A3 true WO2009156090A3 (en) 2010-04-08

Family

ID=40039731

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2009/004391 WO2009156090A2 (en) 2008-06-26 2009-06-18 Insecticidal sulfur-derivatized 1-azinylpyrazoles

Country Status (3)

Country Link
AR (1) AR072673A1 (en)
TW (1) TW201012812A (en)
WO (1) WO2009156090A2 (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2266973A1 (en) * 2009-05-29 2010-12-29 Bayer CropScience AG Pyrazinylpyrazole
CN102499218B (en) * 2011-10-21 2014-04-09 福建农林大学 Pretreatment device and method for toxicological experiments of pesticides
BR112014012243A2 (en) 2011-11-21 2017-05-30 Basf Se compound preparation process
EP2844651A1 (en) 2012-05-04 2015-03-11 Basf Se Substituted pyrazole-containing compounds and their use as pesticides
WO2021151976A1 (en) * 2020-01-31 2021-08-05 Bayer Aktiengesellschaft [(1,4,5-trisubstituted-1h-pyrazol-3-yl)sulfanyl]acetic acid derivatives, salts thereof, and use thereof as herbicidal ingredients
WO2024121263A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121262A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121261A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives
WO2024121264A1 (en) 2022-12-09 2024-06-13 Syngenta Crop Protection Ag Insecticidal compound based on pyrazole derivatives

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0234622A1 (en) * 1986-02-19 1987-09-02 Duphar International Research B.V New thio compounds having fungicidal activity
WO1995022530A1 (en) * 1994-02-18 1995-08-24 Bayer Aktiengesellschaft N-pyrazolyl anilines and n-pyrazolyl aminopyridines as pesticides
JPH08208620A (en) * 1995-02-03 1996-08-13 Takeda Chem Ind Ltd Aminopyrazole derivative, its production and use
WO2001007413A1 (en) * 1999-07-22 2001-02-01 3-Dimensional Pharmaceuticals, Inc. 1-aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0234622A1 (en) * 1986-02-19 1987-09-02 Duphar International Research B.V New thio compounds having fungicidal activity
WO1995022530A1 (en) * 1994-02-18 1995-08-24 Bayer Aktiengesellschaft N-pyrazolyl anilines and n-pyrazolyl aminopyridines as pesticides
JPH08208620A (en) * 1995-02-03 1996-08-13 Takeda Chem Ind Ltd Aminopyrazole derivative, its production and use
WO2001007413A1 (en) * 1999-07-22 2001-02-01 3-Dimensional Pharmaceuticals, Inc. 1-aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
DATABASE WPI Week 199642, Derwent World Patents Index; AN 1996-421965, XP002506499 *
THOMAS A ET AL: "CYCLOCONDENSATION OF OXOKETENE DITHIOACETALS WITH 3-AMINOPYRAZOLES:A FACILE HIGHLY REGIOSELECTIVE GENERAL ROUTE TO SUBSTITUTED AND FUSED PYRAZOLO not A 3/4 PYRIMIDINES", TETRAHEDRON, ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM, NL, vol. 46, no. 2, 1 January 1990 (1990-01-01), pages 577 - 586, XP002921816, ISSN: 0040-4020 *

Also Published As

Publication number Publication date
WO2009156090A2 (en) 2009-12-30
AR072673A1 (en) 2010-09-15
TW201012812A (en) 2010-04-01

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