WO2009069736A1 - 含窒素化合物 - Google Patents

含窒素化合物 Download PDF

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Publication number
WO2009069736A1
WO2009069736A1 PCT/JP2008/071627 JP2008071627W WO2009069736A1 WO 2009069736 A1 WO2009069736 A1 WO 2009069736A1 JP 2008071627 W JP2008071627 W JP 2008071627W WO 2009069736 A1 WO2009069736 A1 WO 2009069736A1
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hydrogen atom
formula
nitrogenated compound
nitrogenated
substituent
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PCT/JP2008/071627
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English (en)
French (fr)
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Koji Yanagawa
Kiyotoshi Mori
Yoshisuke Nakasato
Jun Funahashi
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Kyowa Hakko Kirin Co., Ltd.
Funahashi, Mami
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Application filed by Kyowa Hakko Kirin Co., Ltd., Funahashi, Mami filed Critical Kyowa Hakko Kirin Co., Ltd.
Publication of WO2009069736A1 publication Critical patent/WO2009069736A1/ja

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Abstract

　式（Ｉ）［Aは、置換基を有していてもよいアリール等を表し、Bはそれぞれ、同一または異なって、水素原子、ハロゲン等を表し、ｎは１から置換可能な最大の整数を表し、R9は、水素原子等を表し、R10は式(III)（式中、R11は、芳香族複素環基等を表し、R12は水素原子等を表す）等を表す］で表される含窒素化合物またはその薬学的に許容される塩等を提供する。
PCT/JP2008/071627 2007-11-28 2008-11-28 含窒素化合物 WO2009069736A1 (ja)

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WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
WO2011161030A1 (de) 2010-06-21 2011-12-29 Sanofi Heterocyclisch substituierte methoxyphenylderivate mit oxogruppe, verfahren zu ihrer herstellung und ihre verwendung als gpr40 rezeptor modulatoren
WO2012004269A1 (de) 2010-07-05 2012-01-12 Sanofi ( 2 -aryloxy -acetylamino) - phenyl - propionsäurederivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
WO2012004270A1 (de) 2010-07-05 2012-01-12 Sanofi Spirocyclisch substituierte 1,3-propandioxidderivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
WO2012010413A1 (de) 2010-07-05 2012-01-26 Sanofi Aryloxy-alkylen-substituierte hydroxy-phenyl-hexinsäuren, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013045413A1 (en) 2011-09-27 2013-04-04 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
US9814698B2 (en) 2015-04-21 2017-11-14 University Of Tennessee Research Foundation Selective androgen receptor degrader (SARD) ligands and methods of use thereof
US9815776B2 (en) 2015-04-21 2017-11-14 University Of Tennessee Research Foundation Selective androgen receptor degrader (SARD) ligands and methods of use thereof
US9834507B2 (en) 2015-04-21 2017-12-05 University Of Tennessee Research Foundation Selective androgen receptor degrader (SARD) ligands and methods of use thereof
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WO2012004269A1 (de) 2010-07-05 2012-01-12 Sanofi ( 2 -aryloxy -acetylamino) - phenyl - propionsäurederivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
WO2012004270A1 (de) 2010-07-05 2012-01-12 Sanofi Spirocyclisch substituierte 1,3-propandioxidderivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
WO2012010413A1 (de) 2010-07-05 2012-01-26 Sanofi Aryloxy-alkylen-substituierte hydroxy-phenyl-hexinsäuren, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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