WO2005023198A3 - Modafinil compositions - Google Patents
Modafinil compositions Download PDFInfo
- Publication number
- WO2005023198A3 WO2005023198A3 PCT/US2004/029013 US2004029013W WO2005023198A3 WO 2005023198 A3 WO2005023198 A3 WO 2005023198A3 US 2004029013 W US2004029013 W US 2004029013W WO 2005023198 A3 WO2005023198 A3 WO 2005023198A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- modafinil
- modulated
- modafinil compositions
- enantiomerically
- compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/18—Sulfonamides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
- C07C53/126—Acids containing more than four carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C55/00—Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
- C07C55/02—Dicarboxylic acids
- C07C55/06—Oxalic acid
- C07C55/07—Salts thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C55/00—Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
- C07C55/02—Dicarboxylic acids
- C07C55/08—Malonic acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C55/00—Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
- C07C55/02—Dicarboxylic acids
- C07C55/12—Glutaric acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/235—Saturated compounds containing more than one carboxyl group
- C07C59/245—Saturated compounds containing more than one carboxyl group containing hydroxy or O-metal groups
- C07C59/255—Tartaric acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/235—Saturated compounds containing more than one carboxyl group
- C07C59/245—Saturated compounds containing more than one carboxyl group containing hydroxy or O-metal groups
- C07C59/265—Citric acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C65/00—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C65/01—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups
- C07C65/03—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups monocyclic and having all hydroxy or O-metal groups bound to the ring
- C07C65/05—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups monocyclic and having all hydroxy or O-metal groups bound to the ring o-Hydroxy carboxylic acids
- C07C65/10—Salicylic acid
Abstract
Priority Applications (27)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN2004800319825A CN1874993B (en) | 2003-09-04 | 2004-09-04 | Modafinil compositionsc |
KR1020067004425A KR101184797B1 (en) | 2003-09-04 | 2004-09-04 | Modafinil compositions |
US10/570,405 US7566805B2 (en) | 2003-09-04 | 2004-09-04 | Modafinil compositions |
MXPA06002507A MXPA06002507A (en) | 2003-09-04 | 2004-09-04 | Modafinil compositions. |
CA2534664A CA2534664C (en) | 2003-09-04 | 2004-09-04 | Modafinil compositions |
AU2004270238A AU2004270238B2 (en) | 2003-09-04 | 2004-09-04 | Modafinil compositions |
BRPI0413777-9A BRPI0413777A (en) | 2003-09-04 | 2004-09-04 | modafinil compositions |
EP20040783308 EP1670753A4 (en) | 2003-09-04 | 2004-09-04 | Modafinil compositions |
JP2006525508A JP4842819B2 (en) | 2003-09-04 | 2004-09-04 | Modafinil composition |
NZ545133A NZ545133A (en) | 2003-09-04 | 2004-09-04 | Modafinil compositions |
AU2005212229A AU2005212229B2 (en) | 2004-02-06 | 2005-02-01 | Modafinil compositions |
PCT/US2005/002782 WO2005077894A1 (en) | 2004-02-06 | 2005-02-01 | Modafinil compositions |
JP2006552169A JP4917441B2 (en) | 2004-02-06 | 2005-02-01 | Modafinil composition |
EA200601390A EA009949B1 (en) | 2004-02-06 | 2005-02-01 | Modafinil compositions |
CN2005800041104A CN1980888B (en) | 2004-02-06 | 2005-02-01 | Modafinil compositions |
US10/587,086 US20090018202A1 (en) | 2004-02-06 | 2005-02-01 | Modafinil compositions |
EP05712282A EP1718607A4 (en) | 2004-02-06 | 2005-02-01 | Modafinil compositions |
BRPI0507455-0A BRPI0507455A (en) | 2000-07-15 | 2005-02-01 | composition, methods of making a r - (-) - modafinil polymorph, making 2: 1 of r - (-) - modafinil: s - (+) - modafinil, making forms iii, iv and v of r - (-) modafinil and treatment of an individual suffering from diseases, and r - (-) - modafinil solvate, and methods of treating an individual suffering from excessive daytime sleep associated with narcolepsy, narcolepsy or sleep apnea and attention deficit hyperactivity disorder (adhd) |
CA002556106A CA2556106A1 (en) | 2004-02-06 | 2005-02-01 | Modafinil compositions |
EP10001997A EP2292213A1 (en) | 2004-02-06 | 2005-02-01 | Compositions comprising a polymorphic form of armodafinil |
IL173575A IL173575A0 (en) | 2003-09-04 | 2006-02-07 | Modafinil compositions |
NO20060669A NO20060669L (en) | 2003-09-11 | 2006-02-10 | Modafinilsammensetninger |
IL176934A IL176934A (en) | 2004-02-06 | 2006-07-18 | Use of form v of r-(-)-modafinil in the preparation of a medicament for treating excessive daytime sleepiness and attention deficit hyperactivity disorder (adhd) |
NO20063957A NO20063957L (en) | 2004-02-06 | 2006-09-05 | Modafinilsammensetninger |
IL199140A IL199140A (en) | 2003-09-04 | 2009-06-03 | Modafinil compositions |
US12/708,998 US8338646B2 (en) | 2004-02-06 | 2010-02-19 | Modafinil compositions |
US13/706,835 US8809586B2 (en) | 2004-02-06 | 2012-12-06 | Modafinil compositions |
Applications Claiming Priority (22)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US32777203A | 2003-09-04 | 2003-09-04 | |
USUS03/27772 | 2003-09-04 | ||
US10/660,202 US7927613B2 (en) | 2002-02-15 | 2003-09-11 | Pharmaceutical co-crystal compositions |
US10/660,202 | 2003-09-11 | ||
US50820803P | 2003-10-02 | 2003-10-02 | |
US60/508,208 | 2003-10-02 | ||
US54275204P | 2004-02-06 | 2004-02-06 | |
US60/542,752 | 2004-02-06 | ||
US40628804A | 2004-02-26 | 2004-02-26 | |
USUS04/06288 | 2004-02-26 | ||
US56041104P | 2004-04-06 | 2004-04-06 | |
US60/560,411 | 2004-04-06 | ||
US57341204P | 2004-05-21 | 2004-05-21 | |
US60/573,412 | 2004-05-21 | ||
US57917604P | 2004-06-12 | 2004-06-12 | |
US60/579,176 | 2004-06-12 | ||
US58199204P | 2004-06-22 | 2004-06-22 | |
US60/581,992 | 2004-06-22 | ||
US58675204P | 2004-07-09 | 2004-07-09 | |
US60/586,752 | 2004-07-09 | ||
US58823604P | 2004-07-15 | 2004-07-15 | |
US60/588,236 | 2004-07-15 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2005023198A2 WO2005023198A2 (en) | 2005-03-17 |
WO2005023198A3 true WO2005023198A3 (en) | 2005-07-14 |
Family
ID=34280325
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2004/029013 WO2005023198A2 (en) | 2000-07-15 | 2004-09-04 | Modafinil compositions |
Country Status (6)
Country | Link |
---|---|
KR (1) | KR101184797B1 (en) |
AU (1) | AU2004270238B2 (en) |
CA (1) | CA2534664C (en) |
MX (1) | MXPA06002507A (en) |
NZ (1) | NZ545133A (en) |
WO (1) | WO2005023198A2 (en) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7927613B2 (en) | 2002-02-15 | 2011-04-19 | University Of South Florida | Pharmaceutical co-crystal compositions |
US7790905B2 (en) | 2002-02-15 | 2010-09-07 | Mcneil-Ppc, Inc. | Pharmaceutical propylene glycol solvate compositions |
US20050025791A1 (en) | 2002-06-21 | 2005-02-03 | Julius Remenar | Pharmaceutical compositions with improved dissolution |
AU2003213719A1 (en) | 2002-03-01 | 2003-09-16 | Regents Of The University Of Michigan | Multiple-component solid phases containing at least one active pharmaceutical ingredient |
FR2849029B1 (en) | 2002-12-20 | 2005-03-18 | Lafon Labor | PROCESS FOR THE PREPARATION AND CRYSTALLINE FORMS OF OPTICAL ENANTIOMERS OF MODAFINIL. |
US8183290B2 (en) | 2002-12-30 | 2012-05-22 | Mcneil-Ppc, Inc. | Pharmaceutically acceptable propylene glycol solvate of naproxen |
WO2005099822A2 (en) * | 2004-04-13 | 2005-10-27 | Cephalon, Inc. | Reduction of drug / drug interactions with modafinil |
ATE483455T1 (en) * | 2004-05-28 | 2010-10-15 | Transform Pharmaceuticals Inc | MIXED CRYSTALS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
WO2007013962A2 (en) * | 2005-07-21 | 2007-02-01 | Neurohealing Pharmaceuticals, Inc. | Rapid onset and short term modafinil compositions and methods of use thereof |
ITMI20051971A1 (en) * | 2005-10-18 | 2007-04-19 | Dipharma Spa | PROCEDURE FOR THE PREPARATION OF - MODAFINIL |
US20070293702A1 (en) * | 2006-02-21 | 2007-12-20 | Viviana Braude | Novel crystalline forms of armodafinil and preparation thereof |
TWI370818B (en) * | 2006-04-05 | 2012-08-21 | Astellas Pharma Inc | Cocrystal of c-glycoside derivative and l-proline |
US20100130616A1 (en) * | 2006-11-09 | 2010-05-27 | Novartis Ag | Salt of aliskiren with orotic acid |
WO2008075736A1 (en) | 2006-12-21 | 2008-06-26 | Astellas Pharma Inc. | Method for producing c-glycoside derivative and synthetic intermediate thereof |
WO2009025791A2 (en) | 2007-08-16 | 2009-02-26 | Teva Pharmaceutical Industries Ltd. | Purification of armodafinil |
US20090105346A1 (en) * | 2007-10-02 | 2009-04-23 | Alexandr Jegorov | Novel crystalline forms of armodafinil and preparation thereof |
US8871793B2 (en) * | 2009-12-23 | 2014-10-28 | Nuformix Limited | Metaxalone cocrystals |
KR102372908B1 (en) * | 2021-09-27 | 2022-03-10 | 유니셀랩 주식회사 | Novel co-crystal of pelubiprofen/mandelic acid |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2002056915A2 (en) * | 2000-12-19 | 2002-07-25 | Cephalon, Inc. | Complex of modafinil and cyclodextrin |
WO2003074474A2 (en) * | 2002-03-01 | 2003-09-12 | University Of South Florida | Multiple-component solid phases containing at least one active pharmaceutical ingredient |
US20040019211A1 (en) * | 2002-05-31 | 2004-01-29 | Transform Pharmaceuticals, Inc. | Novel conazole crystalline forms and related processes, pharmaceutical compositions and methods |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2593809B1 (en) * | 1986-01-31 | 1988-07-22 | Lafon Labor | BENZHYDRYLSULFINYLACETAMIDE, PROCESS FOR PREPARATION AND THERAPEUTIC USE |
EP1608339B8 (en) * | 2003-02-28 | 2012-04-25 | McNeill-PPC, Inc. | Pharmaceutical co-crystal of celecoxib-nicotinamide |
-
2004
- 2004-09-04 NZ NZ545133A patent/NZ545133A/en not_active IP Right Cessation
- 2004-09-04 MX MXPA06002507A patent/MXPA06002507A/en active IP Right Grant
- 2004-09-04 KR KR1020067004425A patent/KR101184797B1/en not_active IP Right Cessation
- 2004-09-04 WO PCT/US2004/029013 patent/WO2005023198A2/en active Application Filing
- 2004-09-04 AU AU2004270238A patent/AU2004270238B2/en not_active Ceased
- 2004-09-04 CA CA2534664A patent/CA2534664C/en not_active Expired - Fee Related
Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2002056915A2 (en) * | 2000-12-19 | 2002-07-25 | Cephalon, Inc. | Complex of modafinil and cyclodextrin |
WO2003074474A2 (en) * | 2002-03-01 | 2003-09-12 | University Of South Florida | Multiple-component solid phases containing at least one active pharmaceutical ingredient |
US20030224006A1 (en) * | 2002-03-01 | 2003-12-04 | Zaworotko Michael J. | Multiple-component solid phases containing at least one active pharmaceutical ingredient |
US20040019211A1 (en) * | 2002-05-31 | 2004-01-29 | Transform Pharmaceuticals, Inc. | Novel conazole crystalline forms and related processes, pharmaceutical compositions and methods |
Non-Patent Citations (1)
Title |
---|
See also references of EP1670753A4 * |
Also Published As
Publication number | Publication date |
---|---|
CA2534664C (en) | 2012-10-30 |
AU2004270238A1 (en) | 2005-03-17 |
WO2005023198A2 (en) | 2005-03-17 |
CA2534664A1 (en) | 2005-03-17 |
KR101184797B1 (en) | 2012-09-20 |
MXPA06002507A (en) | 2006-06-20 |
NZ545133A (en) | 2009-12-24 |
AU2004270238B2 (en) | 2010-07-29 |
KR20060128831A (en) | 2006-12-14 |
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