UY37362A - Sulfonilureas y compuestos relacionados y sus usos - Google Patents
Sulfonilureas y compuestos relacionados y sus usosInfo
- Publication number
- UY37362A UY37362A UY0001037362A UY37362A UY37362A UY 37362 A UY37362 A UY 37362A UY 0001037362 A UY0001037362 A UY 0001037362A UY 37362 A UY37362 A UY 37362A UY 37362 A UY37362 A UY 37362A
- Authority
- UY
- Uruguay
- Prior art keywords
- sulfonile
- related compounds
- compounds
- acylamide
- heterocyclyl
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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Abstract
Compuestos de fórmula (I), sales, solvatos, profármacos farmacéuticamente aceptables:donde Q se selecciona de O, S, Se; J es S o Se; W1 y W2, se seleccionan de f N y C; R1 y R2 se seleccionan de hidrógeno, alquilo C1-C12, alquenilo C2-C12, alquinilo C2-C12, arilo, heterociclilo, heteroarilo, cicloalquilo, cicloalquenilo, amino, amido, alquiltio, acilo, arilalquilo, acilamido, donde al menos uno de W1 y W2 es un átomo de nitrógeno y cuando R1 o R2 son restos cíclicos, W1 o W2 puede formar parte de la estructura anular; composiciones farmacéuticas, métodos de tratamiento y usos asociados.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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AU2016900535A AU2016900535A0 (en) | 2016-02-16 | Sulfonylureas and related compounds and use of same | |
PCT/EP2017/053498 WO2017140778A1 (en) | 2016-02-16 | 2017-02-16 | Sulfonylureas and related compounds and use of same |
Publications (1)
Publication Number | Publication Date |
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UY37362A true UY37362A (es) | 2018-09-28 |
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UY0001037362A UY37362A (es) | 2016-02-16 | 2017-08-15 | Sulfonilureas y compuestos relacionados y sus usos |
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US (1) | US11858922B2 (es) |
EP (1) | EP3416948B1 (es) |
JP (1) | JP2019512009A (es) |
KR (1) | KR20180133244A (es) |
CN (1) | CN109071454B (es) |
AR (1) | AR109348A1 (es) |
AU (1) | AU2017219204A1 (es) |
BR (1) | BR112018016671A2 (es) |
CA (1) | CA3014487A1 (es) |
HK (1) | HK1257569A1 (es) |
IL (1) | IL261035A (es) |
MA (1) | MA44225A (es) |
MX (1) | MX2018009840A (es) |
SG (1) | SG11201806745RA (es) |
UY (1) | UY37362A (es) |
WO (1) | WO2017140778A1 (es) |
Families Citing this family (52)
Publication number | Priority date | Publication date | Assignee | Title |
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MX2017010528A (es) | 2015-02-16 | 2018-11-12 | Univ Queensland | Sulfonilureas y compuestos relacionados y uso de estos. |
AU2017219204A1 (en) | 2016-02-16 | 2018-08-23 | The Provost, Fellows, Foundation Scholars, And The Other Members Of Board, Of The College Of The Holy And Undivided Trinity Of Queen Elizabeth Near Dublin | Sulfonylureas and related compounds and use of same |
JP7219213B2 (ja) | 2016-09-06 | 2023-02-07 | ジャズ ファーマスティカルズ アイルランド リミテッド | (r)-2-アミノ-3-フェニルプロピルカルバメートの溶媒和物フォーム |
UA126675C2 (uk) | 2017-01-23 | 2023-01-11 | Дженентек, Інк. | Хімічні сполуки як інгібітори активності інтерлейкіну-1 |
BR112019024831A2 (pt) | 2017-05-24 | 2020-06-09 | The University Of Queensland | composto, sal, solvato ou pró-droga, composição farmacêutica, método de tratamento ou prevenção de uma doença, método para inibir o nlrp3 |
US11370776B2 (en) | 2017-07-07 | 2022-06-28 | Inflazome Limited | Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors |
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GB201721185D0 (en) | 2017-12-18 | 2018-01-31 | Nodthera Ltd | Sulphonyl urea derivatives |
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CN108404117B (zh) * | 2018-05-29 | 2020-06-30 | 广东龙帆生物科技有限公司 | 核苷酸结合寡聚化结构域样受体蛋白在治疗寨卡病毒感染药物中的应用 |
EP3823726A1 (en) | 2018-07-20 | 2021-05-26 | F. Hoffmann-La Roche SA | Sulfonylurea compounds as inhibitors of interleukin-1 activity |
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- 2017-02-16 CN CN201780022601.4A patent/CN109071454B/zh active Active
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WO2017140778A1 (en) | 2017-08-24 |
IL261035A (en) | 2018-10-31 |
US20200299284A1 (en) | 2020-09-24 |
AR109348A1 (es) | 2018-11-21 |
AU2017219204A1 (en) | 2018-08-23 |
BR112018016671A2 (pt) | 2018-12-26 |
EP3416948B1 (en) | 2024-07-24 |
CA3014487A1 (en) | 2017-08-24 |
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