UY34223A - Formulaciones de (trimetoxifenilamino)pirimidinilo nuevas - Google Patents

Formulaciones de (trimetoxifenilamino)pirimidinilo nuevas

Info

Publication number
UY34223A
UY34223A UY0001034223A UY34223A UY34223A UY 34223 A UY34223 A UY 34223A UY 0001034223 A UY0001034223 A UY 0001034223A UY 34223 A UY34223 A UY 34223A UY 34223 A UY34223 A UY 34223A
Authority
UY
Uruguay
Prior art keywords
trimetoxifenilamino
pyrimidinyl
formulations
new
página
Prior art date
Application number
UY0001034223A
Other languages
English (en)
Inventor
Farhan Abdul Karim Alhusban
Ian Paul Gabbott
Sievwright Dawn
David Bradley Brook Simpson
Gururajan Bindhumadhavan
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46875902&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY34223(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY34223A publication Critical patent/UY34223A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007—Effervescent
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5383—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid

Abstract

Se proporcionan composiciones farmacéuticas que comprenden más de un 15% p/p del compuesto de Fórmula (I), según se define en la presente, y/o un hidrato de este y una cantidad de uno o más agentes efervescentes que sea suficiente para proporcionar una disolución satisfactoria in vitro; y que comprenden además uno o más ingredientes farmacéuticamente aceptables; y procesos para obtenerlas.
UY0001034223A 2011-07-28 2012-07-26 Formulaciones de (trimetoxifenilamino)pirimidinilo nuevas UY34223A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201161512621P 2011-07-28 2011-07-28

Publications (1)

Publication Number Publication Date
UY34223A true UY34223A (es) 2013-02-28

Family

ID=46875902

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001034223A UY34223A (es) 2011-07-28 2012-07-26 Formulaciones de (trimetoxifenilamino)pirimidinilo nuevas

Country Status (26)

Country Link
US (2) US8771648B2 (es)
EP (1) EP2736487B1 (es)
JP (1) JP6019116B2 (es)
KR (2) KR102024120B1 (es)
CN (1) CN103826610B (es)
AR (1) AR087371A1 (es)
AU (1) AU2012288632B2 (es)
BR (1) BR112014001999B1 (es)
CA (1) CA2843138C (es)
CY (1) CY1122596T1 (es)
DK (1) DK2736487T3 (es)
EA (1) EA028432B1 (es)
ES (1) ES2710423T3 (es)
HK (1) HK1198741A1 (es)
HR (1) HRP20190186T1 (es)
HU (1) HUE042611T2 (es)
LT (1) LT2736487T (es)
MX (1) MX339685B (es)
PL (1) PL2736487T3 (es)
PT (1) PT2736487T (es)
RS (1) RS58433B1 (es)
SI (1) SI2736487T1 (es)
TR (1) TR201901792T4 (es)
TW (1) TW201311251A (es)
UY (1) UY34223A (es)
WO (1) WO2013014454A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK2078026T3 (da) * 2006-11-21 2012-04-30 Rigel Pharmaceuticals Inc Prodrug-salte af 2, 4-pyrimidinediamine-forbindelser og anvendelser deraf
ES2710423T3 (es) 2011-07-28 2019-04-25 Rigel Pharmaceuticals Inc Formulaciones de (trimetoxifenilamino) pirimidinilo nuevas
BR112017021126B1 (pt) 2015-04-02 2021-12-21 Stora Enso Oyj Composição de lignina ativada, método para a sua produção e utilização
WO2016172053A1 (en) 2015-04-24 2016-10-27 Rigel Pharmaceuticals, Inc. Methods of treating ibrutinib-resistant disease
WO2022017864A1 (en) * 2020-07-24 2022-01-27 Dsm Ip Assets B.V. New fast dissolvable tablets

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
ES2445208T3 (es) 2002-07-29 2014-02-28 Rigel Pharmaceuticals, Inc. Compuestos de 2,4-pirimidindiamina para uso en métodos para tratar o prevenir enfermedades autoinmunitarias
KR101201603B1 (ko) 2003-07-30 2012-11-14 리겔 파마슈티칼스, 인크. 자가면역 질환의 치료 또는 예방에 사용하기 위한2,4-피리미딘디아민 화합물
EP1663242B1 (en) 2003-08-07 2011-04-27 Rigel Pharmaceuticals, Inc. 2,4-pyrimidinediamine compounds and uses as anti-proliferative agents
WO2006012502A2 (en) * 2004-07-23 2006-02-02 Rigel Pharmaceuticals, Inc. Formulation of insoluble small molecule therapeutics in lipid-based carriers
CA2580838A1 (en) * 2004-09-27 2006-04-06 Amgen Inc. Substituted heterocyclic compounds and methods of use
ATE451381T1 (de) * 2005-01-19 2009-12-15 Rigel Pharmaceuticals Inc Prodrugs aus 2,4-pyrimidindiamin-verbindungen und ihre verwendungen
US8227455B2 (en) 2005-04-18 2012-07-24 Rigel Pharmaceuticals, Inc. Methods of treating cell proliferative disorders
WO2007111720A2 (en) * 2005-12-06 2007-10-04 Rigel Pharmaceuticals, Inc. Formulation of insoluble small molecule therapeutics in lipid-based carriers
PL1984357T3 (pl) * 2006-02-17 2014-03-31 Rigel Pharmaceuticals Inc Związki 2,4-pirymidynodiaminy do leczenia lub zapobiegania chorób autoimmunologicznych
WO2008061201A1 (en) * 2006-11-15 2008-05-22 Rigel Pharmaceuticals, Inc. Methods for treating renal tumors using 2,4-pyrimidinediamine drug and prodrug compounds
DK2078026T3 (da) * 2006-11-21 2012-04-30 Rigel Pharmaceuticals Inc Prodrug-salte af 2, 4-pyrimidinediamine-forbindelser og anvendelser deraf
WO2009003136A1 (en) * 2007-06-26 2008-12-31 Rigel Pharmaceuticals, Inc. Substituted pyrimidine-2, 4 -diamines for treating cell proliferative disorders
WO2009029682A1 (en) * 2007-08-28 2009-03-05 Rigel Pharmaceuticals, Inc. Combination therapy with syk kinase inhibitor
MY169761A (en) * 2007-11-07 2019-05-15 Rigel Pharmaceuticals Inc Wet granulation using a water sequestering agent
CN102014917A (zh) 2008-02-22 2011-04-13 里格尔药品股份有限公司 2，4-嘧啶二胺用于治疗动脉粥样硬化的用途
UA108077C2 (xx) 2009-07-02 2015-03-25 Синтез динатрієвої солі n4-(2,2-диметил-4-$(дигідрофосфонокси)метил]-3-оксо-5-піридо$1,4]оксазин-6-іл)-5-фтор-n2-(3,4,5-триметоксифеніл)-2,4-піримідиндіаміну
CA2768368A1 (en) 2009-07-17 2011-01-20 Rigel Pharmaceuticals, Inc. Deuterated 2, 4-pyrimidinediamine compounds and prodrugs thereof and their uses
ES2524127T3 (es) 2009-11-20 2014-12-04 Rigel Pharmaceuticals, Inc. Compuestos de 2,4-pirimidinodiamina y sus profármacos y sus usos
US8618095B2 (en) 2010-04-13 2013-12-31 Rigel Pharmaceuticals, Inc. 2, 4-pyrimidinediamine compounds and prodrugs thereof and their uses
ES2710423T3 (es) 2011-07-28 2019-04-25 Rigel Pharmaceuticals Inc Formulaciones de (trimetoxifenilamino) pirimidinilo nuevas

Also Published As

Publication number Publication date
JP2014521630A (ja) 2014-08-28
MX339685B (es) 2016-06-06
CA2843138C (en) 2020-06-02
US8951504B2 (en) 2015-02-10
AU2012288632A1 (en) 2014-02-20
WO2013014454A1 (en) 2013-01-31
MX2014001065A (es) 2014-08-01
HUE042611T2 (hu) 2019-07-29
PL2736487T3 (pl) 2019-06-28
EP2736487B1 (en) 2018-11-07
TR201901792T4 (tr) 2019-03-21
CN103826610A (zh) 2014-05-28
EA028432B1 (ru) 2017-11-30
PT2736487T (pt) 2019-02-13
KR20190109576A (ko) 2019-09-25
US20140271493A1 (en) 2014-09-18
KR102090440B1 (ko) 2020-03-17
DK2736487T3 (en) 2019-03-04
US20130058876A1 (en) 2013-03-07
BR112014001999B1 (pt) 2023-11-28
CY1122596T1 (el) 2021-01-27
SI2736487T1 (sl) 2019-04-30
ES2710423T3 (es) 2019-04-25
KR102024120B1 (ko) 2019-09-23
RS58433B1 (sr) 2019-04-30
AR087371A1 (es) 2014-03-19
LT2736487T (lt) 2019-02-25
KR20140058576A (ko) 2014-05-14
HK1198741A1 (en) 2015-06-05
BR112014001999A2 (pt) 2017-02-21
JP6019116B2 (ja) 2016-11-02
AU2012288632B2 (en) 2017-08-17
HRP20190186T1 (hr) 2019-03-22
EP2736487A1 (en) 2014-06-04
US8771648B2 (en) 2014-07-08
TW201311251A (zh) 2013-03-16
CN103826610B (zh) 2017-08-04
EA201490363A1 (ru) 2014-06-30
CA2843138A1 (en) 2013-01-31

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