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Publication of UY27501A1publicationCriticalpatent/UY27501A1/en
Formulaciones que contienen análogos de ciclosporina que son estructuralmente similares a la ciclosporina A, en particular mezclas isoméricas de análogos de ciclosporina que son estructuralmente similares a la ciclosporina A. Las formulaciones forman preconcentrados de microemulsiones estables y pueden proveer una biodisponibilidad superior de droga y/o pueden reducir uno o más efectos adversos asociados con la administración de ciclosporina. También se describen métodos para usar y preparar las formulaciones.Formulations containing cyclosporine analogs that are structurally similar to cyclosporin A, in particular isomeric mixtures of cyclosporin analogs that are structurally similar to cyclosporin A. The formulations form preconcentrated stable microemulsions and can provide superior drug bioavailability and / or they can reduce one or more adverse effects associated with the administration of cyclosporine. Methods for using and preparing the formulations are also described.
UY27501A2001-10-192002-10-17
NEW FORMULATIONS OF CYCLOSPORINE ANALOGS
UY27501A1
(en)