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Application filed by Emisphere Tech IncfiledCriticalEmisphere Tech Inc
Priority to UY26365ApriorityCriticalpatent/UY26365A1/en
Publication of UY26365A1publicationCriticalpatent/UY26365A1/en
La presente invención provee un solvato de alcohol, como solvato de etanol, de una sal de disodio de un agente de liberación de fórmula I, un hidrato de sal de disodio de un agente de liberación de dicha fórmula. Preferentemente los agentes de liberación incluyen, pero no están limitados a ácido N (5-clorosalisiloil) -8-aminocaprilico (5-CNAC), ácido N- (10-(2-hidroxibenzoil) amino) decanoico (SNAD),y caprilato de sodio N-(8-(2-hidroxibenzoil)amino (SNAC). También provee métodos de preparación de sal de disodio, el solvato de etanol, y el hidrato y composiciones que contiene a la sal de disodio, el solvato de etanol, y/o el hidrato.-The present invention provides an alcohol solvate, such as ethanol solvate, of a disodium salt of a release agent of formula I, a disodium salt hydrate of a release agent of said formula. Release agents preferably include, but are not limited to, N (5-chlorosalisiloyl) -8-aminocaprylic acid (5-CNAC), N- (10- (2-hydroxybenzoyl) amino) decanoic acid (SNAD), and sodium N- (8- (2-hydroxybenzoyl) amino (SNAC). Also provides methods of preparing disodium salt, the ethanol solvate, and the hydrate and compositions containing the disodium salt, the ethanol solvate, and / or hydrate.-
UY26365A2000-10-042000-10-04
DISODIUM SALTS, MONOHYDRATES, ETHANOL SOLVATES FOR THE RELEASE OF ACTIVE AGENTS
UY26365A1
(en)
PROCESS FOR MANUALLY MANUFACTURING HEMIPENTAHYDRATE AND MONOPENTAHYDRATE ACID 3-PIRIDIL-12HYDROXI-ETILIDEN-1, 1-BISFOPHOSNIC SODIUM AND PHARMACETIC COMPOSITION CONTAINING THEM
DERIVATIVES OF QUINOLINA. PROCEDURE FOR THE PREPARATION, PHARMACEUTICAL COMPOSITION THAT INCLUDES THEM, AND THE USE OF THEM FOR THE MANUFACTURE OF A MEDICINE
DERIVATIVES OF FENIL-4-TIAZOLES SUBSTITUTED, PROCEDURE FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND DERIVATIVES DEFENIL-4-TIAZOLES SUBSTITUTED USED IN SUCH PROCEDURE.