UY26365A1 - DISODIUM SALTS, MONOHYDRATES, ETHANOL SOLVATES FOR THE RELEASE OF ACTIVE AGENTS - Google Patents

DISODIUM SALTS, MONOHYDRATES, ETHANOL SOLVATES FOR THE RELEASE OF ACTIVE AGENTS

Info

Publication number
UY26365A1
UY26365A1 UY26365A UY26365A UY26365A1 UY 26365 A1 UY26365 A1 UY 26365A1 UY 26365 A UY26365 A UY 26365A UY 26365 A UY26365 A UY 26365A UY 26365 A1 UY26365 A1 UY 26365A1
Authority
UY
Uruguay
Prior art keywords
release
disodium salt
monohydrates
active agents
hydrate
Prior art date
Application number
UY26365A
Other languages
Spanish (es)
Inventor
William E Bay
Rajesh K Agarwal
Chaudhary Kiran
Majuru Shingai
Michael M Goldberg
Joanne P Corvino
Original Assignee
Emisphere Tech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Emisphere Tech Inc filed Critical Emisphere Tech Inc
Priority to UY26365A priority Critical patent/UY26365A1/en
Publication of UY26365A1 publication Critical patent/UY26365A1/en

Links

Abstract

La presente invención provee un solvato de alcohol, como solvato de etanol, de una sal de disodio de un agente de liberación de fórmula I, un hidrato de sal de disodio de un agente de liberación de dicha fórmula. Preferentemente los agentes de liberación incluyen, pero no están limitados a ácido N (5-clorosalisiloil) -8-aminocaprilico (5-CNAC), ácido N- (10-(2-hidroxibenzoil) amino) decanoico (SNAD),y caprilato de sodio N-(8-(2-hidroxibenzoil)amino (SNAC). También provee métodos de preparación de sal de disodio, el solvato de etanol, y el hidrato y composiciones que contiene a la sal de disodio, el solvato de etanol, y/o el hidrato.-The present invention provides an alcohol solvate, such as ethanol solvate, of a disodium salt of a release agent of formula I, a disodium salt hydrate of a release agent of said formula. Release agents preferably include, but are not limited to, N (5-chlorosalisiloyl) -8-aminocaprylic acid (5-CNAC), N- (10- (2-hydroxybenzoyl) amino) decanoic acid (SNAD), and sodium N- (8- (2-hydroxybenzoyl) amino (SNAC). Also provides methods of preparing disodium salt, the ethanol solvate, and the hydrate and compositions containing the disodium salt, the ethanol solvate, and / or hydrate.-

UY26365A 2000-10-04 2000-10-04 DISODIUM SALTS, MONOHYDRATES, ETHANOL SOLVATES FOR THE RELEASE OF ACTIVE AGENTS UY26365A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
UY26365A UY26365A1 (en) 2000-10-04 2000-10-04 DISODIUM SALTS, MONOHYDRATES, ETHANOL SOLVATES FOR THE RELEASE OF ACTIVE AGENTS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
UY26365A UY26365A1 (en) 2000-10-04 2000-10-04 DISODIUM SALTS, MONOHYDRATES, ETHANOL SOLVATES FOR THE RELEASE OF ACTIVE AGENTS

Publications (1)

Publication Number Publication Date
UY26365A1 true UY26365A1 (en) 2001-09-28

Family

ID=38812239

Family Applications (1)

Application Number Title Priority Date Filing Date
UY26365A UY26365A1 (en) 2000-10-04 2000-10-04 DISODIUM SALTS, MONOHYDRATES, ETHANOL SOLVATES FOR THE RELEASE OF ACTIVE AGENTS

Country Status (1)

Country Link
UY (1) UY26365A1 (en)

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Legal Events

Date Code Title Description
105 Application deemed to be withdrawn (no grant fee paid)

Effective date: 20171005