UA86777C2 - 6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors - Google Patents

6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors

Info

Publication number
UA86777C2
UA86777C2 UAA200603731A UAA200603731A UA86777C2 UA 86777 C2 UA86777 C2 UA 86777C2 UA A200603731 A UAA200603731 A UA A200603731A UA A200603731 A UAA200603731 A UA A200603731A UA 86777 C2 UA86777 C2 UA 86777C2
Authority
UA
Ukraine
Prior art keywords
quinoxalinones
quinolinones
adp
ribose
alkenyl
Prior art date
Application number
UAA200603731A
Other languages
Russian (ru)
Inventor
Доминик Жан-Пьер Мабир
Жером Эмиль Жорж Жильмон
Дун Якобус Алфонсус Джосепхус ван
Мария Викторина Франциска Сомерс
Валтер Боудевиджн Леопольд Воутерс
Original Assignee
Янссен Фармацевтика Н.В.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Янссен Фармацевтика Н.В. filed Critical Янссен Фармацевтика Н.В.
Publication of UA86777C2 publication Critical patent/UA86777C2/en

Links

Abstract

The present invention provides compounds of formula (I) and compounds of formula (I), (VII-a), as well as pharmaceutical compositions comprising said compounds and their use as PARP inhibitors wherein n, RR, R, R, R, R, R, R, Rand X have defined meanings.
UAA200603731A 2003-11-20 2004-11-18 6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors UA86777C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP0313028 2003-11-20

Publications (1)

Publication Number Publication Date
UA86777C2 true UA86777C2 (en) 2009-05-25

Family

ID=34957030

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200603731A UA86777C2 (en) 2003-11-20 2004-11-18 6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(adp-ribose) polymerase inhibitors

Country Status (3)

Country Link
CN (1) CN1882547B (en)
UA (1) UA86777C2 (en)
ZA (1) ZA200604075B (en)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2002864C (en) * 1988-11-29 1999-11-16 Eddy J. E. Freyne (1h-azol-1-ylmethyl) substituted quinoline, quinazoline or quinoxaline derivatives

Also Published As

Publication number Publication date
ZA200604075B (en) 2007-09-26
CN1882547A (en) 2006-12-20
CN1882547B (en) 2011-04-13

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