UA112586C2 - BENZIMIDAZOLPROLINE DERIVATIVES - Google Patents

BENZIMIDAZOLPROLINE DERIVATIVES

Info

Publication number
UA112586C2
UA112586C2 UAA201413919A UAA201413919A UA112586C2 UA 112586 C2 UA112586 C2 UA 112586C2 UA A201413919 A UAA201413919 A UA A201413919A UA A201413919 A UAA201413919 A UA A201413919A UA 112586 C2 UA112586 C2 UA 112586C2
Authority
UA
Ukraine
Prior art keywords
benzimidazolproline
derivatives
formula
compounds
pharmaceuticals
Prior art date
Application number
UAA201413919A
Other languages
Ukrainian (uk)
Inventor
Крістоф Босс
Христина Бротші
Маркус ГУДЕ
Бібія Хейдманн
Тьєрі Сіфферлен
Джоді Т. Вілльямс
Original Assignee
Актеліон Фармасьютікалз Лтд
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Актеліон Фармасьютікалз Лтд filed Critical Актеліон Фармасьютікалз Лтд
Priority claimed from PCT/IB2013/054567 external-priority patent/WO2013182972A1/en
Publication of UA112586C2 publication Critical patent/UA112586C2/en

Links

Abstract

Даний винахід належить до сполук формули (І), Формула (I)де Аr, R, R, R, R, Rта (R)приймають значення, як описано у описі, до їх одержання, до їх фармацевтично прийнятних солей та до їх застосування як фармацевтичних засобів, до фармацевтичних композицій, що містять одну або більше сполук формули (І), та особливо до їх застосування як антагоністів рецептора орексину.The present invention relates to compounds of formula (I), Formula (I) where Ar, R, R, R, R, R and (R) take the values as described in the description, to obtain them, to their pharmaceutically acceptable salts and to their use as pharmaceuticals, to pharmaceutical compositions containing one or more compounds of formula (I), and in particular to their use as orexin receptor antagonists.

UAA201413919A 2012-06-04 2013-03-06 BENZIMIDAZOLPROLINE DERIVATIVES UA112586C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12170748 2012-06-04
PCT/IB2013/054567 WO2013182972A1 (en) 2012-06-04 2013-06-03 Benzimidazole-proline derivatives

Publications (1)

Publication Number Publication Date
UA112586C2 true UA112586C2 (en) 2016-09-26

Family

ID=54338069

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201413919A UA112586C2 (en) 2012-06-04 2013-03-06 BENZIMIDAZOLPROLINE DERIVATIVES

Country Status (2)

Country Link
MA (1) MA37741B1 (en)
UA (1) UA112586C2 (en)

Also Published As

Publication number Publication date
MA20150282A2 (en) 2015-08-31
MA37741B1 (en) 2017-01-31

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