TR201907729T4 - Bir anti-çekirdekleştirici ajan içeren farmasötik bileşim. - Google Patents
Bir anti-çekirdekleştirici ajan içeren farmasötik bileşim. Download PDFInfo
- Publication number
- TR201907729T4 TR201907729T4 TR2019/07729T TR201907729T TR201907729T4 TR 201907729 T4 TR201907729 T4 TR 201907729T4 TR 2019/07729 T TR2019/07729 T TR 2019/07729T TR 201907729 T TR201907729 T TR 201907729T TR 201907729 T4 TR201907729 T4 TR 201907729T4
- Authority
- TR
- Turkey
- Prior art keywords
- nucleating agent
- pharmaceutical composition
- composition containing
- salt
- drug
- Prior art date
Links
- 230000002821 anti-nucleating effect Effects 0.000 title abstract 2
- 239000002667 nucleating agent Substances 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 239000003814 drug Substances 0.000 abstract 3
- 229940079593 drug Drugs 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 238000006243 chemical reaction Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000007909 solid dosage form Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Inorganic Chemistry (AREA)
- Virology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- AIDS & HIV (AREA)
- Communicable Diseases (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Katı dozaj formlarında oral uygulamaya yönelik olarak uygun farmasötik bileşimler açıklanır. Bileşimler, bir tuz formunda bir etkili miktarda bir ilaç bileşiği içerir, burada ilaç tuzu belirli pH koşulları altında ilaç bileşiğinin bir daha az çözünebilir formuna dönüştürülmesi ve bir anti-çekirdekleştirici ajan ile karakterize edilir.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US63285904P | 2004-12-03 | 2004-12-03 |
Publications (1)
Publication Number | Publication Date |
---|---|
TR201907729T4 true TR201907729T4 (tr) | 2019-06-21 |
Family
ID=36565788
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2019/07729T TR201907729T4 (tr) | 2004-12-03 | 2005-12-02 | Bir anti-çekirdekleştirici ajan içeren farmasötik bileşim. |
Country Status (9)
Country | Link |
---|---|
US (1) | US8771733B2 (tr) |
EP (2) | EP1819323B2 (tr) |
JP (3) | JP2008521929A (tr) |
CN (1) | CN101068533B (tr) |
AU (1) | AU2005311714B2 (tr) |
CA (1) | CA2588465C (tr) |
ES (1) | ES2727577T3 (tr) |
TR (1) | TR201907729T4 (tr) |
WO (1) | WO2006060681A2 (tr) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20070085702A (ko) * | 2004-12-03 | 2007-08-27 | 머크 앤드 캄파니 인코포레이티드 | Ugt1a1에 의해 대사된 약물의 약력학을 개선시키기위한 아타자나비르의 용도 |
MX2007006635A (es) | 2004-12-03 | 2007-06-19 | Merck & Co Inc | Formulacion farmaceutica de inhibidores dela carboxamida vih integrasa que contienen una composicion que controla la velocidad de liberacion. |
US8771733B2 (en) | 2004-12-03 | 2014-07-08 | Merck Sharp & Dohme Corp. | Pharmaceutical composition containing an anti-nucleating agent |
UA87884C2 (uk) | 2004-12-03 | 2009-08-25 | Мерк Энд Ко., Инк. | Безводна кристалічна калієва сіль інгібітора віл-інтегрази |
CN101595133B (zh) * | 2006-10-27 | 2012-11-14 | 比利时胶囊公司 | 羟丙基甲基纤维素硬胶囊及制备方法 |
CN101197832B (zh) * | 2007-12-13 | 2012-01-25 | 华为技术有限公司 | 一种实现iptv业务的方法、***、装置 |
EP2438062B1 (en) | 2009-06-02 | 2015-07-29 | Hetero Research Foundation | Process for the preparation of amorphous raltegravir potassium |
IN2012DN03377A (tr) * | 2009-10-26 | 2015-10-23 | Merck Sharp & Dohme | |
SI2796458T1 (en) * | 2010-04-01 | 2018-04-30 | Teva Pharmaceutical Industries Ltd. | CRYSTALINIC SODIUM RALTEGRAVIR SOLUTIONS |
US9968607B2 (en) * | 2011-04-25 | 2018-05-15 | Hetero Research Foundation | Pharmaceutical compositions of raltegravir, methods of preparation and methods of use therof |
WO2021148992A1 (en) | 2020-01-23 | 2021-07-29 | Lupin Limited | Pharmaceutical compositions of raltegravir |
US20230277587A1 (en) * | 2022-03-03 | 2023-09-07 | Dermacisen, S.A. | Food supplement for oral administration |
Family Cites Families (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4540566A (en) * | 1984-04-02 | 1985-09-10 | Forest Laboratories, Inc. | Prolonged release drug dosage forms based on modified low viscosity grade hydroxypropylmethylcellulose |
JPH0347124A (ja) * | 1989-04-20 | 1991-02-28 | Fujisawa Pharmaceut Co Ltd | 経口吸収用製剤 |
CA2019324C (en) * | 1989-07-10 | 1996-08-20 | Robert L. Jerzewski | Fosinopril tablet formulations |
JP2707023B2 (ja) * | 1992-07-01 | 1998-01-28 | 株式会社大塚製薬工場 | 経口吸収用製剤 |
WO2000018384A2 (en) † | 1998-09-28 | 2000-04-06 | Glaxo Group Limited | Antiviral combinations comprising (s)-2-ethyl-7-fluoro-3-oxo-3,4-dihydro-2h-quinoxaline-1-carboxylic acid isopropyl ester and amprenavir |
ATE411286T1 (de) * | 1998-12-25 | 2008-10-15 | Shionogi & Co | Aromatische heterocyclen mit hiv integrase inhibierenden eigenschaften |
GB9922963D0 (en) * | 1999-09-28 | 1999-12-01 | Pfizer Ltd | Polymorphic salt |
AU783981C (en) * | 2000-05-08 | 2007-05-03 | Janssen Pharmaceutica N.V. | HIV replication inhibitors |
US7115565B2 (en) † | 2001-01-18 | 2006-10-03 | Pharmacia & Upjohn Company | Chemotherapeutic microemulsion compositions of paclitaxel with improved oral bioavailability |
EP1441734B1 (en) | 2001-10-26 | 2007-02-28 | Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. | Dihydroxypyrimidine carboxamide inhibitors of hiv integrase |
US7169780B2 (en) | 2001-10-26 | 2007-01-30 | Istitute Di Ricerche Di Biologia Molecolare P. Angeletti S.P.A. | N-substituted hydroxypyrimidinone carboxamide inhibitors of HIV integrase |
AU2003220186A1 (en) † | 2002-04-10 | 2003-10-27 | Merck And Co., Inc. | Pharmaceutical compositions containing an hiv integrase inhibitor and a nonionic surfactant |
BR0317749A (pt) | 2002-12-27 | 2005-11-22 | Angeletti P Ist Richerche Bio | Composto, composição farmacêutica, e, uso de um composto |
US20040224916A1 (en) † | 2003-01-14 | 2004-11-11 | Gilead Sciences, Inc. | Compositions and methods for combination antiviral therapy |
MX2007006635A (es) * | 2004-12-03 | 2007-06-19 | Merck & Co Inc | Formulacion farmaceutica de inhibidores dela carboxamida vih integrasa que contienen una composicion que controla la velocidad de liberacion. |
US8771733B2 (en) | 2004-12-03 | 2014-07-08 | Merck Sharp & Dohme Corp. | Pharmaceutical composition containing an anti-nucleating agent |
UA87884C2 (uk) | 2004-12-03 | 2009-08-25 | Мерк Энд Ко., Инк. | Безводна кристалічна калієва сіль інгібітора віл-інтегрази |
KR20070085702A (ko) | 2004-12-03 | 2007-08-27 | 머크 앤드 캄파니 인코포레이티드 | Ugt1a1에 의해 대사된 약물의 약력학을 개선시키기위한 아타자나비르의 용도 |
US9968607B2 (en) | 2011-04-25 | 2018-05-15 | Hetero Research Foundation | Pharmaceutical compositions of raltegravir, methods of preparation and methods of use therof |
-
2005
- 2005-12-02 US US11/792,190 patent/US8771733B2/en active Active
- 2005-12-02 JP JP2007544548A patent/JP2008521929A/ja active Pending
- 2005-12-02 EP EP05852790.4A patent/EP1819323B2/en active Active
- 2005-12-02 EP EP16198994.2A patent/EP3165220B1/en active Active
- 2005-12-02 ES ES16198994T patent/ES2727577T3/es active Active
- 2005-12-02 TR TR2019/07729T patent/TR201907729T4/tr unknown
- 2005-12-02 CA CA2588465A patent/CA2588465C/en not_active Expired - Fee Related
- 2005-12-02 WO PCT/US2005/043675 patent/WO2006060681A2/en active Application Filing
- 2005-12-02 CN CN2005800415795A patent/CN101068533B/zh not_active Expired - Fee Related
- 2005-12-02 AU AU2005311714A patent/AU2005311714B2/en not_active Ceased
-
2012
- 2012-05-21 JP JP2012116010A patent/JP2012184250A/ja active Pending
- 2012-11-29 JP JP2012260995A patent/JP2013063999A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
AU2005311714A1 (en) | 2006-06-08 |
EP1819323B2 (en) | 2023-03-22 |
AU2005311714B2 (en) | 2010-09-30 |
JP2008521929A (ja) | 2008-06-26 |
CN101068533B (zh) | 2011-04-27 |
ES2727577T3 (es) | 2019-10-17 |
EP3165220A1 (en) | 2017-05-10 |
EP1819323A2 (en) | 2007-08-22 |
CA2588465A1 (en) | 2006-06-08 |
JP2012184250A (ja) | 2012-09-27 |
US8771733B2 (en) | 2014-07-08 |
EP1819323A4 (en) | 2012-07-18 |
US20080118559A1 (en) | 2008-05-22 |
WO2006060681A2 (en) | 2006-06-08 |
JP2013063999A (ja) | 2013-04-11 |
EP1819323B1 (en) | 2016-11-16 |
WO2006060681A3 (en) | 2006-10-12 |
EP3165220B1 (en) | 2019-04-03 |
CA2588465C (en) | 2013-10-01 |
CN101068533A (zh) | 2007-11-07 |
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