TR201821285T4 - CCR3 antagonisti içeren farmasötik formülasyonlar. - Google Patents
CCR3 antagonisti içeren farmasötik formülasyonlar. Download PDFInfo
- Publication number
- TR201821285T4 TR201821285T4 TR2018/21285T TR201821285T TR201821285T4 TR 201821285 T4 TR201821285 T4 TR 201821285T4 TR 2018/21285 T TR2018/21285 T TR 2018/21285T TR 201821285 T TR201821285 T TR 201821285T TR 201821285 T4 TR201821285 T4 TR 201821285T4
- Authority
- TR
- Turkey
- Prior art keywords
- pharmaceutical formulations
- formulations containing
- ccr3 antagonist
- ccr3
- antagonist
- Prior art date
Links
- NDZYPHLNJZSQJY-QNWVGRARSA-N 1-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-3-[(1r,2s)-2-[[(3s)-3-[(4-fluorophenyl)methyl]piperidin-1-yl]methyl]cyclohexyl]urea Chemical compound CC1=C(C(=O)C)SC(NC(=O)N[C@H]2[C@@H](CCCC2)CN2C[C@H](CC=3C=CC(F)=CC=3)CCC2)=N1 NDZYPHLNJZSQJY-QNWVGRARSA-N 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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Abstract
Mevcut buluş, CCR3 antagonisti içeren farmasötik formülasyonlar ile ilgilidir.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12163078 | 2012-04-04 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR201821285T4 true TR201821285T4 (tr) | 2019-01-21 |
Family
ID=49292482
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2018/21285T TR201821285T4 (tr) | 2012-04-04 | 2013-04-02 | CCR3 antagonisti içeren farmasötik formülasyonlar. |
Country Status (30)
| Country | Link |
|---|---|
| US (3) | US10213421B2 (tr) |
| EP (3) | EP3970693A1 (tr) |
| JP (4) | JP6320990B2 (tr) |
| KR (2) | KR102338465B1 (tr) |
| CN (1) | CN104203213A (tr) |
| AR (1) | AR090596A1 (tr) |
| AU (1) | AU2013245028B2 (tr) |
| BR (1) | BR112014024479A8 (tr) |
| CA (1) | CA2869058C (tr) |
| CL (1) | CL2014002524A1 (tr) |
| CY (1) | CY1121137T1 (tr) |
| DK (2) | DK3524230T3 (tr) |
| EA (1) | EA027627B1 (tr) |
| ES (2) | ES2898179T3 (tr) |
| HR (1) | HRP20190069T1 (tr) |
| HU (2) | HUE056943T2 (tr) |
| IL (1) | IL234299A (tr) |
| IN (1) | IN2014DN07082A (tr) |
| LT (1) | LT2833864T (tr) |
| MX (1) | MX358307B (tr) |
| NZ (1) | NZ628993A (tr) |
| PH (1) | PH12014502241A1 (tr) |
| PL (2) | PL3524230T3 (tr) |
| PT (2) | PT2833864T (tr) |
| RS (1) | RS58360B1 (tr) |
| SI (1) | SI2833864T1 (tr) |
| TR (1) | TR201821285T4 (tr) |
| TW (1) | TW201400115A (tr) |
| UY (1) | UY34730A (tr) |
| WO (1) | WO2013149987A1 (tr) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8278302B2 (en) | 2009-04-08 | 2012-10-02 | Boehringer Ingelheim International Gmbh | Substituted piperidines as CCR3 antagonists |
| UA109290C2 (uk) | 2010-10-07 | 2015-08-10 | Спільні кристали і солі інгібіторів ccr3 | |
| AR090566A1 (es) | 2012-04-02 | 2014-11-19 | Boehringer Ingelheim Int | Proceso para la produccion de inhibidores de crr |
| US20130261153A1 (en) * | 2012-04-03 | 2013-10-03 | Boehringer Ingelheim International Gmbh | Use of ccr3-inhibitors |
| US10213421B2 (en) | 2012-04-04 | 2019-02-26 | Alkahest, Inc. | Pharmaceutical formulations comprising CCR3 antagonists |
| KR102658724B1 (ko) * | 2017-04-05 | 2024-04-18 | 알카헤스트 인코포레이티드 | Ccr3-저해제를 사용하여 망막-관련 질병을 치료하는 방법 및 조성물 |
| CN110636844A (zh) * | 2017-04-05 | 2019-12-31 | 万能溶剂有限公司 | 使用ccr3-抑制剂治疗衰老相关损伤的方法及组合物 |
| SG11202002437VA (en) * | 2017-10-13 | 2020-04-29 | Alkahest Inc | Methods and compositions for treating pruritus, xerosis, and associated disease using ccr3-inhibitors |
| BR112020023001A2 (pt) | 2018-05-15 | 2021-02-02 | Alkahest, Inc. | tratamento de doença associada ao envelhecimento com moduladores da leucotrieno a4 hidrolase |
| JP2022502441A (ja) * | 2018-09-26 | 2022-01-11 | アルカヘスト，インコーポレイテッド | Ｃｃｒ３阻害剤を用いて、加齢性機能障害を治療するための方法および組成物 |
| CN115989200A (zh) | 2020-08-27 | 2023-04-18 | Ａｇｃ株式会社 | 无碱玻璃和玻璃板 |
| AU2022376563A1 (en) | 2021-11-01 | 2023-12-07 | Alkahest, Inc. | Benzodioxane modulators of leukotriene a4 hydrolase (lta4h) for prevention and treatment of aging-associated diseases |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE7907121L (sv) | 1979-08-27 | 1981-02-28 | Astra Laekemedel Ab | Ftalimidinderivat |
| US4992277A (en) | 1989-08-25 | 1991-02-12 | Schering Corporation | Immediate release diltiazem formulation |
| JP2807577B2 (ja) | 1990-06-15 | 1998-10-08 | エーザイ株式会社 | 環状アミド誘導体 |
| IL116539A (en) * | 1995-01-06 | 2002-02-10 | Noven Pharma | Preparations given through the skin of unstable anti-acid drugs |
| JP2001524131A (ja) * | 1997-05-09 | 2001-11-27 | セイジ、ファーマスーティカルズ、インク | 安定な経口医薬品剤形 |
| EP1047675A1 (en) | 1998-01-21 | 2000-11-02 | Millennium Pharmaceuticals, Inc. | Chemokine receptor antagonists and methods of use therefor |
| JP2002501898A (ja) | 1998-02-02 | 2002-01-22 | メルク エンド カムパニー インコーポレーテッド | ケモカイン受容体活性の環状アミン調節剤 |
| US6140349A (en) | 1998-02-02 | 2000-10-31 | Merck & Co., Inc. | Cyclic amine modulators of chemokine receptor activity |
| SE9802973D0 (sv) | 1998-09-03 | 1998-09-03 | Astra Ab | Immediate release tablet |
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