TR201009399A2 - Rapidly soluble effervescent rosuvastatin formulations. - Google Patents

Rapidly soluble effervescent rosuvastatin formulations.

Info

Publication number
TR201009399A2
TR201009399A2 TR2010/09399A TR201009399A TR201009399A2 TR 201009399 A2 TR201009399 A2 TR 201009399A2 TR 2010/09399 A TR2010/09399 A TR 2010/09399A TR 201009399 A TR201009399 A TR 201009399A TR 201009399 A2 TR201009399 A2 TR 201009399A2
Authority
TR
Turkey
Prior art keywords
rapidly soluble
soluble effervescent
rosuvastatin
formulations
rosuvastatin formulations
Prior art date
Application number
TR2010/09399A
Other languages
Turkish (tr)
Inventor
Bi̇lgi̇ç Mahmut
Original Assignee
Bi̇lgi̇ç Mahmut
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bi̇lgi̇ç Mahmut filed Critical Bi̇lgi̇ç Mahmut
Priority to TR2010/09399A priority Critical patent/TR201009399A2/en
Priority to PCT/TR2011/000248 priority patent/WO2012064306A2/en
Publication of TR201009399A2 publication Critical patent/TR201009399A2/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007Effervescent
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Medicinal Preparation (AREA)

Abstract

Mevcut buluş, etken madde olarak rosuvastatin ve/veya farmasötik kabul edilebilir bir tuzunu içeren hızlı çözünen efervesan formülasyonlara ilişkindir.The present invention relates to fast dissolving effervescent formulations containing rosuvastatin and / or a pharmaceutically acceptable salt thereof as an active ingredient.

TR2010/09399A 2010-11-11 2010-11-11 Rapidly soluble effervescent rosuvastatin formulations. TR201009399A2 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
TR2010/09399A TR201009399A2 (en) 2010-11-11 2010-11-11 Rapidly soluble effervescent rosuvastatin formulations.
PCT/TR2011/000248 WO2012064306A2 (en) 2010-11-11 2011-11-03 Effervescent formulations of rosuvastatin

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
TR2010/09399A TR201009399A2 (en) 2010-11-11 2010-11-11 Rapidly soluble effervescent rosuvastatin formulations.

Publications (1)

Publication Number Publication Date
TR201009399A2 true TR201009399A2 (en) 2012-05-21

Family

ID=45607337

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2010/09399A TR201009399A2 (en) 2010-11-11 2010-11-11 Rapidly soluble effervescent rosuvastatin formulations.

Country Status (2)

Country Link
TR (1) TR201009399A2 (en)
WO (1) WO2012064306A2 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112017005362A2 (en) 2014-09-17 2018-01-23 Steerlife India Private Ltd composition, oral solid dosage form, process for preparing porous effervescent granules, dual screw processor, and porous effervescent granules.
US11219594B2 (en) 2015-12-12 2022-01-11 Steerlife India Private Limited Effervescent compositions of metformin and processes for preparation thereof

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2648897B2 (en) 1991-07-01 1997-09-03 塩野義製薬株式会社 Pyrimidine derivatives
EP0872544A1 (en) * 1997-04-14 1998-10-21 The Procter & Gamble Company Dry effervescent granules and granular compositions comprising the same
US20070048375A1 (en) * 2003-12-19 2007-03-01 Wolfgang Wiehl Effervescent preparation of a basic medicinally active substance
WO2006037348A1 (en) * 2004-10-01 2006-04-13 Lifecycle Pharma A/S Pharmaceutical compositions comprising fenofibrate and a statin
WO2006134604A1 (en) * 2005-06-15 2006-12-21 Hetero Drugs Limited Combination composition of cholesterol absorption inhibitor and 3-hydroxy-3-methylglutaryl-coenzyme a (hmg-coa) reductase inhibitor
WO2008062476A2 (en) * 2006-10-31 2008-05-29 Glenmark Pharmaceutical Limited Pharmaceutical composition comprising rosuvastatin or pharmaceutically accepatble salts thereof
US20090304602A1 (en) * 2008-06-06 2009-12-10 Tuchinsky David B Nutritional supplement
PL386051A1 (en) * 2008-09-09 2010-03-15 Zakłady Farmaceutyczne POLPHARMA Spółka Akcyjna Stable, oral compound pharmaceutical containing pharmaceutically permissible content of [(E)-7-[4-(4-fluorphenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino]pyrimidine-5-yl] (3R,5S)-3,5-dihydroxy-hept-6-enoate acid salt
CN101618215A (en) * 2009-08-16 2010-01-06 王丽燕 Pharmaceutical composition containing calcium blocker, AII receptor blocker and statins
TR201009397A2 (en) * 2010-11-11 2012-05-21 Bi̇lgi̇ç Mahmut Pharmaceutical compositions containing rosuvastatin.
EP2575757A1 (en) * 2010-06-03 2013-04-10 Mahmut Bilgic Water soluble formulation comprising a combination of amlodipine and a statin

Also Published As

Publication number Publication date
WO2012064306A2 (en) 2012-05-18
WO2012064306A3 (en) 2012-08-09

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