TR200401875T2 - Endoparazit öldürücü bileşimler - Google Patents
Endoparazit öldürücü bileşimlerInfo
- Publication number
- TR200401875T2 TR200401875T2 TR2004/01875T TR200401875T TR200401875T2 TR 200401875 T2 TR200401875 T2 TR 200401875T2 TR 2004/01875 T TR2004/01875 T TR 2004/01875T TR 200401875 T TR200401875 T TR 200401875T TR 200401875 T2 TR200401875 T2 TR 200401875T2
- Authority
- TR
- Turkey
- Prior art keywords
- endoparasiticidal
- compounds
- piperazines
- amino acids
- cyclic depsipeptides
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 3
- 108010002156 Depsipeptides Proteins 0.000 abstract 2
- GLUUGHFHXGJENI-UHFFFAOYSA-N Piperazine Chemical compound C1CNCCN1 GLUUGHFHXGJENI-UHFFFAOYSA-N 0.000 abstract 2
- 150000001413 amino acids Chemical class 0.000 abstract 2
- BVKZGUZCCUSVTD-UHFFFAOYSA-N carbonic acid Chemical class OC(O)=O BVKZGUZCCUSVTD-UHFFFAOYSA-N 0.000 abstract 2
- 150000004885 piperazines Chemical class 0.000 abstract 2
- 230000000694 effects Effects 0.000 abstract 1
- 230000001939 inductive effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/15—Depsipeptides; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Bu bulus, endoparazit öldürücü bilesimlerde, halka üniteleri olarak amino asitlerden ve hidroksikarboksilik asitlerden olusan ve 24 halka atomuna sahip olan siklik depsipeptitlerin endoparazit öldürücü etkisinin arttirilmasi için piperazinlerin kullanimina ve endoparazit öldürücü bilesimlerin üretilmesi için halka üniteleri olarak amino asitlerden ve hidroksikarboksilik asitlerden olusan ve 24 halka atomuna sahip olan siklik depsipeptitlerin ve piperazinlerin kullanimina iliskindir.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19921887A DE19921887A1 (de) | 1999-05-12 | 1999-05-12 | Endoparasitizide Mittel |
Publications (1)
Publication Number | Publication Date |
---|---|
TR200401875T2 true TR200401875T2 (tr) | 2005-01-24 |
Family
ID=7907825
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2001/03240T TR200103240T2 (tr) | 1999-05-12 | 2000-05-04 | Endoparazit öldürücü bileşimler. |
TR2004/01875T TR200401875T2 (tr) | 1999-05-12 | 2000-05-04 | Endoparazit öldürücü bileşimler |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2001/03240T TR200103240T2 (tr) | 1999-05-12 | 2000-05-04 | Endoparazit öldürücü bileşimler. |
Country Status (26)
Country | Link |
---|---|
EP (1) | EP1189615B1 (tr) |
JP (1) | JP2002544224A (tr) |
KR (1) | KR100704717B1 (tr) |
CN (1) | CN1224391C (tr) |
AT (1) | ATE258795T1 (tr) |
AU (1) | AU768910B2 (tr) |
BR (1) | BR0010499A (tr) |
CA (1) | CA2373827C (tr) |
CZ (1) | CZ300782B6 (tr) |
DE (2) | DE19921887A1 (tr) |
DK (1) | DK1189615T3 (tr) |
ES (1) | ES2211558T3 (tr) |
HK (1) | HK1047228B (tr) |
HR (1) | HRP20010918B1 (tr) |
HU (1) | HUP0201201A3 (tr) |
MX (1) | MXPA01011455A (tr) |
NO (1) | NO328870B1 (tr) |
PL (1) | PL200951B1 (tr) |
PT (1) | PT1189615E (tr) |
RS (1) | RS50169B (tr) |
RU (1) | RU2250779C2 (tr) |
SK (1) | SK285494B6 (tr) |
TR (2) | TR200103240T2 (tr) |
UA (1) | UA72520C2 (tr) |
WO (1) | WO2000069425A2 (tr) |
ZA (1) | ZA200108238B (tr) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10008128A1 (de) * | 2000-02-22 | 2001-08-23 | Bayer Ag | Endoparasitizide Mittel |
DE10358525A1 (de) * | 2003-12-13 | 2005-07-07 | Bayer Healthcare Ag | Endoparasitizide Mittel zur topischen Applikation |
KR101671325B1 (ko) * | 2015-01-09 | 2016-11-02 | 한국생명공학연구원 | 신규한 고리형 뎁시펩타이드계 화합물, 이의 제조방법 및 이를 유효성분으로 함유하는 항균용 약학적 조성물 |
RS62130B1 (sr) | 2015-05-20 | 2021-08-31 | Boehringer Ingelheim Animal Health Usa Inc | Antihelmintička depsipeptidna jedinjenja |
RU2715556C2 (ru) | 2015-12-28 | 2020-03-02 | Мериал, Инк. | Противогельминтные депсипептидные соединения |
WO2018093920A1 (en) | 2016-11-16 | 2018-05-24 | Merial, Inc. | Anthelmintic depsipeptide compounds |
WO2022051862A1 (en) * | 2020-09-11 | 2022-03-17 | The Governing Council Of The University Of Toronto | Piperazinyl compounds and methods for treating nematode infections |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZA842571B (en) * | 1983-04-07 | 1985-11-27 | Merck & Co Inc | Novel synergistic antiparasitic combinations |
JPS6471865A (en) * | 1987-09-11 | 1989-03-16 | Nichibai Boeki Kk | 1-alkylcarbamoyl-4-methylpiperazine derivative |
NO176766C (no) * | 1989-02-07 | 1995-05-24 | Meiji Seika Kaisha | Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet |
ES2170101T3 (es) * | 1993-09-06 | 2002-08-01 | Fujisawa Pharmaceutical Co | Compuesto ciclodepsipeptido. |
DE4400464A1 (de) * | 1994-01-11 | 1995-07-13 | Bayer Ag | Endoparasitizide Mittel |
DE19520275A1 (de) * | 1995-06-02 | 1996-12-05 | Bayer Ag | Endoparasitizide Mittel |
KR19990044489A (ko) * | 1995-09-07 | 1999-06-25 | 로렌스 티. 마이젠헬더 | 환식 구충제 |
AU6229898A (en) * | 1997-02-19 | 1998-09-09 | Bayer Aktiengesellschaft | Derivatives of cyclodepsipeptide, pf1022 substance |
CN1076349C (zh) * | 1997-06-04 | 2001-12-19 | 拜尔公司 | 去氧环缩肽及其防治体内寄生虫的用途 |
WO2000008047A1 (fr) * | 1998-08-04 | 2000-02-17 | Nisshin Flour Milling Co., Ltd. | Derives de depsipeptides comportant des noyaux de piperazinone |
-
1999
- 1999-05-12 DE DE19921887A patent/DE19921887A1/de not_active Withdrawn
-
2000
- 2000-04-05 UA UA2001128532A patent/UA72520C2/uk unknown
- 2000-05-04 CN CNB00807450XA patent/CN1224391C/zh not_active Expired - Fee Related
- 2000-05-04 EP EP00940235A patent/EP1189615B1/de not_active Expired - Lifetime
- 2000-05-04 SK SK1626-2001A patent/SK285494B6/sk not_active IP Right Cessation
- 2000-05-04 AU AU55237/00A patent/AU768910B2/en not_active Ceased
- 2000-05-04 MX MXPA01011455A patent/MXPA01011455A/es active IP Right Grant
- 2000-05-04 AT AT00940235T patent/ATE258795T1/de active
- 2000-05-04 CZ CZ20014060A patent/CZ300782B6/cs not_active IP Right Cessation
- 2000-05-04 BR BR0010499-0A patent/BR0010499A/pt not_active Application Discontinuation
- 2000-05-04 PT PT00940235T patent/PT1189615E/pt unknown
- 2000-05-04 JP JP2000617884A patent/JP2002544224A/ja active Pending
- 2000-05-04 DE DE50005213T patent/DE50005213D1/de not_active Expired - Lifetime
- 2000-05-04 RS YUP-805/01A patent/RS50169B/sr unknown
- 2000-05-04 TR TR2001/03240T patent/TR200103240T2/tr unknown
- 2000-05-04 KR KR1020017013555A patent/KR100704717B1/ko not_active IP Right Cessation
- 2000-05-04 TR TR2004/01875T patent/TR200401875T2/tr unknown
- 2000-05-04 CA CA002373827A patent/CA2373827C/en not_active Expired - Fee Related
- 2000-05-04 RU RU2001133380/15A patent/RU2250779C2/ru not_active IP Right Cessation
- 2000-05-04 DK DK00940235T patent/DK1189615T3/da active
- 2000-05-04 PL PL351376A patent/PL200951B1/pl not_active IP Right Cessation
- 2000-05-04 HU HU0201201A patent/HUP0201201A3/hu unknown
- 2000-05-04 ES ES00940235T patent/ES2211558T3/es not_active Expired - Lifetime
- 2000-05-04 WO PCT/EP2000/004014 patent/WO2000069425A2/de active IP Right Grant
-
2001
- 2001-10-08 ZA ZA200108238A patent/ZA200108238B/xx unknown
- 2001-11-05 NO NO20015398A patent/NO328870B1/no not_active IP Right Cessation
- 2001-12-11 HR HR20010918A patent/HRP20010918B1/xx not_active IP Right Cessation
-
2002
- 2002-11-26 HK HK02108544.2A patent/HK1047228B/zh not_active IP Right Cessation
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