TR200002790T2 - 5-(4-(2-(N-metil-N-2-piridil) amino)etoksi) benzil)tiazolidin-2,4-dion içeren terkip - Google Patents

5-(4-(2-(N-metil-N-2-piridil) amino)etoksi) benzil)tiazolidin-2,4-dion içeren terkip

Info

Publication number
TR200002790T2
TR200002790T2 TR2000/02790T TR200002790T TR200002790T2 TR 200002790 T2 TR200002790 T2 TR 200002790T2 TR 2000/02790 T TR2000/02790 T TR 2000/02790T TR 200002790 T TR200002790 T TR 200002790T TR 200002790 T2 TR200002790 T2 TR 200002790T2
Authority
TR
Turkey
Prior art keywords
thiazolidin
dione
pyridyl
ethoxy
benzyl
Prior art date
Application number
TR2000/02790T
Other languages
English (en)
Turkish (tr)
Inventor
Patel Jai
Ross Hamish
Price Robin
Roger Granett Jeffrey
Nigel Wray Paul
Original Assignee
Smithkline Beecham P.L.C.
Smithkline Beecham Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9712851.6A external-priority patent/GB9712851D0/en
Application filed by Smithkline Beecham P.L.C., Smithkline Beecham Corporation filed Critical Smithkline Beecham P.L.C.
Publication of TR200002790T2 publication Critical patent/TR200002790T2/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
TR2000/02790T 1997-06-05 1998-06-02 5-(4-(2-(N-metil-N-2-piridil) amino)etoksi) benzil)tiazolidin-2,4-dion içeren terkip TR200002790T2 (tr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9711683.4A GB9711683D0 (en) 1997-06-05 1997-06-05 Composition
GBGB9712851.6A GB9712851D0 (en) 1997-06-18 1997-06-18 Composition

Publications (1)

Publication Number Publication Date
TR200002790T2 true TR200002790T2 (tr) 2001-11-21

Family

ID=26311662

Family Applications (2)

Application Number Title Priority Date Filing Date
TR2000/02790T TR200002790T2 (tr) 1997-06-05 1998-06-02 5-(4-(2-(N-metil-N-2-piridil) amino)etoksi) benzil)tiazolidin-2,4-dion içeren terkip
TR1999/02963T TR199902963T2 (xx) 1997-06-05 1998-06-02 5-$4-$2-(N-Metil-N-2-Piridil)Amino) Etoksi]Benzil]Tiazolidin-2,4-Dion i�eren terkip

Family Applications After (1)

Application Number Title Priority Date Filing Date
TR1999/02963T TR199902963T2 (xx) 1997-06-05 1998-06-02 5-$4-$2-(N-Metil-N-2-Piridil)Amino) Etoksi]Benzil]Tiazolidin-2,4-Dion i�eren terkip

Country Status (29)

Country Link
EP (1) EP0998284A1 (xx)
JP (1) JP2001521553A (xx)
KR (1) KR20010013410A (xx)
CN (3) CN1526391A (xx)
AP (1) AP1214A (xx)
AR (2) AR015120A1 (xx)
AU (1) AU8215098A (xx)
BG (1) BG104048A (xx)
BR (1) BR9810405A (xx)
CA (2) CA2333352A1 (xx)
CO (1) CO4940400A1 (xx)
DZ (1) DZ2510A1 (xx)
EA (1) EA002384B1 (xx)
GB (1) GB9711683D0 (xx)
HU (1) HUP0004070A3 (xx)
ID (1) ID24264A (xx)
IL (1) IL133074A0 (xx)
MX (1) MXPA99011322A (xx)
NO (2) NO995938L (xx)
NZ (2) NZ523725A (xx)
OA (1) OA11306A (xx)
PE (1) PE78899A1 (xx)
PL (1) PL337201A1 (xx)
SK (1) SK164899A3 (xx)
TR (2) TR200002790T2 (xx)
TW (1) TW570797B (xx)
UY (1) UY25032A1 (xx)
WO (1) WO1998055122A1 (xx)
ZA (2) ZA9811572B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL351684A1 (en) 1999-04-23 2003-06-02 Smithkline Beecham Plc Polymorph of 5−[4−[2− (n−methyl−n−( 2−pyridyl)amino) ethoxy]benzyl] thiazolidine−2,4−dione, maleic acid salt
BR0009934A (pt) 1999-04-23 2002-06-04 Smithkline Beecham Plc Produto farmacêutico
US20040248945A1 (en) 1999-04-23 2004-12-09 Smithkline Beecham P.L.C. Thiazolidinedione derivative and its use as antidiabetic
GB0021978D0 (en) 2000-09-07 2000-10-25 Smithkline Beecham Plc Novel pharmaceutical
GB0127805D0 (en) * 2001-11-20 2002-01-09 Smithkline Beecham Plc Pharmaceutical composition
GB0129871D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
AU2002350965A1 (en) * 2001-12-13 2003-06-23 Smithkline Beecham Plc Toluenesulfonate hydrates of a thiazolidinedione derivative
GB0129876D0 (en) * 2001-12-13 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
GB0130509D0 (en) * 2001-12-20 2002-02-06 Smithkline Beecham Plc Novel pharmaceutical
US7435741B2 (en) 2006-05-09 2008-10-14 Teva Pharmaceutical Industries, Ltd. 2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
EP1854794A1 (en) * 2006-05-09 2007-11-14 Teva Pharmaceutical Industries Ltd. 2-N-{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2-4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
WO2015008234A1 (en) * 2013-07-17 2015-01-22 Glenmark Pharmaceuticals S.A. Bicyclic heterocyclic compounds as ror gamma modulators

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE186724T1 (de) * 1987-09-04 1999-12-15 Beecham Group Plc Substituierte thiazolidindionderivate
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
SG47100A1 (en) * 1994-02-10 1998-03-20 Smithkline Beecham Plc Use of insulin sensitisers for treating renal diseases
WO1997005875A2 (en) * 1995-08-10 1997-02-20 Warner-Lambert Company A method of reducing the amount of exogenous insulin administered to a patient having noninsulin-dependent diabetes mellitus
AU7604596A (en) * 1995-11-17 1997-06-11 Warner-Lambert Company A method of treating myotonic dystrophy
IL120443A (en) * 1996-03-18 2000-07-16 Sankyo Co Use of an insulin sensitizer for the manufacture of a medicament for the treatment or prophylaxis of pancreatitis
WO1998002159A1 (en) * 1996-07-12 1998-01-22 Smithkline Beecham Plc Novel treatment of leptine resistance

Also Published As

Publication number Publication date
BG104048A (bg) 2000-07-31
NO995938L (no) 2000-02-02
NO995938D0 (no) 1999-12-03
NZ523725A (en) 2004-09-24
OA11306A (en) 2003-10-22
SK164899A3 (en) 2000-11-07
CN1430959A (zh) 2003-07-23
HUP0004070A3 (en) 2002-03-28
CA2292629A1 (en) 1998-12-10
EA199901116A1 (ru) 2000-06-26
EA002384B1 (ru) 2002-04-25
WO1998055122A1 (en) 1998-12-10
CN1259050A (zh) 2000-07-05
NZ513922A (en) 2001-09-28
ID24264A (id) 2000-07-13
BR9810405A (pt) 2000-08-29
CA2333352A1 (en) 1998-12-10
HUP0004070A2 (hu) 2002-02-28
AU8215098A (en) 1998-12-21
PL337201A1 (en) 2000-08-14
CN1526391A (zh) 2004-09-08
DZ2510A1 (fr) 2003-01-25
AR015120A1 (es) 2001-04-18
IL133074A0 (en) 2001-03-19
UY25032A1 (es) 1998-11-26
TR199902963T2 (xx) 2000-02-21
AP1214A (en) 2003-10-08
KR20010013410A (ko) 2001-02-26
GB9711683D0 (en) 1997-08-06
ZA984826B (en) 1999-08-03
AP9901696A0 (en) 1999-12-31
PE78899A1 (es) 1999-10-22
JP2001521553A (ja) 2001-11-06
EP0998284A1 (en) 2000-05-10
NO20040738L (no) 2000-02-02
ZA9811572B (en) 1999-07-22
MXPA99011322A (es) 2004-12-02
CA2292629C (en) 2004-01-06
TW570797B (en) 2004-01-11
CO4940400A1 (es) 2000-07-24
CN1112926C (zh) 2003-07-02
AR008198A1 (es) 1999-12-29

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