TNSN01083A1 - 2-AMINOCARBONYL-9H-PURINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM - Google Patents

2-AMINOCARBONYL-9H-PURINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM

Info

Publication number
TNSN01083A1
TNSN01083A1 TNTNSN01083A TNSN01083A TNSN01083A1 TN SN01083 A1 TNSN01083 A1 TN SN01083A1 TN TNSN01083 A TNTNSN01083 A TN TNSN01083A TN SN01083 A TNSN01083 A TN SN01083A TN SN01083 A1 TNSN01083 A1 TN SN01083A1
Authority
TN
Tunisia
Prior art keywords
preparation
processes
compositions containing
aminocarbonyl
purine derivatives
Prior art date
Application number
TNTNSN01083A
Other languages
French (fr)
Inventor
John Mantell Simon
Thomas Stephenson Peter
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0024920A external-priority patent/GB0024920D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of TNSN01083A1 publication Critical patent/TNSN01083A1/en

Links

Abstract

LA PRESENTE INVENTION CONCERNE DES COMPOSES DE FORMULE (I) : DANS LAQUELLE R1, R2, R3, R4, R5, R15, X ET Y REPRESENTENT DIVERS RADICAUX. ELLE CONCERNE EGALEMENT DES PROCEDES POUR LEUR PREPARATION ET LES INTERMEDIAIRES UTILISES DANS CETTE PREPARATION, AINSI QUE DES COMPOSITIONS LES CONTENANT. APPLICATION : UTILISATION DE CES COMPOSES ET COMPOSITIONS COMME AGONISTES DES RECEPTEURS A2a D'ADENOSINE, POUR LE TRAITEMENT DE DIVERSES MALADIES, NOTAMMENT DU TRACTUS RESPIRATOIRE.THE PRESENT INVENTION CONCERNS COMPOUNDS OF FORMULA (I): IN WHICH R1, R2, R3, R4, R5, R15, X AND Y REPRESENT VARIOUS RADICALS. IT ALSO CONCERNS PROCESSES FOR THEIR PREPARATION AND THE INTERMEDIATES USED IN THIS PREPARATION, AS WELL AS COMPOSITIONS CONTAINING THEM. APPLICATION: USE OF THESE COMPOUNDS AND COMPOSITIONS AS AGONISTS OF A2a ADENOSINE RECEPTORS, FOR THE TREATMENT OF VARIOUS DISEASES, ESPECIALLY OF THE RESPIRATORY TRACT.

TNTNSN01083A 2000-06-06 2001-06-05 2-AMINOCARBONYL-9H-PURINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM TNSN01083A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0014048A GB0014048D0 (en) 2000-06-06 2000-06-06 Purine derivatives
GB0018246A GB0018246D0 (en) 2000-06-06 2000-07-25 Purine derivatives
GB0024920A GB0024920D0 (en) 2000-06-06 2000-10-11 Purine derivatives

Publications (1)

Publication Number Publication Date
TNSN01083A1 true TNSN01083A1 (en) 2005-11-10

Family

ID=9893285

Family Applications (1)

Application Number Title Priority Date Filing Date
TNTNSN01083A TNSN01083A1 (en) 2000-06-06 2001-06-05 2-AMINOCARBONYL-9H-PURINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM

Country Status (15)

Country Link
CN (1) CN100374454C (en)
AP (1) AP2001002179A0 (en)
CR (1) CR6829A (en)
DO (1) DOP2001000182A (en)
EC (1) ECSP024370A (en)
GB (2) GB0014048D0 (en)
GE (1) GEP20053513B (en)
GT (1) GT200100105A (en)
IL (1) IL152783A (en)
MY (1) MY128457A (en)
PE (1) PE20020065A1 (en)
SV (1) SV2002000477A (en)
TN (1) TNSN01083A1 (en)
YU (1) YU82302A (en)
ZA (1) ZA200209875B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105481861B (en) * 2014-09-19 2018-04-17 北京普禄德医药科技有限公司 A kind of platelet aggregation inhibitor and its preparation method and application

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2347512C (en) * 1998-10-16 2005-12-06 Pfizer Inc. Adenine derivatives

Also Published As

Publication number Publication date
DOP2001000182A (en) 2002-08-30
AP2001002179A0 (en) 2002-11-30
ZA200209875B (en) 2003-12-05
GB0018246D0 (en) 2000-09-13
CN100374454C (en) 2008-03-12
MY128457A (en) 2007-02-28
GEP20053513B (en) 2005-05-10
GT200100105A (en) 2002-01-31
PE20020065A1 (en) 2002-02-12
CN1810822A (en) 2006-08-02
YU82302A (en) 2005-11-28
CR6829A (en) 2004-03-11
GB0014048D0 (en) 2000-08-02
ECSP024370A (en) 2003-03-10
SV2002000477A (en) 2002-10-24
IL152783A (en) 2008-11-26

Similar Documents

Publication Publication Date Title
TNSN01096A1 (en) NEW PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM
TNSN01134A1 (en) NEW PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM.
TNSN99106A1 (en) NOVEL ISOTHIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
TNSN02010A1 (en) NOVEL PYRIMIDINE DERIVATIVES OF MMP INHIBITORS, AND COMPOSITIONS CONTAINING THEM
TNSN02008A1 (en) NEW MMP INHIBITOR ISOPHTHALIC ACID DERIVATIVES AND COMPOSITIONS CONTAINING THEM
TNSN02009A1 (en) NEW CONDENSED BICYCLIC PYRIMIDINONES, INHIBITORS OF MMP, AND COMPOSITIONS CONTAINING THEM.
TNSN02014A1 (en) NOVEL PPAR AGONIST COMPOUNDS AND COMPOSITIONS CONTAINING SAME
TNSN02011A1 (en) NOVEL BICYCLIC PYRIMIDINE DERIVATIVES, MMP INHIBITORS, AND COMPOSITIONS CONTAINING THEM
TNSN01048A1 (en) MALONAMIC ACIDS AND DERIVATIVES THEREOF, AND COMPOSITIONS CONTAINING THEM
TNSN01114A1 (en) NEW IMIDAZOLE DERIVATIVES AND COMPOSITIONS CONTAINING THEM
TNSN00202A1 (en) NOVEL N - [(PURINE - 2- YL) METHYL] -SULFONAMIDE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM
TNSN01095A1 (en) NOVEL PYRROLO [2,3-d] PYRIMIDINE DERIVATIVES AND COMPOSITIONS CONTAINING THEM
TNSN01028A1 (en) NOVEL PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM
TNSN97198A1 (en) 6-PHENYLPYRIDYL-2-AMINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
TNSN01102A1 (en) NOVEL PYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM.
TNSN00203A1 (en) NEW PURINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM
TNSN99155A1 (en) 1-ARYL-3-ARYLMETHYL-1,8-NAPHTYRIDINE-4 (1H) -ONES NOVELS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
TNSN01145A1 (en) IMIDAZOLE DERIVATIVES WITH CONDENSED ARYLATED OR HETEROARYL CORE, AND COMPOSITIONS CONTAINING THEM.
TNSN99095A1 (en) 4 - NEW PHENYLPIPERIDINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
TNSN98017A1 (en) SULFONYLUREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
TNSN98084A1 (en) DERIVATIVES OF SUBSTITUTED MACROLIDES IN POSITION C-4
TNSN01019A1 (en) PYRIMIDINECARBOXAMIDES USEFUL AS INHIBITORS OF ISOEZYMES PDE4, AND COMPOSITIONS CONTAINING THEM
TNSN99006A1 (en) 4- (2-CETO-1-BENZIMIDAZOLINYL) NOVEL PIPERIDINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
TNSN00191A1 (en) NOVEL COMPOUNDS, COMPOSITIONS CONTAINING THEM AND THEIR USE IN THE TREATMENT OF ISCHEMIA
MA27883A1 (en) PYRIDO [2,1-A] ISOQUINOLINE DERIVATIVES AS INHIBITORS OF DPP-IV