SK283859B6 - 1-[2'-(Substituovaný)vinyl]-5H-2,3-benzodiazepínové deriváty, spôsob ich prípravy a medziprodukty na ich prípravu, liečivá ich obsahujúce a ich použitie - Google Patents
1-[2'-(Substituovaný)vinyl]-5H-2,3-benzodiazepínové deriváty, spôsob ich prípravy a medziprodukty na ich prípravu, liečivá ich obsahujúce a ich použitie Download PDFInfo
- Publication number
- SK283859B6 SK283859B6 SK167-96A SK16796A SK283859B6 SK 283859 B6 SK283859 B6 SK 283859B6 SK 16796 A SK16796 A SK 16796A SK 283859 B6 SK283859 B6 SK 283859B6
- Authority
- SK
- Slovakia
- Prior art keywords
- substituted
- vinyl
- group
- benzodiazepine derivatives
- benzodiazepine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/02—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Anesthesiology (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU9500385A HU224438B1 (hu) | 1995-02-09 | 1995-02-09 | Benzodiazepin-származékok, eljárás előállításukra, alkalmazásuk és ezeket tartalmazó gyógyászati készítmények |
HU9503353A HU221508B (en) | 1995-11-24 | 1995-11-24 | 1-vinyl-5h-2,3-benzodiazepine derivatives, pharmaceutical compositions containing them, process for the preparation of the compounds and intermediates |
Publications (2)
Publication Number | Publication Date |
---|---|
SK16796A3 SK16796A3 (en) | 1997-01-08 |
SK283859B6 true SK283859B6 (sk) | 2004-03-02 |
Family
ID=26318220
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SK167-96A SK283859B6 (sk) | 1995-02-09 | 1996-02-07 | 1-[2'-(Substituovaný)vinyl]-5H-2,3-benzodiazepínové deriváty, spôsob ich prípravy a medziprodukty na ich prípravu, liečivá ich obsahujúce a ich použitie |
Country Status (14)
Country | Link |
---|---|
US (1) | US5942506A (fi) |
JP (1) | JP3128750B2 (fi) |
KR (1) | KR100330658B1 (fi) |
BE (1) | BE1009516A3 (fi) |
CA (1) | CA2169115C (fi) |
CZ (1) | CZ291833B6 (fi) |
FI (1) | FI960615A (fi) |
FR (1) | FR2730489B1 (fi) |
GB (1) | GB2297750B (fi) |
HR (1) | HRP960064A2 (fi) |
PL (1) | PL191032B1 (fi) |
RU (1) | RU2161607C2 (fi) |
SK (1) | SK283859B6 (fi) |
YU (1) | YU8296A (fi) |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE761315A (fi) * | 1970-01-12 | 1971-07-07 | S M B Anciens Etablissements J | |
HU179018B (en) * | 1978-10-19 | 1982-08-28 | Gyogyszerkutato Intezet | Process for producing new 5h-2,3-benzodiazepine derivatives |
HU186760B (en) * | 1981-03-12 | 1985-09-30 | Gyogyszerkutato Intezet | Process for preparing 3,4-dihydro-5h-2,3-aenzodiazepine derivatives |
HU195788B (en) * | 1986-05-21 | 1988-07-28 | Gyogyszerkutato Intezet | Process for producing 1-/hydroxy-stiryl/-5h-2,3-benzobiazepines and pharmaceutical compositions containing them |
-
1996
- 1996-02-07 SK SK167-96A patent/SK283859B6/sk unknown
- 1996-02-08 HR HRP9503353A patent/HRP960064A2/hr not_active Application Discontinuation
- 1996-02-08 CZ CZ1996378A patent/CZ291833B6/cs not_active IP Right Cessation
- 1996-02-08 PL PL312706A patent/PL191032B1/pl not_active IP Right Cessation
- 1996-02-08 FR FR9601552A patent/FR2730489B1/fr not_active Expired - Fee Related
- 1996-02-08 RU RU96102669/04A patent/RU2161607C2/ru not_active IP Right Cessation
- 1996-02-08 CA CA002169115A patent/CA2169115C/en not_active Expired - Fee Related
- 1996-02-08 BE BE9600111A patent/BE1009516A3/fr not_active IP Right Cessation
- 1996-02-09 KR KR1019960003128A patent/KR100330658B1/ko not_active IP Right Cessation
- 1996-02-09 JP JP08024269A patent/JP3128750B2/ja not_active Expired - Fee Related
- 1996-02-09 FI FI960615A patent/FI960615A/fi unknown
- 1996-02-09 US US08/599,236 patent/US5942506A/en not_active Expired - Fee Related
- 1996-02-09 GB GB9602703A patent/GB2297750B/en not_active Expired - Fee Related
- 1996-02-09 YU YU8296A patent/YU8296A/sh unknown
Also Published As
Publication number | Publication date |
---|---|
GB2297750A (en) | 1996-08-14 |
FR2730489A1 (fr) | 1996-08-14 |
RU2161607C2 (ru) | 2001-01-10 |
CA2169115A1 (en) | 1996-08-10 |
YU8296A (sh) | 1999-03-04 |
CZ37896A3 (en) | 1996-08-14 |
BE1009516A3 (fr) | 1997-04-01 |
CA2169115C (en) | 2000-07-25 |
SK16796A3 (en) | 1997-01-08 |
GB9602703D0 (en) | 1996-04-10 |
FR2730489B1 (fr) | 1997-04-11 |
HRP960064A2 (en) | 1997-10-31 |
KR960031443A (ko) | 1996-09-17 |
PL312706A1 (en) | 1996-08-19 |
US5942506A (en) | 1999-08-24 |
CZ291833B6 (cs) | 2003-06-18 |
FI960615A0 (fi) | 1996-02-09 |
JP3128750B2 (ja) | 2001-01-29 |
KR100330658B1 (ko) | 2002-11-07 |
GB2297750B (en) | 1998-07-01 |
PL191032B1 (pl) | 2006-03-31 |
FI960615A (fi) | 1996-08-10 |
JPH08295676A (ja) | 1996-11-12 |
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