SI1670773T1 - Postopki za pripravo benzoksazol sulfonamidnih spojin in njihovih intermediatov - Google Patents
Postopki za pripravo benzoksazol sulfonamidnih spojin in njihovih intermediatovInfo
- Publication number
- SI1670773T1 SI1670773T1 SI200430265T SI200430265T SI1670773T1 SI 1670773 T1 SI1670773 T1 SI 1670773T1 SI 200430265 T SI200430265 T SI 200430265T SI 200430265 T SI200430265 T SI 200430265T SI 1670773 T1 SI1670773 T1 SI 1670773T1
- Authority
- SI
- Slovenia
- Prior art keywords
- intermediates
- preparation
- methods
- sulfonamide compounds
- benzoxazole sulfonamide
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP03103630 | 2003-09-30 | ||
| US50799603P | 2003-10-02 | 2003-10-02 | |
| EP04766869A EP1670773B1 (en) | 2003-09-30 | 2004-09-30 | Methods for the preparation of benzoxazole sulfonamide compounds and intermediates thereof |
| PCT/EP2004/052382 WO2005030739A1 (en) | 2003-09-30 | 2004-09-30 | Methods for the preparation of benzoxazole sulfonamide compounds and intermediates thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SI1670773T1 true SI1670773T1 (sl) | 2007-06-30 |
Family
ID=34395298
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SI200430265T SI1670773T1 (sl) | 2003-09-30 | 2004-09-30 | Postopki za pripravo benzoksazol sulfonamidnih spojin in njihovih intermediatov |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US20070123574A1 (sl) |
| EP (1) | EP1670773B1 (sl) |
| JP (1) | JP4919802B2 (sl) |
| KR (1) | KR101090102B1 (sl) |
| CN (1) | CN1860107B (sl) |
| AP (1) | AP1985A (sl) |
| AT (1) | ATE353323T1 (sl) |
| AU (1) | AU2004276017B2 (sl) |
| BR (1) | BRPI0414916A (sl) |
| CA (1) | CA2537877C (sl) |
| DE (1) | DE602004004674T2 (sl) |
| DK (1) | DK1670773T3 (sl) |
| EA (1) | EA011891B1 (sl) |
| ES (1) | ES2281828T3 (sl) |
| IL (1) | IL173891A0 (sl) |
| IN (1) | IN2012DN02301A (sl) |
| MX (1) | MXPA06003575A (sl) |
| NO (1) | NO20061951L (sl) |
| NZ (1) | NZ546279A (sl) |
| PL (1) | PL1670773T3 (sl) |
| PT (1) | PT1670773E (sl) |
| SI (1) | SI1670773T1 (sl) |
| WO (1) | WO2005030739A1 (sl) |
| ZA (1) | ZA200602603B (sl) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR053845A1 (es) * | 2005-04-15 | 2007-05-23 | Tibotec Pharm Ltd | 5-tiazolilmetil[(1s,2r)-3-[[(2-amino-6-benzoxazolil)sulfonil)](2-metilpropil)amino]-2-hidroxi-1-(fenilmetil)propil]carbamato como mejorador de farmacos metabolizados por el citocromo p450 |
| US8575186B2 (en) | 2009-10-05 | 2013-11-05 | Albany Molecular Research, Inc. | Epiminocycloalkyl[b] indole derivatives as serotonin sub-type 6 (5-HT6) modulators and uses thereof |
| AU2012207335A1 (en) | 2011-01-19 | 2013-07-25 | Albany Molecular Research, Inc. | Benzofuro[3,2-c] pyridines and related analogs as serotonin sub-type 6 (5-HT6) modulators for the treatment of obesity, metabolic syndrome, cognition and schizophrenia |
| WO2014194519A1 (en) | 2013-06-07 | 2014-12-11 | Merck Sharp & Dohme Corp. | Imidazole derivatives and methods of use thereof for improving pharmacokinetics of drug |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5968942A (en) * | 1992-08-25 | 1999-10-19 | G. D. Searle & Co. | α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors |
| HUP9800518A3 (en) * | 1995-03-10 | 1998-09-28 | G D Searle & Co Chicago | Heterocyclecarbonyl amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors |
| US5753660A (en) * | 1995-11-15 | 1998-05-19 | G. D. Searle & Co. | Substituted sulfonylalkanoylamino hydroxyethylamino sulfonamide retroviral protease inhibitors |
| JP4008708B2 (ja) * | 2000-04-07 | 2007-11-14 | サムスン エレクトロニクス カンパニー リミテッド | マトリックスメタロプロテイナーゼの阻害剤としてのスルホンアミド誘導体 |
| US6455738B1 (en) * | 2000-07-13 | 2002-09-24 | Rhodia Chimie | Process for the sulfonation of an aromatic compound |
| ES2275866T3 (es) * | 2001-02-14 | 2007-06-16 | Tibotec Pharmaceuticals Ltd. | 2-(aminosustituido)-benzotiazol-sulfonamidas de amplio esprecto inhibidoras de la proteasa de vih. |
| CN100549007C (zh) * | 2001-05-11 | 2009-10-14 | 泰博特克药品有限公司 | 广谱2-氨基-苯并唑磺酰胺hiv蛋白酶抑制剂 |
| AR037797A1 (es) * | 2001-12-12 | 2004-12-01 | Tibotec Pharm Ltd | Combinacion de inhibidores de proteasa dependientes del citocromo p450 |
| MY142238A (en) * | 2002-03-12 | 2010-11-15 | Tibotec Pharm Ltd | Broadspectrum substituted benzimidazole sulfonamide hiv protease inhibitors |
-
2004
- 2004-09-30 SI SI200430265T patent/SI1670773T1/sl unknown
- 2004-09-30 IN IN2301DEN2012 patent/IN2012DN02301A/en unknown
- 2004-09-30 MX MXPA06003575A patent/MXPA06003575A/es active IP Right Grant
- 2004-09-30 NZ NZ546279A patent/NZ546279A/en not_active IP Right Cessation
- 2004-09-30 CA CA2537877A patent/CA2537877C/en not_active Expired - Fee Related
- 2004-09-30 US US10/574,157 patent/US20070123574A1/en not_active Abandoned
- 2004-09-30 PL PL04766869T patent/PL1670773T3/pl unknown
- 2004-09-30 BR BRPI0414916-5A patent/BRPI0414916A/pt not_active IP Right Cessation
- 2004-09-30 AU AU2004276017A patent/AU2004276017B2/en not_active Ceased
- 2004-09-30 EA EA200600699A patent/EA011891B1/ru not_active IP Right Cessation
- 2004-09-30 AP AP2006003603A patent/AP1985A/xx active
- 2004-09-30 ES ES04766869T patent/ES2281828T3/es active Active
- 2004-09-30 WO PCT/EP2004/052382 patent/WO2005030739A1/en active IP Right Grant
- 2004-09-30 KR KR1020067005992A patent/KR101090102B1/ko not_active IP Right Cessation
- 2004-09-30 AT AT04766869T patent/ATE353323T1/de active
- 2004-09-30 CN CN2004800280971A patent/CN1860107B/zh not_active Expired - Fee Related
- 2004-09-30 EP EP04766869A patent/EP1670773B1/en active Active
- 2004-09-30 DE DE602004004674T patent/DE602004004674T2/de active Active
- 2004-09-30 JP JP2006530265A patent/JP4919802B2/ja not_active Expired - Fee Related
- 2004-09-30 DK DK04766869T patent/DK1670773T3/da active
- 2004-09-30 PT PT04766869T patent/PT1670773E/pt unknown
-
2006
- 2006-02-22 IL IL173891A patent/IL173891A0/en not_active IP Right Cessation
- 2006-03-29 ZA ZA200602603A patent/ZA200602603B/xx unknown
- 2006-05-02 NO NO20061951A patent/NO20061951L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| PT1670773E (pt) | 2007-05-31 |
| KR101090102B1 (ko) | 2011-12-07 |
| DE602004004674D1 (de) | 2007-03-22 |
| AU2004276017B2 (en) | 2010-08-19 |
| US20070123574A1 (en) | 2007-05-31 |
| AP2006003603A0 (en) | 2006-04-30 |
| CN1860107A (zh) | 2006-11-08 |
| DE602004004674T2 (de) | 2007-11-22 |
| IN2012DN02301A (sl) | 2015-08-14 |
| AP1985A (en) | 2009-03-30 |
| MXPA06003575A (es) | 2006-06-05 |
| KR20060092224A (ko) | 2006-08-22 |
| PL1670773T3 (pl) | 2007-06-29 |
| DK1670773T3 (da) | 2007-05-29 |
| CA2537877A1 (en) | 2005-04-07 |
| CA2537877C (en) | 2015-03-17 |
| EA011891B1 (ru) | 2009-06-30 |
| NZ546279A (en) | 2008-09-26 |
| EP1670773B1 (en) | 2007-02-07 |
| WO2005030739A1 (en) | 2005-04-07 |
| AU2004276017A1 (en) | 2005-04-07 |
| IL173891A0 (en) | 2006-07-05 |
| JP4919802B2 (ja) | 2012-04-18 |
| NO20061951L (no) | 2006-05-02 |
| EP1670773A1 (en) | 2006-06-21 |
| CN1860107B (zh) | 2013-08-21 |
| EA200600699A1 (ru) | 2006-08-25 |
| JP2007507468A (ja) | 2007-03-29 |
| ES2281828T3 (es) | 2007-10-01 |
| ATE353323T1 (de) | 2007-02-15 |
| ZA200602603B (en) | 2008-05-28 |
| BRPI0414916A (pt) | 2006-11-07 |
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