SG155885A1 - Furamate of 4-((4-((4-(2-cyanoethenyl)-2,6-dimethylphenyl)amino)-2- pyrimidinyl)amino)benzonitrile - Google Patents

Furamate of 4-((4-((4-(2-cyanoethenyl)-2,6-dimethylphenyl)amino)-2- pyrimidinyl)amino)benzonitrile

Info

Publication number
SG155885A1
SG155885A1 SG200905799-3A SG2009057993A SG155885A1 SG 155885 A1 SG155885 A1 SG 155885A1 SG 2009057993 A SG2009057993 A SG 2009057993A SG 155885 A1 SG155885 A1 SG 155885A1
Authority
SG
Singapore
Prior art keywords
amino
cyanoethenyl
benzonitrile
dimethylphenyl
pyrimidinyl
Prior art date
Application number
SG200905799-3A
Inventor
Paul Theodoor Agnes Stevens
Jozef Peeters
Roger Petrus Gerebern Vandecruys
Alfred Elisabeth Stappers
Alex Herman Copmans
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38137294&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG155885(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from MYPI20043578A external-priority patent/MY169670A/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of SG155885A1 publication Critical patent/SG155885A1/en

Links

Abstract

FURAMATE, OF 4-((4-((4-(2-CYANOETHENYL)-2,6 DIMETHYLPHENYL)AMINO)-2-PYRIMIDINYL) AMINO)BENZONITRILE The present invention relates to the fumarate salt of 4-[[4-[[4-(2- cyanoethenyl)-2,6-dimethylphenyl]amino] -2-pyrimidinyl]amino] benzonitrile, pharmaceutical compositions comprising as active ingredient said salt and to processes for their preparation.
SG200905799-3A 2004-09-02 2005-09-02 Furamate of 4-((4-((4-(2-cyanoethenyl)-2,6-dimethylphenyl)amino)-2- pyrimidinyl)amino)benzonitrile SG155885A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
MYPI20043578A MY169670A (en) 2003-09-03 2004-09-02 Combinations of a pyrimidine containing nnrti with rt inhibitors
PCT/EP2004/052028 WO2005021001A1 (en) 2003-09-03 2004-09-03 Combinations of a pyrimidine containing nnrti with rt inhibitors

Publications (1)

Publication Number Publication Date
SG155885A1 true SG155885A1 (en) 2009-10-29

Family

ID=38137294

Family Applications (1)

Application Number Title Priority Date Filing Date
SG200905799-3A SG155885A1 (en) 2004-09-02 2005-09-02 Furamate of 4-((4-((4-(2-cyanoethenyl)-2,6-dimethylphenyl)amino)-2- pyrimidinyl)amino)benzonitrile

Country Status (6)

Country Link
CN (2) CN101056673A (en)
AP (1) AP2296A (en)
CR (1) CR9031A (en)
SG (1) SG155885A1 (en)
UA (2) UA92467C2 (en)
ZA (1) ZA200701826B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103420920B (en) * 2012-05-14 2016-04-27 上海迪赛诺药业有限公司 Rilpivrine hydrochloride alcoholate polymorphic form and preparation method thereof
WO2013170421A1 (en) * 2012-05-14 2013-11-21 上海迪赛诺药业有限公司 Rilpivirine hydrochloride alcoholate polymorph and preparation method thereof
JP7197474B2 (en) * 2016-10-24 2022-12-27 ヤンセン・サイエンシズ・アイルランド・アンリミテッド・カンパニー dispersible composition

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY169670A (en) * 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
JO3429B1 (en) * 2001-08-13 2019-10-20 Janssen Pharmaceutica Nv Hiv inhibiting pyrimidines derivatives
CN100554245C (en) * 2002-08-09 2009-10-28 詹森药业有限公司 Preparation 4-[[4-[[4-(2-cyano group vinyl)-2,6-3,5-dimethylphenyl] amino]-the 2-pyrimidyl] amino] method of benzonitrile

Also Published As

Publication number Publication date
UA92467C2 (en) 2010-11-10
AP2296A (en) 2011-10-31
CR9031A (en) 2009-01-16
CN101068597A (en) 2007-11-07
ZA200701826B (en) 2008-07-30
UA92469C2 (en) 2010-11-10
CN101068597B (en) 2012-04-18
AP2007003934A0 (en) 2007-04-30
CN101056673A (en) 2007-10-17

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