SG11202013029UA - Pyridopyrimidinone derivatives for use as axl inhibitors - Google Patents

Pyridopyrimidinone derivatives for use as axl inhibitors

Info

Publication number
SG11202013029UA
SG11202013029UA SG11202013029UA SG11202013029UA SG11202013029UA SG 11202013029U A SG11202013029U A SG 11202013029UA SG 11202013029U A SG11202013029U A SG 11202013029UA SG 11202013029U A SG11202013029U A SG 11202013029UA SG 11202013029U A SG11202013029U A SG 11202013029UA
Authority
SG
Singapore
Prior art keywords
axl inhibitors
pyridopyrimidinone derivatives
pyridopyrimidinone
derivatives
axl
Prior art date
Application number
SG11202013029UA
Inventor
Jung-Ho Kim
Jang-Sik Choi
Hee Kyu Lee
Dong-Sik Jung
Sung-Ho Park
Yung-Geun Choi
Original Assignee
Oscotec Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Oscotec Inc filed Critical Oscotec Inc
Publication of SG11202013029UA publication Critical patent/SG11202013029UA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K39/395Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum
    • A61K39/39533Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals
    • A61K39/3955Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals against proteinaceous materials, e.g. enzymes, hormones, lymphokines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/505Medicinal preparations containing antigens or antibodies comprising antibodies
SG11202013029UA 2018-06-27 2019-06-26 Pyridopyrimidinone derivatives for use as axl inhibitors SG11202013029UA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862690620P 2018-06-27 2018-06-27
PCT/KR2019/007733 WO2020004938A1 (en) 2018-06-27 2019-06-26 Pyridopyrimidinone derivatives for use as axl inhibitors

Publications (1)

Publication Number Publication Date
SG11202013029UA true SG11202013029UA (en) 2021-01-28

Family

ID=68987456

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11202013029UA SG11202013029UA (en) 2018-06-27 2019-06-26 Pyridopyrimidinone derivatives for use as axl inhibitors

Country Status (15)

Country Link
US (1) US20210275532A1 (en)
EP (1) EP3814350A4 (en)
JP (1) JP7200453B2 (en)
KR (1) KR20210014212A (en)
CN (1) CN112351985B (en)
AU (1) AU2019292207B2 (en)
BR (1) BR112020026641A2 (en)
CA (1) CA3103160C (en)
CL (1) CL2020003340A1 (en)
EA (1) EA202190125A1 (en)
IL (1) IL279593A (en)
MX (1) MX2020013805A (en)
SG (1) SG11202013029UA (en)
WO (1) WO2020004938A1 (en)
ZA (1) ZA202100140B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK3814348T3 (en) 2018-06-27 2023-10-30 Bristol Myers Squibb Co SUBSTITUTED NAPHTHYRIDINONE COMPOUNDS USEFUL AS T CELL ACTIVATORS

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL112249A (en) * 1994-01-25 2001-11-25 Warner Lambert Co Pharmaceutical compositions containing di and tricyclic pyrimidine derivatives for inhibiting tyrosine kinases of the epidermal growth factor receptor family and some new such compounds
RS49779B (en) * 1998-01-12 2008-06-05 Glaxo Group Limited, Byciclic heteroaromatic compounds as protein tyrosine kinase inhibitors
US8404677B2 (en) 2009-10-29 2013-03-26 Genosco Kinase inhibitors
AU2013235344B2 (en) * 2012-03-22 2017-03-16 Oscotec Inc. Substituted pyridopyrimidine compounds and their use as FLT3 inhibitors
US9533989B2 (en) * 2012-09-18 2017-01-03 Ziarco Pharma Ltd. Substituted pyrimidine-5-carboxamides as spleen tyrosine kinase inhibitors
GB201509338D0 (en) * 2015-05-29 2015-07-15 Bergenbio As Combination therapy
WO2017059280A1 (en) * 2015-10-02 2017-04-06 The University Of North Carolina At Chapel Hill Novel pan-tam inhibitors and mer/axl dual inhibitors
EP3469001A4 (en) 2016-06-09 2020-05-06 Seattle Genetics, Inc. Combinations of pbd-based antibody drug conjugates with flt3 inhibitors

Also Published As

Publication number Publication date
CN112351985A (en) 2021-02-09
WO2020004938A1 (en) 2020-01-02
EP3814350A4 (en) 2022-05-04
IL279593A (en) 2021-03-01
EP3814350A1 (en) 2021-05-05
JP2021528383A (en) 2021-10-21
JP7200453B2 (en) 2023-01-10
MX2020013805A (en) 2021-03-09
CA3103160A1 (en) 2020-01-02
BR112020026641A2 (en) 2021-03-30
US20210275532A1 (en) 2021-09-09
ZA202100140B (en) 2022-07-27
CA3103160C (en) 2023-03-07
AU2019292207B2 (en) 2022-06-30
CN112351985B (en) 2023-12-15
CL2020003340A1 (en) 2021-04-23
AU2019292207A1 (en) 2021-02-18
EA202190125A1 (en) 2021-05-24
KR20210014212A (en) 2021-02-08

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