SG11202001868RA - Solid forms of 2-(5-(4-(2-morpholinoethoxy)phenyl)pyridin-2-yl)-n-benzylacetamide - Google Patents
Solid forms of 2-(5-(4-(2-morpholinoethoxy)phenyl)pyridin-2-yl)-n-benzylacetamideInfo
- Publication number
- SG11202001868RA SG11202001868RA SG11202001868RA SG11202001868RA SG11202001868RA SG 11202001868R A SG11202001868R A SG 11202001868RA SG 11202001868R A SG11202001868R A SG 11202001868RA SG 11202001868R A SG11202001868R A SG 11202001868RA SG 11202001868R A SG11202001868R A SG 11202001868RA
- Authority
- SG
- Singapore
- Prior art keywords
- benzylacetamide
- morpholinoethoxy
- pyridin
- phenyl
- solid forms
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/56—Amides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Physics & Mathematics (AREA)
- Condensed Matter Physics & Semiconductors (AREA)
- Crystallography & Structural Chemistry (AREA)
- General Physics & Mathematics (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762555390P | 2017-09-07 | 2017-09-07 | |
| PCT/US2018/049829 WO2019051147A1 (en) | 2017-09-07 | 2018-09-07 | Solid forms of 2-(5-(4-(2-morpholinoethoxy)phenyl)pyridin-2-yl)-n-benzylacetamide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG11202001868RA true SG11202001868RA (en) | 2020-03-30 |
Family
ID=65517772
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG11202001868RA SG11202001868RA (en) | 2017-09-07 | 2018-09-07 | Solid forms of 2-(5-(4-(2-morpholinoethoxy)phenyl)pyridin-2-yl)-n-benzylacetamide |
Country Status (12)
| Country | Link |
|---|---|
| US (3) | US10669236B2 (en) |
| EP (1) | EP3679016A4 (en) |
| JP (2) | JP2020533412A (en) |
| CN (1) | CN111278808B (en) |
| AU (2) | AU2018330163B2 (en) |
| BR (1) | BR112020004419A2 (en) |
| CA (1) | CA3074831A1 (en) |
| IL (1) | IL272992A (en) |
| MX (2) | MX2020002622A (en) |
| SG (1) | SG11202001868RA (en) |
| TW (1) | TWI815820B (en) |
| WO (1) | WO2019051147A1 (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7968574B2 (en) * | 2004-12-28 | 2011-06-28 | Kinex Pharmaceuticals, Llc | Biaryl compositions and methods for modulating a kinase cascade |
| EP4186890A1 (en) | 2021-11-29 | 2023-05-31 | Moehs Ibérica, S.L. | Preparation of n-benzyl-2-(5-bromo-pyridin-2-yl)-acetamide for the synthesis of tirbanibulin |
| CN115010655A (en) * | 2022-07-21 | 2022-09-06 | 重庆迈德凯医药有限公司 | Purification method of tinib bulin |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4522811A (en) | 1982-07-08 | 1985-06-11 | Syntex (U.S.A.) Inc. | Serial injection of muramyldipeptides and liposomes enhances the anti-infective activity of muramyldipeptides |
| US7141593B1 (en) * | 1999-06-04 | 2006-11-28 | Abbott Laboratories | Pharmaceutical formulations |
| EA007618B1 (en) * | 2001-05-22 | 2006-12-29 | Пфайзер Продактс Инк. | Crystalline sesquihydrate azithromycin, pharmaceutical composition and method for treatment based thereon |
| US6821502B2 (en) * | 2002-06-12 | 2004-11-23 | Chevron U.S.A. Inc. | Method of making aluminum-containing zeolite with IFR structure |
| US7351833B2 (en) * | 2004-07-23 | 2008-04-01 | Abbott Laboratories | (1S,5S)-3-(5,6-dichloropyridin-3-yl)-3,6-diazabicyclo[3.2.0]heptane benzenesulfonate |
| DK1836169T5 (en) | 2004-12-28 | 2023-10-09 | Atnx Spv Llc | COMPOSITIONS AND METHODS FOR TREATING CELL PROLIFERATION DISORDERS |
| MY152185A (en) * | 2005-06-10 | 2014-08-29 | Novartis Ag | Modified release 1-[(3-hydroxy-adamant-1-ylamino)-acetyl]-pyrrolidine-2(s)-carbonitrile formulation |
| TW200804409A (en) * | 2005-09-13 | 2008-01-16 | Sicor Inc | Processes for the synthesis of rocuronium bromide |
| DK2041071T3 (en) | 2006-06-29 | 2014-09-01 | Kinex Pharmaceuticals Llc | BIARLYL COMPOSITIONS AND PROCEDURES FOR MODULATING A CHINA CASE |
| KR20090064400A (en) * | 2006-09-28 | 2009-06-18 | 머크 앤드 캄파니 인코포레이티드 | Pharmaceutical compositions of hdac inhibitors and chelatable metal compounds, and metal-hdac inhibitor chelate complexes |
| US7837978B2 (en) * | 2006-10-13 | 2010-11-23 | Chevron U.S.A. Inc. | Process for preparing aluminum-containing molecular sieve SSZ-26 |
| PE20081506A1 (en) * | 2006-12-12 | 2008-12-09 | Infinity Discovery Inc | ANSAMYCIN FORMULATIONS |
| US7935697B2 (en) * | 2006-12-28 | 2011-05-03 | Kinex Pharmaceuticals, Llc | Compositions for modulating a kinase cascade and methods of use thereof |
| US7939529B2 (en) | 2007-05-17 | 2011-05-10 | Kinex Pharmaceuticals, Llc | Process for the preparation of compositions for modulating a kinase cascade and methods of use thereof |
| TWI457336B (en) | 2006-12-28 | 2014-10-21 | Kinex Pharmaceuticals Llc | Composition and methods for modulating a kinase cascade |
| AU2008253803A1 (en) * | 2007-05-22 | 2008-11-27 | Ultimorphix Technolgies B.V. | Tenofovir disoproxil hemi-fumaric acid Co-crystal |
| WO2015069217A1 (en) | 2013-11-05 | 2015-05-14 | Baylor College Of Medicine | Src kinase inhibition as treatment for lympangioleiomyomatosis and tuberous sclerosis |
| CN106810490A (en) * | 2017-02-06 | 2017-06-09 | 重庆泰润制药有限公司 | A kind of crystal formation of biaryl compound and its preparation method and application |
-
2018
- 2018-09-07 TW TW107131540A patent/TWI815820B/en active
- 2018-09-07 JP JP2020536496A patent/JP2020533412A/en active Pending
- 2018-09-07 CA CA3074831A patent/CA3074831A1/en active Pending
- 2018-09-07 AU AU2018330163A patent/AU2018330163B2/en active Active
- 2018-09-07 WO PCT/US2018/049829 patent/WO2019051147A1/en unknown
- 2018-09-07 BR BR112020004419-9A patent/BR112020004419A2/en unknown
- 2018-09-07 EP EP18854688.1A patent/EP3679016A4/en active Pending
- 2018-09-07 US US16/124,281 patent/US10669236B2/en active Active
- 2018-09-07 CN CN201880069894.6A patent/CN111278808B/en active Active
- 2018-09-07 MX MX2020002622A patent/MX2020002622A/en unknown
- 2018-09-07 SG SG11202001868RA patent/SG11202001868RA/en unknown
-
2020
- 2020-03-01 IL IL272992A patent/IL272992A/en unknown
- 2020-03-06 MX MX2023001805A patent/MX2023001805A/en unknown
- 2020-04-27 US US16/858,854 patent/US11230527B2/en active Active
-
2021
- 2021-12-09 US US17/546,133 patent/US20220098152A1/en active Pending
-
2023
- 2023-02-21 AU AU2023201010A patent/AU2023201010A1/en active Pending
- 2023-06-30 JP JP2023107781A patent/JP2023157909A/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| CN111278808A (en) | 2020-06-12 |
| AU2018330163B2 (en) | 2023-02-02 |
| RU2020112539A3 (en) | 2022-04-19 |
| BR112020004419A2 (en) | 2020-09-08 |
| MX2020002622A (en) | 2020-10-01 |
| EP3679016A4 (en) | 2021-09-29 |
| TWI815820B (en) | 2023-09-21 |
| US20200255380A1 (en) | 2020-08-13 |
| MX2023001805A (en) | 2023-03-13 |
| US20220098152A1 (en) | 2022-03-31 |
| KR20200081359A (en) | 2020-07-07 |
| EP3679016A1 (en) | 2020-07-15 |
| US20190071402A1 (en) | 2019-03-07 |
| IL272992A (en) | 2020-04-30 |
| TW201920160A (en) | 2019-06-01 |
| AU2023201010A1 (en) | 2023-03-23 |
| JP2023157909A (en) | 2023-10-26 |
| AU2018330163A1 (en) | 2020-03-26 |
| CA3074831A1 (en) | 2019-03-14 |
| CN111278808B (en) | 2024-04-26 |
| WO2019051147A1 (en) | 2019-03-14 |
| US11230527B2 (en) | 2022-01-25 |
| RU2020112539A (en) | 2021-10-08 |
| JP2020533412A (en) | 2020-11-19 |
| US10669236B2 (en) | 2020-06-02 |
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