SG11201704576SA - Method for producing crystals of diazabicyclooctane derivative and stable lyophilized preparation - Google Patents

Method for producing crystals of diazabicyclooctane derivative and stable lyophilized preparation

Info

Publication number
SG11201704576SA
SG11201704576SA SG11201704576SA SG11201704576SA SG11201704576SA SG 11201704576S A SG11201704576S A SG 11201704576SA SG 11201704576S A SG11201704576S A SG 11201704576SA SG 11201704576S A SG11201704576S A SG 11201704576SA SG 11201704576S A SG11201704576S A SG 11201704576SA
Authority
SG
Singapore
Prior art keywords
lyophilized preparation
stable lyophilized
producing crystals
diazabicyclooctane derivative
diazabicyclooctane
Prior art date
Application number
SG11201704576SA
Inventor
Takaya Ogawa
Takuya Yokoyama
Shusuke Furuyama
Masato Ichiki
Kenichi Fushihara
Original Assignee
Meiji Seika Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Meiji Seika Pharma Co Ltd filed Critical Meiji Seika Pharma Co Ltd
Publication of SG11201704576SA publication Critical patent/SG11201704576SA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Dermatology (AREA)
  • Inorganic Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
SG11201704576SA 2014-12-05 2015-12-04 Method for producing crystals of diazabicyclooctane derivative and stable lyophilized preparation SG11201704576SA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2014246425 2014-12-05
PCT/JP2015/084094 WO2016088863A1 (en) 2014-12-05 2015-12-04 Method for producing crystals of diazabicyclooctane derivative and stable lyophilized preparation

Publications (1)

Publication Number Publication Date
SG11201704576SA true SG11201704576SA (en) 2017-07-28

Family

ID=56091802

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201704576SA SG11201704576SA (en) 2014-12-05 2015-12-04 Method for producing crystals of diazabicyclooctane derivative and stable lyophilized preparation

Country Status (18)

Country Link
US (2) US10294224B2 (en)
EP (1) EP3228620B1 (en)
JP (1) JP6779787B2 (en)
KR (1) KR102555657B1 (en)
CN (1) CN107001366B (en)
AR (1) AR102915A1 (en)
AU (1) AU2015355970B2 (en)
BR (1) BR112017010445B8 (en)
CA (1) CA2969192C (en)
ES (1) ES2821826T3 (en)
IL (1) IL252691B (en)
MX (1) MX2017007191A (en)
MY (1) MY190283A (en)
RU (1) RU2732129C2 (en)
SG (1) SG11201704576SA (en)
TW (1) TWI691499B (en)
WO (1) WO2016088863A1 (en)
ZA (1) ZA201704063B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013180197A1 (en) 2012-05-30 2013-12-05 Meiji Seikaファルマ株式会社 NOVEL β-LACTAMASE INHIBITOR AND METHOD FOR PRODUCING SAME
ES2901198T3 (en) 2013-10-08 2022-03-21 Meiji Seika Pharma Co Ltd Crystalline forms of diazabicyclooctane derivative and production process thereof
RU2732129C2 (en) 2014-12-05 2020-09-11 Мейдзи Сейка Фарма Ко., Лтд. Method of producing crystals of a diazabicyclooctane derivative and a stable lyophilized preparation
KR20200091395A (en) * 2017-09-27 2020-07-30 페도라 파마슈티칼스 인코포레이티드 Crystal form of diazabicyclooctane derivative and method for preparing same
JP7179058B2 (en) * 2017-09-27 2022-11-28 Meiji Seikaファルマ株式会社 Dosage form of diazabicyclooctane derivative and its production process
JP7200235B2 (en) * 2017-09-27 2023-01-06 Meiji Seikaファルマ株式会社 Dosage form of diazabicyclooctane derivative and production method thereof
JP6375463B1 (en) * 2018-02-28 2018-08-15 日本曹達株式会社 Method for producing bis (fluorosulfonyl) amide alkali metal salt powder
CN110314163A (en) * 2018-03-30 2019-10-11 杭州森泽医药科技有限公司 A kind of latamoxef sodium pharmaceutical composition and application
JP2022094481A (en) * 2020-12-15 2022-06-27 大阪瓦斯株式会社 Method for producing hydroxyalkanoic acid crystal and crystalline polymorph of hydroxyalkanoic acid

Family Cites Families (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6019759B2 (en) 1977-11-24 1985-05-17 イ−ライ・リリ−・アンド・カンパニ− For parenteral administration 11115152139199 2-3-13 Kyobashi, Chuo-ku, Tokyo
GB1589317A (en) * 1977-11-24 1981-05-13 Lilly Co Eli Freeze drying cephalothin sodium
JPS6019759A (en) 1983-07-15 1985-01-31 Nippon Soda Co Ltd Formamidoxime derivative, its preparation and agricultural and horticultural fungicide
JPS60255723A (en) 1984-05-31 1985-12-17 Ono Pharmaceut Co Ltd Freeze-dried crystalline preparation of gabexate mesylate, and its production
JPH07117533B2 (en) 1985-08-28 1995-12-18 株式会社生体科学研究所 Transferrin and its uses
PL157979B1 (en) 1989-02-14 1992-07-31 Spring with two states of fixed equilibrium
US20030220521A1 (en) 1989-07-27 2003-11-27 G.D. Searle & Co. Renal-selective prodrugs for control of renal sympathetic nerve activity in the treatment of hypertension
TW264475B (en) 1991-09-20 1995-12-01 Takeda Pharm Industry Co Ltd
JP2843444B2 (en) * 1994-05-02 1999-01-06 塩野義製薬株式会社 Crystal of pyrrolidylthiocarbapenem derivative, freeze-dried preparation containing the crystal, and method for producing the same
AU700545B2 (en) 1994-05-02 1999-01-07 Shionogi & Co., Ltd. Crystal of pyrrolidylthiocarbapenem derivative, lyophilized preparation containing said crystal, and process for producing the same
DE19531874C1 (en) 1995-08-30 1996-10-02 Daimler Benz Ag Side wall sub assembly
TWI233805B (en) * 1999-07-01 2005-06-11 Fujisawa Pharmaceutical Co Stabilized pharmaceutical composition in lyophilized form as antifungal agent
FR2812635B1 (en) 2000-08-01 2002-10-11 Aventis Pharma Sa NOVEL HETEROCYCLIC COMPOUNDS, PREPARATION AND USE AS MEDICAMENTS IN PARTICULAR AS ANTI-BACTERIALS
FR2825705B1 (en) 2001-06-08 2005-05-20 Aventis Pharma Sa NOVEL HETEROCYCLIC COMPOUNDS, THEIR PREPARATION AND THEIR USE AS MEDICAMENTS, IN PARTICULAR AS ANTI-BACTERIANS
FR2835186B1 (en) 2002-01-28 2006-10-20 Aventis Pharma Sa NOVEL HETEROCYCLIC COMPOUNDS ACTIVE AS BETA-LACTAMASES INHIBITORS
FR2921060B1 (en) 2007-09-14 2012-06-15 Novexel NOVEL PROCESS FOR PREPARING DISUBSIDED PIPERIDINE AND NOVEL INTERMEDIATES
PT2666774E (en) 2008-01-18 2015-04-13 Merck Sharp & Dohme Beta-lactamase inhibitors
FR2930553B1 (en) 2008-04-29 2010-05-21 Novexel AZABICYCLIC COMPOUNDS, THEIR PREPARATION AND THEIR USE AS MEDICAMENTS, IN PARTICULAR BETA-LACTAMASES INHIBITORS
FR2936798B1 (en) 2008-10-03 2012-09-28 Novexel NOVEL HETEROCYCLIC NITROGEN COMPOUNDS, THEIR PREPARATION AND THEIR USE AS ANTIBACTERIAL MEDICINES.
US20120053350A1 (en) 2009-04-30 2012-03-01 Ian Mangion Preparation of alkyl esters of n-protected oxo-azacycloalkylcarboxylic acids
FR2951171A1 (en) 2009-10-09 2011-04-15 Novexel NOVEL SODIUM SALT OF A CRYSTALLIZED ENANTIOMER AZABICYCLIC COMPOUND AND NOVEL POLYMORPHIC AND PSEUDOPOLYMORPHIC FORMS AND THEIR PREPARATION
US8772490B2 (en) 2010-12-22 2014-07-08 Meiji Seika Pharma Co., Ltd. Optically active diazabicyclooctane derivatives and process for preparing the same
ES2622004T3 (en) 2010-12-22 2017-07-05 Meiji Seika Pharma Co., Ltd. Optically active diazabicyclooctane derivative and method for preparing it
US8829191B2 (en) 2011-06-17 2014-09-09 Melanie Simone Ronsheim Processes for preparing heterocyclic compounds including trans-7-oxo-6-(sulphooxy)-1,6-diazabicyclo[3,2,1]octane-2-carboxamide and salts thereof
KR101512738B1 (en) 2011-08-27 2015-04-17 욱크하르트 리미티드 1,6-diazabicyclo[3,2,1]octan-7-one derivatives and their use in the treatment of bacterial infections
WO2013030735A1 (en) 2011-08-30 2013-03-07 Wockhardt Limited 1,6- diazabicyclo [3,2,1] octan- 7 - one derivatives and their use in the treatment of bacterial infections
WO2013038330A1 (en) 2011-09-13 2013-03-21 Wockhardt Limited Nitrogen containing compounds and their use
US8796257B2 (en) 2011-12-02 2014-08-05 Naeja Pharmaceutical Inc. Bicyclic compounds and their use as antibacterial agents and β-lactamase inhibitors
US9505761B2 (en) 2011-12-02 2016-11-29 Fedora Pharmaceuticals Inc. Bicyclic compounds and their use as antibacterial agents and beta-lactamase inhibitors
WO2013180197A1 (en) 2012-05-30 2013-12-05 Meiji Seikaファルマ株式会社 NOVEL β-LACTAMASE INHIBITOR AND METHOD FOR PRODUCING SAME
DK3050883T3 (en) 2013-09-24 2020-05-25 Meiji Seika Pharma Co Ltd PROCEDURE FOR THE PREPARATION OF DIAZABICYCLOOCTAND DERIVATIVES AND INTERMEDIATES
ES2901198T3 (en) 2013-10-08 2022-03-21 Meiji Seika Pharma Co Ltd Crystalline forms of diazabicyclooctane derivative and production process thereof
RU2732129C2 (en) 2014-12-05 2020-09-11 Мейдзи Сейка Фарма Ко., Лтд. Method of producing crystals of a diazabicyclooctane derivative and a stable lyophilized preparation

Also Published As

Publication number Publication date
BR112017010445A2 (en) 2017-12-26
AU2015355970A1 (en) 2017-06-15
RU2732129C2 (en) 2020-09-11
RU2017123112A3 (en) 2019-06-25
EP3228620A1 (en) 2017-10-11
US20190202831A1 (en) 2019-07-04
TWI691499B (en) 2020-04-21
MY190283A (en) 2022-04-12
JPWO2016088863A1 (en) 2017-09-14
ES2821826T3 (en) 2021-04-27
IL252691B (en) 2020-08-31
TW201629062A (en) 2016-08-16
NZ732214A (en) 2021-10-29
CA2969192A1 (en) 2016-06-09
AU2015355970B2 (en) 2020-05-21
CN107001366B (en) 2020-08-28
US10294224B2 (en) 2019-05-21
WO2016088863A1 (en) 2016-06-09
US20170327499A1 (en) 2017-11-16
KR102555657B1 (en) 2023-07-18
AR102915A1 (en) 2017-04-05
KR20170094272A (en) 2017-08-17
EP3228620A4 (en) 2018-05-02
CA2969192C (en) 2023-02-28
RU2017123112A (en) 2019-01-09
MX2017007191A (en) 2017-08-28
BR112017010445B8 (en) 2024-02-27
BR112017010445B1 (en) 2024-01-30
ZA201704063B (en) 2021-10-27
US11117895B2 (en) 2021-09-14
EP3228620B1 (en) 2020-09-02
JP6779787B2 (en) 2020-11-04
CN107001366A (en) 2017-08-01
IL252691A0 (en) 2017-08-31

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