SG11201500973WA - Amino-quinolines as kinase inhibitors - Google Patents
Amino-quinolines as kinase inhibitorsInfo
- Publication number
- SG11201500973WA SG11201500973WA SG11201500973WA SG11201500973WA SG11201500973WA SG 11201500973W A SG11201500973W A SG 11201500973WA SG 11201500973W A SG11201500973W A SG 11201500973WA SG 11201500973W A SG11201500973W A SG 11201500973WA SG 11201500973W A SG11201500973W A SG 11201500973WA
- Authority
- SG
- Singapore
- Prior art keywords
- quinolines
- amino
- kinase inhibitors
- kinase
- inhibitors
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261700536P | 2012-09-13 | 2012-09-13 | |
US201361767378P | 2013-02-21 | 2013-02-21 | |
PCT/US2013/059600 WO2014043437A1 (en) | 2012-09-13 | 2013-09-13 | Amino-quinolines as kinase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
SG11201500973WA true SG11201500973WA (en) | 2015-04-29 |
Family
ID=50278701
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11201500973WA SG11201500973WA (en) | 2012-09-13 | 2013-09-13 | Amino-quinolines as kinase inhibitors |
Country Status (21)
Country | Link |
---|---|
US (1) | US9216965B2 (en) |
EP (1) | EP2895167B1 (en) |
JP (1) | JP6258331B2 (en) |
KR (1) | KR20150053920A (en) |
CN (1) | CN104602692B (en) |
AR (1) | AR092530A1 (en) |
AU (1) | AU2013315387B2 (en) |
BR (1) | BR112015004967A2 (en) |
CA (1) | CA2883155A1 (en) |
CL (1) | CL2015000615A1 (en) |
CR (1) | CR20150133A (en) |
DO (1) | DOP2015000059A (en) |
EA (1) | EA027984B1 (en) |
ES (1) | ES2713172T3 (en) |
IL (1) | IL237158A0 (en) |
MX (1) | MX2015003275A (en) |
PE (1) | PE20150774A1 (en) |
PH (1) | PH12015500345A1 (en) |
SG (1) | SG11201500973WA (en) |
TW (1) | TW201425307A (en) |
WO (1) | WO2014043437A1 (en) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UY33549A (en) * | 2010-08-10 | 2012-01-31 | Glaxo Group Ltd | QUINOLIL AMINAS AS INHIBITING AGENTS OF KINASES |
BR112013022307A2 (en) | 2011-03-04 | 2020-09-24 | Glaxosmithkline Intellectual Property (No. 2) Limited | aminoquinolines as kinase inhibitors |
TWI547494B (en) | 2011-08-18 | 2016-09-01 | 葛蘭素史克智慧財產發展有限公司 | Amino quinazolines as kinase inhibitors |
AR092529A1 (en) | 2012-09-13 | 2015-04-22 | Glaxosmithkline Llc | AMINOQUINAZOLINE COMPOUND, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND USE OF THIS COMPOSITE FOR THE PREPARATION OF A MEDICINAL PRODUCT |
AR092530A1 (en) | 2012-09-13 | 2015-04-22 | Glaxosmithkline Llc | AMINO-QUINOLINE COMPOSITE, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND USE OF THIS COMPOUND FOR THE PREPARATION OF A MEDICINAL PRODUCT |
KR20150118152A (en) | 2013-02-21 | 2015-10-21 | 글락소스미스클라인 인털렉츄얼 프로퍼티 디벨로프먼트 리미티드 | Quinazolines as kinase inhibitors |
GB201506872D0 (en) | 2015-04-22 | 2015-06-03 | Ge Oil & Gas Uk Ltd | Novel compounds |
GB201516243D0 (en) | 2015-09-14 | 2015-10-28 | Glaxosmithkline Ip Dev Ltd | Novel compounds |
CN108473435A (en) | 2015-10-05 | 2018-08-31 | 纽约市哥伦比亚大学理事会 | The treatment of the removing and protein sickness of the activator of autophagy tide and phospholipase D and the protein masses including TAU |
CN107158385B (en) * | 2016-03-14 | 2020-07-14 | 苏州大学 | Application of RIP3 inhibitor in preparation of anti-platelet thrombosis drugs |
CN109311867A (en) | 2016-04-20 | 2019-02-05 | 葛兰素史克知识产权开发有限公司 | Conjugate comprising RIPK2 inhibitor |
WO2020094613A1 (en) | 2018-11-06 | 2020-05-14 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Nod2 inhibitors for the treatment of hereditary periodic fevers |
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US20130023532A1 (en) | 2010-03-26 | 2013-01-24 | Casillas Linda N | Indazolyl-pyrimidines as kinase inhibitors |
US20130023534A1 (en) | 2010-03-26 | 2013-01-24 | Casillas Linda N | Pyrazolyl-pyrimidines as kinase inhibitors |
EP2552208A4 (en) | 2010-03-31 | 2014-07-09 | Glaxo Group Ltd | Imidazolyl-imidazoles as kinase inhibitors |
JP2013526484A (en) | 2010-05-07 | 2013-06-24 | グラクソ グループ リミテッド | Amino-quinolines as kinase inhibitors |
UY33549A (en) * | 2010-08-10 | 2012-01-31 | Glaxo Group Ltd | QUINOLIL AMINAS AS INHIBITING AGENTS OF KINASES |
WO2012027495A1 (en) | 2010-08-27 | 2012-03-01 | University Of The Pacific | Piperazinylpyrimidine analogues as protein kinase inhibitors |
JP5707518B2 (en) | 2011-02-28 | 2015-04-30 | カリトル サイエンシズ, エルエルシー | Substituted quinoline compounds and methods of use |
BR112013022307A2 (en) | 2011-03-04 | 2020-09-24 | Glaxosmithkline Intellectual Property (No. 2) Limited | aminoquinolines as kinase inhibitors |
TWI547494B (en) | 2011-08-18 | 2016-09-01 | 葛蘭素史克智慧財產發展有限公司 | Amino quinazolines as kinase inhibitors |
AR092529A1 (en) | 2012-09-13 | 2015-04-22 | Glaxosmithkline Llc | AMINOQUINAZOLINE COMPOUND, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND USE OF THIS COMPOSITE FOR THE PREPARATION OF A MEDICINAL PRODUCT |
AR092530A1 (en) | 2012-09-13 | 2015-04-22 | Glaxosmithkline Llc | AMINO-QUINOLINE COMPOSITE, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND USE OF THIS COMPOUND FOR THE PREPARATION OF A MEDICINAL PRODUCT |
KR20150118152A (en) | 2013-02-21 | 2015-10-21 | 글락소스미스클라인 인털렉츄얼 프로퍼티 디벨로프먼트 리미티드 | Quinazolines as kinase inhibitors |
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2013
- 2013-09-11 AR ARP130103248A patent/AR092530A1/en unknown
- 2013-09-11 TW TW102132714A patent/TW201425307A/en unknown
- 2013-09-13 EA EA201590552A patent/EA027984B1/en not_active IP Right Cessation
- 2013-09-13 WO PCT/US2013/059600 patent/WO2014043437A1/en active Application Filing
- 2013-09-13 AU AU2013315387A patent/AU2013315387B2/en not_active Ceased
- 2013-09-13 CA CA2883155A patent/CA2883155A1/en not_active Abandoned
- 2013-09-13 US US14/396,559 patent/US9216965B2/en not_active Expired - Fee Related
- 2013-09-13 EP EP13836616.6A patent/EP2895167B1/en active Active
- 2013-09-13 SG SG11201500973WA patent/SG11201500973WA/en unknown
- 2013-09-13 KR KR1020157006177A patent/KR20150053920A/en not_active Application Discontinuation
- 2013-09-13 PE PE2015000276A patent/PE20150774A1/en not_active Application Discontinuation
- 2013-09-13 BR BR112015004967A patent/BR112015004967A2/en active Search and Examination
- 2013-09-13 ES ES13836616T patent/ES2713172T3/en active Active
- 2013-09-13 CN CN201380045559.XA patent/CN104602692B/en not_active Expired - Fee Related
- 2013-09-13 MX MX2015003275A patent/MX2015003275A/en unknown
- 2013-09-13 JP JP2015532064A patent/JP6258331B2/en not_active Expired - Fee Related
-
2015
- 2015-02-09 IL IL237158A patent/IL237158A0/en unknown
- 2015-02-17 PH PH12015500345A patent/PH12015500345A1/en unknown
- 2015-03-12 CL CL2015000615A patent/CL2015000615A1/en unknown
- 2015-03-13 DO DO2015000059A patent/DOP2015000059A/en unknown
- 2015-03-13 CR CR20150133A patent/CR20150133A/en unknown
Also Published As
Publication number | Publication date |
---|---|
TW201425307A (en) | 2014-07-01 |
DOP2015000059A (en) | 2015-05-15 |
AU2013315387A1 (en) | 2015-02-26 |
EP2895167B1 (en) | 2018-12-05 |
EA201590552A1 (en) | 2015-06-30 |
JP6258331B2 (en) | 2018-01-10 |
CN104602692B (en) | 2017-06-23 |
ES2713172T3 (en) | 2019-05-20 |
KR20150053920A (en) | 2015-05-19 |
CN104602692A (en) | 2015-05-06 |
EA027984B1 (en) | 2017-09-29 |
CL2015000615A1 (en) | 2015-08-28 |
US20150094333A1 (en) | 2015-04-02 |
IL237158A0 (en) | 2015-04-30 |
CR20150133A (en) | 2015-05-04 |
JP2015528508A (en) | 2015-09-28 |
PE20150774A1 (en) | 2015-05-28 |
US9216965B2 (en) | 2015-12-22 |
CA2883155A1 (en) | 2014-03-20 |
PH12015500345A1 (en) | 2015-04-20 |
AU2013315387B2 (en) | 2016-09-08 |
EP2895167A1 (en) | 2015-07-22 |
BR112015004967A2 (en) | 2020-04-22 |
WO2014043437A1 (en) | 2014-03-20 |
EP2895167A4 (en) | 2016-03-16 |
AR092530A1 (en) | 2015-04-22 |
MX2015003275A (en) | 2015-07-06 |
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