SG11201500498SA - Urea compounds and their use as enzyme inhibitors - Google Patents
Urea compounds and their use as enzyme inhibitorsInfo
- Publication number
- SG11201500498SA SG11201500498SA SG11201500498SA SG11201500498SA SG11201500498SA SG 11201500498S A SG11201500498S A SG 11201500498SA SG 11201500498S A SG11201500498S A SG 11201500498SA SG 11201500498S A SG11201500498S A SG 11201500498SA SG 11201500498S A SG11201500498S A SG 11201500498SA
- Authority
- SG
- Singapore
- Prior art keywords
- enzyme inhibitors
- urea compounds
- urea
- compounds
- inhibitors
- Prior art date
Links
- 239000002532 enzyme inhibitor Substances 0.000 title 1
- 150000003672 ureas Chemical class 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C07D233/61—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms not forming part of a nitro radical, attached to ring nitrogen atoms
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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- C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C07—ORGANIC CHEMISTRY
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- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
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- C07D233/88—Nitrogen atoms, e.g. allantoin
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- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Neurology (AREA)
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- Psychiatry (AREA)
- Addiction (AREA)
- Epidemiology (AREA)
- Ophthalmology & Optometry (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
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- Pulmonology (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- Child & Adolescent Psychology (AREA)
- Anesthesiology (AREA)
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- Communicable Diseases (AREA)
- Urology & Nephrology (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261674970P | 2012-07-24 | 2012-07-24 | |
PCT/PT2013/000048 WO2014017936A2 (en) | 2012-07-24 | 2013-07-24 | Urea compounds and their use as enzyme inhibitors |
Publications (1)
Publication Number | Publication Date |
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SG11201500498SA true SG11201500498SA (en) | 2015-03-30 |
Family
ID=48986199
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11201500498SA SG11201500498SA (en) | 2012-07-24 | 2013-07-24 | Urea compounds and their use as enzyme inhibitors |
Country Status (33)
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US (3) | US9549915B2 (en) |
EP (1) | EP2890684B1 (en) |
JP (1) | JP6317345B2 (en) |
KR (1) | KR102137714B1 (en) |
CN (1) | CN104487422B (en) |
AR (1) | AR091888A1 (en) |
AU (1) | AU2013293650B2 (en) |
BR (1) | BR112015001546B1 (en) |
CA (1) | CA2879726A1 (en) |
CL (1) | CL2015000178A1 (en) |
CY (1) | CY1120148T1 (en) |
DK (1) | DK2890684T3 (en) |
ES (1) | ES2667056T3 (en) |
HK (1) | HK1211920A1 (en) |
HR (1) | HRP20180543T1 (en) |
HU (1) | HUE037085T2 (en) |
IL (1) | IL236630B (en) |
IN (1) | IN2015DN00688A (en) |
LT (1) | LT2890684T (en) |
ME (1) | ME03018B (en) |
MX (1) | MX365772B (en) |
NO (1) | NO2923395T3 (en) |
NZ (1) | NZ704651A (en) |
PH (1) | PH12015500156B1 (en) |
PL (1) | PL2890684T3 (en) |
PT (1) | PT2890684T (en) |
RS (1) | RS57146B1 (en) |
RU (1) | RU2685425C2 (en) |
SG (1) | SG11201500498SA (en) |
SI (1) | SI2890684T1 (en) |
TW (1) | TWI624460B (en) |
UA (1) | UA116542C2 (en) |
WO (1) | WO2014017936A2 (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR091888A1 (en) * | 2012-07-24 | 2015-03-11 | Bial Portela & Ca Sa | UREA COMPOUNDS AND ITS USE AS ENZYMES INHIBITORS |
US9047327B2 (en) | 2012-12-03 | 2015-06-02 | Google Technology Holdings LLC | Method and apparatus for developing a social hierarchy |
PL3024825T3 (en) | 2013-07-24 | 2017-12-29 | BIAL - PORTELA & Cª, S.A. | Imidazolecarboxamides and their use as faah inhibitors |
GB201401198D0 (en) | 2014-01-24 | 2014-03-12 | Bial Portela & Ca Sa | Process for the syntheis of substituted urea compounds |
US10702487B2 (en) | 2017-08-19 | 2020-07-07 | Frimline Private Limited | Pharmaceutical composition for prevention of diet induced obesity |
MY186286A (en) | 2017-09-05 | 2021-07-05 | Frimline Private Ltd | A pharmaceutical composition for improving or preventing progression of chronic kidney disease |
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DE2458965C3 (en) | 1974-12-13 | 1979-10-11 | Bayer Ag, 5090 Leverkusen | 3-Amino-indazole-N-carboxylic acid derivatives, process for their preparation and pharmaceuticals containing them |
EP0014810A3 (en) | 1979-01-18 | 1980-11-26 | Fbc Limited | Pesticidal pyrazoles, their production, compositions and uses, as well as intermediates and their preparation |
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