SG10202009266PA - Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acid - Google Patents
Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acidInfo
- Publication number
- SG10202009266PA SG10202009266PA SG10202009266PA SG10202009266PA SG10202009266PA SG 10202009266P A SG10202009266P A SG 10202009266PA SG 10202009266P A SG10202009266P A SG 10202009266PA SG 10202009266P A SG10202009266P A SG 10202009266PA SG 10202009266P A SG10202009266P A SG 10202009266PA
- Authority
- SG
- Singapore
- Prior art keywords
- chlorophenoxy
- isoquinoline
- cyano
- carbonyl
- hydroxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201361756361P | 2013-01-24 | 2013-01-24 |
Publications (1)
Publication Number | Publication Date |
---|---|
SG10202009266PA true SG10202009266PA (en) | 2020-10-29 |
Family
ID=50073508
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11201505748UA SG11201505748UA (en) | 2013-01-24 | 2014-01-23 | Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acid |
SG10202009266PA SG10202009266PA (en) | 2013-01-24 | 2014-01-23 | Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acid |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG11201505748UA SG11201505748UA (en) | 2013-01-24 | 2014-01-23 | Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acid |
Country Status (16)
Country | Link |
---|---|
US (1) | US9643928B2 (en) |
EP (1) | EP2951159B1 (en) |
JP (1) | JP6437456B2 (en) |
KR (1) | KR102233081B1 (en) |
CN (1) | CN105452227B (en) |
AU (1) | AU2014209319B2 (en) |
CA (1) | CA2899024C (en) |
DK (1) | DK2951159T3 (en) |
ES (1) | ES2694297T3 (en) |
HK (1) | HK1217331A1 (en) |
IL (1) | IL240066B (en) |
MX (1) | MX360048B (en) |
RU (1) | RU2666144C2 (en) |
SG (2) | SG11201505748UA (en) |
TW (1) | TWI685487B (en) |
WO (1) | WO2014116849A1 (en) |
Families Citing this family (8)
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CA2528232C (en) | 2003-06-06 | 2010-05-25 | Fibrogen, Inc. | Novel nitrogen-containing heteroaryl compounds and their use in increasing endogenous erythropoietin |
WO2010056767A1 (en) | 2008-11-14 | 2010-05-20 | Fibrogen, Inc. | Thiochromene derivatives as hip hydroxylase inhibitors |
EP2872488B1 (en) | 2012-07-16 | 2018-08-22 | Fibrogen, Inc. | Crystalline forms of a prolyl hydroxylase inhibitor |
HUE034409T2 (en) | 2012-07-16 | 2018-02-28 | Fibrogen Inc | Process for making isoquinoline compounds |
US8883823B2 (en) | 2012-07-16 | 2014-11-11 | Fibrogen, Inc. | Crystalline forms of a prolyl hydroxylase inhibitor |
AU2014209319B2 (en) | 2013-01-24 | 2018-04-19 | Fibrogen, Inc. | Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acid |
EP3708154A1 (en) | 2013-06-06 | 2020-09-16 | Fibrogen, Inc. | Pharmaceutical formulations of a hif hydroxylase inhibitor |
AU2015311333B2 (en) | 2014-09-02 | 2017-11-16 | Sunshine Lake Pharma Co., Ltd. | Quinolinone compound and use thereof |
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-
2014
- 2014-01-23 AU AU2014209319A patent/AU2014209319B2/en active Active
- 2014-01-23 CA CA2899024A patent/CA2899024C/en active Active
- 2014-01-23 WO PCT/US2014/012780 patent/WO2014116849A1/en active Application Filing
- 2014-01-23 SG SG11201505748UA patent/SG11201505748UA/en unknown
- 2014-01-23 TW TW103102462A patent/TWI685487B/en active
- 2014-01-23 DK DK14704030.7T patent/DK2951159T3/en active
- 2014-01-23 EP EP14704030.7A patent/EP2951159B1/en active Active
- 2014-01-23 US US14/763,127 patent/US9643928B2/en active Active
- 2014-01-23 RU RU2015134420A patent/RU2666144C2/en active
- 2014-01-23 ES ES14704030.7T patent/ES2694297T3/en active Active
- 2014-01-23 SG SG10202009266PA patent/SG10202009266PA/en unknown
- 2014-01-23 CN CN201480016402.9A patent/CN105452227B/en active Active
- 2014-01-23 KR KR1020157022614A patent/KR102233081B1/en active IP Right Grant
- 2014-01-23 MX MX2015009617A patent/MX360048B/en active IP Right Grant
- 2014-01-23 JP JP2015555276A patent/JP6437456B2/en active Active
-
2015
- 2015-07-21 IL IL240066A patent/IL240066B/en unknown
-
2016
- 2016-05-11 HK HK16105356.9A patent/HK1217331A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
US9643928B2 (en) | 2017-05-09 |
AU2014209319B2 (en) | 2018-04-19 |
ES2694297T3 (en) | 2018-12-19 |
KR20150129679A (en) | 2015-11-20 |
MX2015009617A (en) | 2016-04-20 |
RU2666144C2 (en) | 2018-09-06 |
DK2951159T3 (en) | 2018-11-19 |
EP2951159B1 (en) | 2018-08-22 |
EP2951159A1 (en) | 2015-12-09 |
CA2899024A1 (en) | 2014-07-31 |
CN105452227A (en) | 2016-03-30 |
SG11201505748UA (en) | 2015-08-28 |
AU2014209319A1 (en) | 2015-08-27 |
JP2016505071A (en) | 2016-02-18 |
JP6437456B2 (en) | 2018-12-12 |
IL240066A0 (en) | 2015-09-24 |
KR102233081B1 (en) | 2021-03-29 |
HK1217331A1 (en) | 2017-01-06 |
MX360048B (en) | 2018-10-19 |
TWI685487B (en) | 2020-02-21 |
IL240066B (en) | 2019-08-29 |
CA2899024C (en) | 2022-01-04 |
CN105452227B (en) | 2018-05-29 |
US20160002170A1 (en) | 2016-01-07 |
TW201444800A (en) | 2014-12-01 |
WO2014116849A1 (en) | 2014-07-31 |
RU2015134420A (en) | 2017-03-03 |
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