SG10201503290TA - Anticancer steroidal lactones unsaturated in position 7 (8) - Google Patents

Anticancer steroidal lactones unsaturated in position 7 (8)

Info

Publication number: SG10201503290TA
Authority: SG; Singapore
Prior art keywords: anticancer; unsaturated; steroidal lactones; lactones; steroidal
Prior art date: 2010-04-27

Application number

SG10201503290TA

Inventor

Rodríguez Rogelio Fernández

Benítez José Fernando Reyes

Solloso Andrés Francesch

Marchante María Del Carmen Cuevas

Original Assignee

Pharma Mar Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2010-04-27

Filing date

2011-04-26

Publication date

2015-06-29

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44544049&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG10201503290T(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2011-04-26 Application filed by Pharma Mar Sa filed Critical Pharma Mar Sa

2015-06-29 Publication of SG10201503290TA publication Critical patent/SG10201503290TA/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J19/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 by a lactone ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
- A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)

SG10201503290TA 2010-04-27 2011-04-26 Anticancer steroidal lactones unsaturated in position 7 (8) SG10201503290TA (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP10382095		2010-04-27

Publications (1)

Publication Number	Publication Date
SG10201503290TA true SG10201503290TA (en)	2015-06-29

Family

ID=44544049

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
SG10201503290TA SG10201503290TA (en)	2010-04-27	2011-04-26	Anticancer steroidal lactones unsaturated in position 7 (8)
SG2012079083A SG185032A1 (en)	2010-04-27	2011-04-26	Anticancer steroidal lactones unsaturated in position 7 (8)

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
SG2012079083A SG185032A1 (en)	2010-04-27	2011-04-26	Anticancer steroidal lactones unsaturated in position 7 (8)

Country Status (29)

Country	Link
US (1)	US8962602B2 (en)
EP (1)	EP2563803B1 (en)
JP (1)	JP5815675B2 (en)
KR (1)	KR101855453B1 (en)
CN (1)	CN102947322B (en)
AU (1)	AU2011247634B2 (en)
BR (1)	BR112012027393B1 (en)
CA (1)	CA2797468C (en)
CL (1)	CL2012003006A1 (en)
CY (1)	CY1117541T1 (en)
DK (1)	DK2563803T3 (en)
ES (1)	ES2574205T3 (en)
HK (1)	HK1183036A1 (en)
HR (1)	HRP20160523T1 (en)
HU (1)	HUE028751T2 (en)
IL (1)	IL222707B (en)
ME (1)	ME02488B (en)
MX (1)	MX2012012523A (en)
MY (1)	MY162934A (en)
NZ (1)	NZ603261A (en)
PL (1)	PL2563803T3 (en)
RS (1)	RS54780B1 (en)
RU (1)	RU2572595C2 (en)
SG (2)	SG10201503290TA (en)
SI (1)	SI2563803T1 (en)
SM (1)	SMT201600139B (en)
UA (1)	UA112746C2 (en)
WO (1)	WO2011134954A1 (en)
ZA (1)	ZA201208092B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE102011083725A1 (en)	2011-09-29	2013-04-04	Bayer Pharma AG	Estra-1,3,5 (10), 16-tetraene-3-carboxamide derivatives, process for their preparation, pharmaceutical preparations containing them and their use for the preparation of medicaments
KR102359214B1 (en)	2014-04-04	2022-02-07	델 마 파마슈티컬스	Use of dianhydrogalactitol and analogs or derivatives thereof to treat non-small-cell carcinoma of the lung and ovarian cancer
CN105017368B (en) *	2015-06-26	2016-09-28	南通大学	Pananxadiol derivatives and preparation method and application
CN105968167B (en) *	2016-05-05	2017-10-17	江苏省中医药研究院	The preparation method and its purposes as antineoplastic of epoxy toadpoison ketenes
JOP20190254A1 (en)	2017-04-27	2019-10-27	Pharma Mar Sa	Antitumoral compounds
CN117015382A (en) *	2021-02-02	2023-11-07	润新生物公司	Certain chemical entities, compositions and methods

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1577633A (en) *	1976-12-17	1980-10-29	Degussa	Acyl derivatives of hellebrigenin
JPH04290899A (en) *	1991-03-18	1992-10-15	Sankyo Co Ltd	Cardenolide compound
JPH05112596A (en) *	1991-10-20	1993-05-07	Reisa Cho	Medicine containing bufalin and bufadienolide as effective components
CA2362917C (en) *	1999-02-12	2003-08-05	Cellpath, Inc.	Methods for anti-tumor therapy
IL135707A0 (en)	2000-04-17	2001-05-20	Yissum Res Dev Co	19-norbufalin derivatives, their preparation and pharmaceutical compositions containing them
WO2002014343A1 (en) *	2000-08-17	2002-02-21	Terness, Peter	Bufadienolide derivatives and use as immunosuppressive, antiinflammatory and analgesic agents
CA2418458A1 (en)	2003-02-06	2004-08-06	Neokimia Inc.	Total synthesis of 14 beta-fluorosteroids via the transannular diels-alder reaction
GB0509829D0 (en)	2005-05-13	2005-06-22	Guys And St Thomas Nhs Foundat	Compound
CN100384830C (en)	2006-01-12	2008-04-30	天津药物研究院	Derivative of cyclo membranousol kind and application thereof
CA2682385A1 (en) *	2006-05-09	2007-11-15	Jr. Roland Valdes	Treating cancer with cardiac glycosides
US20090018088A1 (en) *	2006-10-27	2009-01-15	University Of Louisville Research Foundation	Treating cancer with cardiac glycosides

2011
- 2011-04-26 DK DK11716407.9T patent/DK2563803T3/en active
- 2011-04-26 ME MEP-2016-88A patent/ME02488B/en unknown
- 2011-04-26 MX MX2012012523A patent/MX2012012523A/en active IP Right Grant
- 2011-04-26 UA UAA201213556A patent/UA112746C2/en unknown
- 2011-04-26 SG SG10201503290TA patent/SG10201503290TA/en unknown
- 2011-04-26 ES ES11716407.9T patent/ES2574205T3/en active Active
- 2011-04-26 KR KR1020127031051A patent/KR101855453B1/en active IP Right Grant
- 2011-04-26 CN CN201180031259.7A patent/CN102947322B/en not_active Expired - Fee Related
- 2011-04-26 EP EP11716407.9A patent/EP2563803B1/en active Active
- 2011-04-26 BR BR112012027393-0A patent/BR112012027393B1/en not_active IP Right Cessation
- 2011-04-26 RU RU2012150501/04A patent/RU2572595C2/en active
- 2011-04-26 JP JP2013506629A patent/JP5815675B2/en active Active
- 2011-04-26 SG SG2012079083A patent/SG185032A1/en unknown
- 2011-04-26 US US13/642,910 patent/US8962602B2/en active Active
- 2011-04-26 MY MYPI2012004732A patent/MY162934A/en unknown
- 2011-04-26 WO PCT/EP2011/056566 patent/WO2011134954A1/en active Application Filing
- 2011-04-26 NZ NZ603261A patent/NZ603261A/en not_active IP Right Cessation
- 2011-04-26 PL PL11716407T patent/PL2563803T3/en unknown
- 2011-04-26 RS RS20160305A patent/RS54780B1/en unknown
- 2011-04-26 HU HUE11716407A patent/HUE028751T2/en unknown
- 2011-04-26 SI SI201130811A patent/SI2563803T1/en unknown
- 2011-04-26 AU AU2011247634A patent/AU2011247634B2/en not_active Ceased
- 2011-04-26 CA CA2797468A patent/CA2797468C/en active Active
2012
- 2012-10-25 IL IL222707A patent/IL222707B/en active IP Right Grant
- 2012-10-26 CL CL2012003006A patent/CL2012003006A1/en unknown
- 2012-10-26 ZA ZA2012/08092A patent/ZA201208092B/en unknown
2013
- 2013-09-02 HK HK13110244.8A patent/HK1183036A1/en not_active IP Right Cessation
2016
- 2016-05-17 HR HRP20160523TT patent/HRP20160523T1/en unknown
- 2016-05-17 SM SM201600139T patent/SMT201600139B/en unknown
- 2016-05-24 CY CY20161100445T patent/CY1117541T1/en unknown

Also Published As

Publication number	Publication date
CN102947322B (en)	2016-09-07
US20130040921A1 (en)	2013-02-14
MY162934A (en)	2017-07-31
HK1183036A1 (en)	2013-12-13
ZA201208092B (en)	2014-03-26
DK2563803T3 (en)	2016-05-30
CY1117541T1 (en)	2017-04-26
CA2797468C (en)	2018-04-24
BR112012027393A2 (en)	2017-08-08
PL2563803T3 (en)	2016-08-31
KR101855453B1 (en)	2018-06-20
SG185032A1 (en)	2012-11-29
CL2012003006A1 (en)	2013-10-18
AU2011247634B2 (en)	2016-07-07
JP2013525403A (en)	2013-06-20
EP2563803B1 (en)	2016-03-09
RU2572595C2 (en)	2016-01-20
CA2797468A1 (en)	2011-11-03
EP2563803A1 (en)	2013-03-06
RU2012150501A (en)	2014-06-10
SMT201600139B (en)	2016-07-01
KR20130118730A (en)	2013-10-30
UA112746C2 (en)	2016-10-25
ME02488B (en)	2017-02-20
SI2563803T1 (en)	2016-06-30
RS54780B1 (en)	2016-10-31
NZ603261A (en)	2014-12-24
US8962602B2 (en)	2015-02-24
IL222707B (en)	2018-06-28
WO2011134954A1 (en)	2011-11-03
HUE028751T2 (en)	2017-01-30
HRP20160523T1 (en)	2016-06-03
IL222707A0 (en)	2012-12-31
BR112012027393B1 (en)	2020-12-29
CN102947322A (en)	2013-02-27
JP5815675B2 (en)	2015-11-17
MX2012012523A (en)	2012-12-17
ES2574205T3 (en)	2016-06-15

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