SE391525B - Forfarande for framstellning av nya 6-aminopenicillinsyraderivat med en substituent vid 6-stellningen - Google Patents

Forfarande for framstellning av nya 6-aminopenicillinsyraderivat med en substituent vid 6-stellningen

Info

Publication number
SE391525B
SE391525B SE7107459A SE745971A SE391525B SE 391525 B SE391525 B SE 391525B SE 7107459 A SE7107459 A SE 7107459A SE 745971 A SE745971 A SE 745971A SE 391525 B SE391525 B SE 391525B
Authority
SE
Sweden
Prior art keywords
procedure
acid derivatives
position substituent
preparing new
aminopenicillinic acid
Prior art date
Application number
SE7107459A
Other languages
English (en)
Inventor
B G Christensen
L D Cama
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of SE391525B publication Critical patent/SE391525B/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • C07F9/65611Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system (X = CH2, O, S, NH) optionally with an additional double bond and/or substituents, e.g. penicillins and analogs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/30Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing six-membered aromatic rings
    • C07C57/38Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing six-membered aromatic rings polycyclic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/64Acyl halides
    • C07C57/72Acyl halides containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/64Acyl halides
    • C07C57/76Acyl halides containing halogen outside the carbonyl halide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/08Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D277/12Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
SE7107459A 1970-06-16 1971-06-09 Forfarande for framstellning av nya 6-aminopenicillinsyraderivat med en substituent vid 6-stellningen SE391525B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB2915770 1970-06-16

Publications (1)

Publication Number Publication Date
SE391525B true SE391525B (sv) 1977-02-21

Family

ID=10287044

Family Applications (2)

Application Number Title Priority Date Filing Date
SE7107459A SE391525B (sv) 1970-06-16 1971-06-09 Forfarande for framstellning av nya 6-aminopenicillinsyraderivat med en substituent vid 6-stellningen
SE7404874A SE7404874L (sv) 1970-06-16 1974-04-10

Family Applications After (1)

Application Number Title Priority Date Filing Date
SE7404874A SE7404874L (sv) 1970-06-16 1974-04-10

Country Status (25)

Country Link
JP (1) JPS5715117B1 (sv)
AR (1) AR205683A1 (sv)
AT (3) AT311550B (sv)
BE (1) BE768529A (sv)
CA (1) CA983478A (sv)
CH (1) CH579572A5 (sv)
CS (1) CS190359B2 (sv)
DE (2) DE2151036C2 (sv)
DK (1) DK133301C (sv)
DO (1) DOP1972001821A (sv)
EG (1) EG10970A (sv)
FI (1) FI57418C (sv)
FR (1) FR2100768B1 (sv)
GB (1) GB1339007A (sv)
HU (2) HU168077B (sv)
IE (1) IE35370B1 (sv)
IL (1) IL36990A (sv)
IT (1) IT1057857B (sv)
LU (1) LU63344A1 (sv)
NL (1) NL178876C (sv)
PH (1) PH10995A (sv)
RO (3) RO61560A (sv)
SE (2) SE391525B (sv)
SU (2) SU460629A3 (sv)
ZA (1) ZA713228B (sv)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2199454A2 (en) * 1972-09-15 1974-04-12 Merck & Co Inc 6-Beta-acyl amino penicillanic acids - antibiotics prepared by acylating a 6-alpha-substd -6-beta-amino penicillanic acid
CA1040620A (en) * 1972-11-14 1978-10-17 Frank J. Urban 6-alkoxy-6-acylamidopenicillins 7-alkoxy-7-acylamido acetoxycephalosporins and process
GB1538051A (en) * 1975-01-17 1979-01-10 Beecham Group Ltd 6-methoxy-6-(alpha-carboxyacetamido)-penicillins
US4308259A (en) 1979-03-01 1981-12-29 Beecham Group Limited Penicillin derivatives
JO1395B1 (en) * 1981-07-10 1986-11-30 بيتشام جروب بي ال سي Method for preparing active and antibacterial sleeper derivatives
GB2107307B (en) * 1981-07-25 1986-02-26 Beecham Group Plc B-lactum antibacterial agents

Also Published As

Publication number Publication date
FI57418B (fi) 1980-04-30
DE2129637A1 (de) 1972-01-05
HU167333B (sv) 1975-09-27
AT322738B (de) 1975-06-10
CA983478A (en) 1976-02-10
FR2100768A1 (sv) 1972-03-24
AR205683A1 (es) 1976-05-31
FR2100768B1 (sv) 1974-11-15
SU584786A3 (ru) 1977-12-15
BE768529A (sv) 1971-12-15
DE2129637C2 (de) 1982-07-01
IE35370L (en) 1971-12-16
RO58733A (sv) 1975-11-15
DK133301C (da) 1976-09-27
CS190359B2 (en) 1979-05-31
AT311550B (de) 1973-11-26
DE2151036C2 (de) 1982-03-04
JPS5715117B1 (sv) 1982-03-29
NL7108283A (sv) 1971-12-20
SE7404874L (sv) 1974-04-10
ZA713228B (en) 1972-12-27
CH579572A5 (sv) 1976-09-15
PH10995A (en) 1977-10-20
FI57418C (fi) 1980-08-11
EG10970A (en) 1976-10-31
DE2151036A1 (de) 1972-08-24
RO61560A (sv) 1977-02-15
LU63344A1 (sv) 1972-03-21
HU168077B (sv) 1976-02-28
IE35370B1 (en) 1976-01-21
IT1057857B (it) 1982-03-30
DK133301B (da) 1976-04-26
IL36990A0 (en) 1971-11-29
GB1339007A (en) 1973-11-28
IL36990A (en) 1976-12-31
RO58734A (sv) 1976-01-15
AT320860B (de) 1975-03-10
DOP1972001821A (es) 1977-07-16
SU460629A3 (ru) 1975-02-15
NL178876C (nl) 1986-06-02

Similar Documents

Publication Publication Date Title
SE402284B (sv) Forfarande for framstellning av pyridinderivat
SE393800B (sv) Forfarande for framstellning av bensoylamino-alkyl-fenoxi-alkylkarbonsyraderivat med lipidsenkande effekt
DK444478A (da) Fremgangsmaade til fremstilling af 7-acylaminocephalosporansyre-derivater
BG19162A3 (bg) Метод за получаване на фенил-имидазолил-алканилови производни
SE385885B (sv) Foerfarande foer framstaellning av 4-amino-6-arylpyrimidinderivat
SE399268B (sv) Forfarande for framstellning av nya purinnukleosidderivat
SE390306B (sv) Forfarande for framstellning av piperidinderivat
DK120996B (da) Analogifremgangsmåde til fremstilling af piperidinderivater eller syreadditionssalte deraf.
SE403106B (sv) Forfarande vid framstellning av 14-hydroximorfinanderivat
SE403288B (sv) Forfarande for framstellning av nya aryl-piperazinderivat
SE405477B (sv) Forfarande for framstellning av tetrazolyl-kinaldinsyraderivat med farmakologisk verkan
SE382809B (sv) Forfarande for framstellning av fenoxiettiksyraderivat
DK126043B (da) Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf.
DK135130B (da) Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf.
SE391525B (sv) Forfarande for framstellning av nya 6-aminopenicillinsyraderivat med en substituent vid 6-stellningen
SE381662B (sv) Forfarande for framstellning av nya pyridinderivat
SE392723B (sv) Forfarande for framstellning av nya derivat av 6-aminopenicilliansyra
SE395885B (sv) Forfarande for framstellning av nya kortikotropinpeptider
SE380273B (sv) Forfarande for framstellning av tiopyrimidinderivat
SE406195B (sv) Forfarande for framstellning av bensocykloheptaisokinolinderivat samt syraadditionssalter derav
SE397355B (sv) Analogiforfarande for framstellning av nya penicillansyraderivat
SE393801B (sv) Forfarande for framstellning av tiokarbaminsyraderivat med antifungistatisk lekemedelsverken
SE386674B (sv) Forfarande for framstellning av nya penicilloinsyraderivat
SE386681B (sv) Forfarande for framstellning av nya cefalosporinderivat
DK138850B (da) Analogifremgangsmåde til fremstilling af benzoesyrederivater eller farmaceutisk acceptable salte eller estere deraf.