PT99795A - PREPARATION PROCESS AND NEW DERIVATIVES OF PIPERIDINYL-BENZIMIDAZOLE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents
PREPARATION PROCESS AND NEW DERIVATIVES OF PIPERIDINYL-BENZIMIDAZOLE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEMInfo
- Publication number
- PT99795A PT99795A PT99795A PT9979591A PT99795A PT 99795 A PT99795 A PT 99795A PT 99795 A PT99795 A PT 99795A PT 9979591 A PT9979591 A PT 9979591A PT 99795 A PT99795 A PT 99795A
- Authority
- PT
- Portugal
- Prior art keywords
- benzimidazole
- piperidinyl
- pharmaceutical compositions
- preparation process
- compositions containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US62768790A | 1990-12-14 | 1990-12-14 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT99795A true PT99795A (en) | 1993-04-30 |
| PT99795B PT99795B (en) | 2000-01-31 |
Family
ID=24515699
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT99795A PT99795B (en) | 1990-12-14 | 1991-12-13 | PREPARATION PROCESS AND NEW DERIVATIVES OF PIPERIDINYL-BENZIMIDAZOLE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US5380731A (en) |
| EP (1) | EP0561973A1 (en) |
| JP (1) | JP3112290B2 (en) |
| KR (1) | KR100226954B1 (en) |
| CA (1) | CA2097317C (en) |
| FI (1) | FI932687A (en) |
| HU (1) | HUT64320A (en) |
| NO (1) | NO932147L (en) |
| NZ (1) | NZ240917A (en) |
| PT (1) | PT99795B (en) |
| WO (1) | WO1992010491A1 (en) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT626968E (en) * | 1992-02-13 | 2002-03-28 | Merrell Pharma Inc | TIACICLIC PIPERIDINYL DERIVATIVES |
| GB9312806D0 (en) * | 1993-06-22 | 1993-08-04 | Boots Co Plc | Therapeutic agents |
| US5741800A (en) * | 1993-06-22 | 1998-04-21 | Knoll Aktiengesellachaft | Azolyl-cyclic amine derivates with immunomodulatory activity |
| TW304878B (en) * | 1993-09-21 | 1997-05-11 | Takeda Pharm Industry Co Ltd | |
| RU2257384C2 (en) * | 2000-02-29 | 2005-07-27 | Мицубиси Фарма Корпорейшн | New derivatives of cyclic amide |
| CA2497827A1 (en) * | 2002-09-06 | 2004-03-18 | Janssen Pharmaceutica, N.V. | (1h-benzoimidazol-2-yl)-(piperazinyl)-methanone derivatives and related compounds as histamine h4-receptor antagonists for the treatment of inflammatory and allergic disorders |
| JP4355917B2 (en) * | 2003-10-29 | 2009-11-04 | 信越化学工業株式会社 | Nitrogen-containing organic compound, resist material, and pattern forming method |
| JP5067968B2 (en) * | 2004-10-07 | 2012-11-07 | ビテ ファーマシューティカルズ， インコーポレイテッド | Diaminoalkane aspartic protease inhibitor |
| TWI411607B (en) * | 2005-11-14 | 2013-10-11 | Vitae Pharmaceuticals Inc | Aspartic protease inhibitors |
| ATE520690T1 (en) * | 2006-09-18 | 2011-09-15 | Vitae Pharmaceuticals Inc | PIPERIDINE DERIVATIVES AS RENIN INHIBITORS |
| CL2007002689A1 (en) | 2006-09-18 | 2008-04-18 | Vitae Pharmaceuticals Inc | COMPOUNDS DERIVED FROM PIPERIDIN-1-CARBOXAMIDA, INHIBITORS OF THE RENINE; INTERMEDIARY COMPOUNDS; PHARMACEUTICAL COMPOSITION; AND USE IN THE TREATMENT OF DISEASES SUCH AS HYPERTENSION, CARDIAC INSUFFICIENCY, CARDIAC FIBROSIS, AMONG OTHERS. |
| WO2008153701A1 (en) * | 2007-05-24 | 2008-12-18 | Schering Corporation | Compounds for inhibiting ksp kinesin activity |
| WO2009096996A1 (en) * | 2007-06-20 | 2009-08-06 | Smithkline Beecham Corporation | Renin inhibitors |
| US20100160424A1 (en) * | 2007-06-20 | 2010-06-24 | Baldwin John J | Renin inhibitors |
| DE102008021445B4 (en) | 2008-04-29 | 2016-03-24 | Robert Bosch Gmbh | Web-processing machine and method for its control |
| JP2011525488A (en) * | 2008-06-20 | 2011-09-22 | ヴァイティー ファーマシューティカルズ，インコーポレイテッド | Renin inhibitor and method of use thereof |
| CN102088850A (en) * | 2008-06-26 | 2011-06-08 | 生命医药公司 | Salts of methyl 2-((R))-(3-chlorophenyl)((R)-1-((S)-2-(methylamino)-3((R)-tetrahydro-2H-pyran-3-yl)propylcarbamoyl)piperidin-3-yl)methoxy)ethylcarbamate |
| AR077692A1 (en) * | 2009-08-06 | 2011-09-14 | Vitae Pharmaceuticals Inc | SALTS OF 2 - ((R) - (3-CHLOROPHENYL) ((R) -1 - ((S) -2- (METHYLAMINE) -3 - ((R) -TETRAHYDRO-2H-PIRAN-3-IL) PROPILCARBAMOIL ) PIPERIDIN -3-IL) METOXI) METHYL ETILCARBAMATE |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4219559A (en) * | 1979-01-10 | 1980-08-26 | Janssen Pharmaceutica N.V. | N-Heterocyclyl-4-piperidinamines |
| PH23995A (en) * | 1984-01-09 | 1990-02-09 | Janssen Pharmaceutica Nv | 4((bicycle heterocyclyl)-methyl and hetero)piperidines |
| US4943580A (en) * | 1987-03-09 | 1990-07-24 | Janssen Pharmaceutica N.V. | Anti-histaminic benzimidazole, imidazopyridine and purine derivatives |
| FR2618435B1 (en) * | 1987-07-23 | 1989-10-27 | Synthelabo | BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| US4929618A (en) * | 1988-03-25 | 1990-05-29 | Ube Industries, Ltd. | Piperdine and piperazine derivatives, and antihistaminic pharmaceutical compositions containing the same |
| IT1226100B (en) * | 1988-07-07 | 1990-12-10 | Dompe Farmaceutici Spa | PHARMACOLOGICALLY ACTIVE BENZIMIDAZOLIC DERIVATIVES. |
| US4908372A (en) * | 1988-10-13 | 1990-03-13 | Merrell Dow Pharmaceuticals Inc. | Antihistaminic piperidinyl benzimidazoles |
| US5064840A (en) * | 1989-08-03 | 1991-11-12 | Merrell Dow Pharmaceuticals | Anti-psychotic piperidylbenzimidazole compounds |
| CA2022451C (en) * | 1989-08-03 | 2001-01-23 | Albert Anthony Carr | Anti-psychotic piperidynl benzimidazole compounds |
| WO1992006086A1 (en) * | 1990-10-01 | 1992-04-16 | Janssen Pharmaceutica N.V. | Novel 4-piperidinylcarbonyl derivatives |
| ES2048109B1 (en) * | 1992-07-20 | 1994-12-16 | Espanola Prod Quimicos | PROCEDURE FOR THE PREPARATION OF NEW PIPERIDIC DERIVATIVES OF BENCIMIDAZOLE. |
-
1991
- 1991-11-22 CA CA002097317A patent/CA2097317C/en not_active Expired - Lifetime
- 1991-11-22 HU HU9301730A patent/HUT64320A/en unknown
- 1991-11-22 WO PCT/US1991/008782 patent/WO1992010491A1/en not_active Application Discontinuation
- 1991-11-22 EP EP92901852A patent/EP0561973A1/en not_active Withdrawn
- 1991-11-22 KR KR1019930701772A patent/KR100226954B1/en not_active IP Right Cessation
- 1991-11-22 JP JP04501987A patent/JP3112290B2/en not_active Expired - Lifetime
- 1991-12-10 NZ NZ240917A patent/NZ240917A/en unknown
- 1991-12-13 PT PT99795A patent/PT99795B/en not_active IP Right Cessation
-
1993
- 1993-06-11 FI FI932687A patent/FI932687A/en unknown
- 1993-06-11 NO NO93932147A patent/NO932147L/en unknown
- 1993-08-17 US US08/108,786 patent/US5380731A/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| AU657507B2 (en) | 1995-03-16 |
| HUT64320A (en) | 1993-12-28 |
| JP3112290B2 (en) | 2000-11-27 |
| CA2097317C (en) | 2002-02-12 |
| FI932687A0 (en) | 1993-06-11 |
| NZ240917A (en) | 1994-09-27 |
| KR930703294A (en) | 1993-11-29 |
| EP0561973A1 (en) | 1993-09-29 |
| FI932687A (en) | 1993-06-11 |
| NO932147D0 (en) | 1993-06-11 |
| NO932147L (en) | 1993-06-11 |
| CA2097317A1 (en) | 1992-06-15 |
| HU9301730D0 (en) | 1993-10-28 |
| JPH06503342A (en) | 1994-04-14 |
| AU9114691A (en) | 1992-07-08 |
| PT99795B (en) | 2000-01-31 |
| US5380731A (en) | 1995-01-10 |
| WO1992010491A1 (en) | 1992-06-25 |
| KR100226954B1 (en) | 1999-10-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BB1A | Laying open of patent application |
Effective date: 19920707 |
|
| FG3A | Patent granted, date of granting |
Effective date: 19991027 |
|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 20020430 |
|
| NF3A | Restitutio in integrum |
Free format text: RESTITUTIO IN INTEGRUMO Effective date: 20021014 |
|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 20050427 |