PT89996A - Processo para a preparacao de 3-(2,3,4,5,6-pentafluorofenoxi)-8-azabiciclo{3.2.1}octanos - Google Patents
Processo para a preparacao de 3-(2,3,4,5,6-pentafluorofenoxi)-8-azabiciclo{3.2.1}octanosInfo
- Publication number
- PT89996A PT89996A PT89996A PT8999689A PT89996A PT 89996 A PT89996 A PT 89996A PT 89996 A PT89996 A PT 89996A PT 8999689 A PT8999689 A PT 8999689A PT 89996 A PT89996 A PT 89996A
- Authority
- PT
- Portugal
- Prior art keywords
- pentafluorofenoxy
- octanes
- azabicyclo
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- C07D451/06—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, ***e
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/167,942 US4861889A (en) | 1988-03-14 | 1988-03-14 | 3-(2,3,4,5,6-pentafluorophenoxy)-8-azabicyclo[3.2.1]octanes |
Publications (1)
Publication Number | Publication Date |
---|---|
PT89996A true PT89996A (pt) | 1989-11-10 |
Family
ID=22609452
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT89996A PT89996A (pt) | 1988-03-14 | 1989-03-13 | Processo para a preparacao de 3-(2,3,4,5,6-pentafluorofenoxi)-8-azabiciclo{3.2.1}octanos |
Country Status (5)
Country | Link |
---|---|
US (1) | US4861889A (pt) |
EP (1) | EP0333026A1 (pt) |
JP (1) | JPH01275579A (pt) |
DK (1) | DK120889A (pt) |
PT (1) | PT89996A (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6951849B2 (en) * | 2001-10-02 | 2005-10-04 | Acadia Pharmaceuticals Inc. | Benzimidazolidinone derivatives as muscarinic agents |
MXPA04003103A (es) * | 2001-10-02 | 2004-07-27 | Acadia Pharm Inc | Derivados de bencimidazolidinona como agentes muscarinicos. |
BRPI0411608A (pt) * | 2003-06-24 | 2006-08-08 | Neurosearch As | derivado de 8-aza-biciclo [3.2.1] octano, composição farmacêutica, uso do composto, e, método de tratamento, prevenção ou alìvio de uma doença, um distúrbio ou uma condição de um organismo animal vivo |
JP2008526923A (ja) * | 2005-01-13 | 2008-07-24 | ノイロサーチ アクティーゼルスカブ | 新規8−置換8−アザ−ビシクロ[3.2.1]オクタン誘導体及びモノアミン神経伝達物質再取り込み阻害剤としてのそれらの使用 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH334838A (de) * | 1955-02-15 | 1958-12-15 | Sandoz Ag | Verfahren zur Herstellung von substituierten Nortropinäthern |
GB1164555A (en) * | 1966-09-20 | 1969-09-17 | Chinoin Gyogyszer Es Vegyeszet | New Tropine Derivatives |
US3657253A (en) * | 1970-08-31 | 1972-04-18 | Robins Co Inc A H | 3-aryloxy-8-carbamoylnortropanes |
GB2060619B (en) * | 1979-09-14 | 1983-06-08 | Wyeth John & Brother Ltd | 4-aryl-4-aryloxypiperidines |
US4458075A (en) * | 1982-04-09 | 1984-07-03 | Hoechst-Roussel Pharmaceuticals Inc. | 6-Fluoro-3-[3-(1-heterocyclo)propyl]-1,2-benzisoxazoles |
-
1988
- 1988-03-14 US US07/167,942 patent/US4861889A/en not_active Expired - Fee Related
-
1989
- 1989-03-09 EP EP89104174A patent/EP0333026A1/en not_active Withdrawn
- 1989-03-13 JP JP1058073A patent/JPH01275579A/ja active Pending
- 1989-03-13 DK DK120889A patent/DK120889A/da not_active Application Discontinuation
- 1989-03-13 PT PT89996A patent/PT89996A/pt not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
US4861889A (en) | 1989-08-29 |
DK120889D0 (da) | 1989-03-13 |
JPH01275579A (ja) | 1989-11-06 |
DK120889A (da) | 1989-09-15 |
EP0333026A1 (en) | 1989-09-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC3A | Refusal |
Effective date: 19940421 |