PT87090A - Processo para a preparacao de derivados de imidazopiridinas e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de derivados de imidazopiridinas e de composicoes farmaceuticas que os contem

Info

Publication number
PT87090A
PT87090A PT87090A PT8709088A PT87090A PT 87090 A PT87090 A PT 87090A PT 87090 A PT87090 A PT 87090A PT 8709088 A PT8709088 A PT 8709088A PT 87090 A PT87090 A PT 87090A
Authority
PT
Portugal
Prior art keywords
imitazopyridine
derivatives
preparing
pharmaceutical compositions
compositions containing
Prior art date
Application number
PT87090A
Other languages
English (en)
Other versions
PT87090B (pt
Inventor
Pascal George
John Allen
Guy Jaurand
Daniele De Peretti
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8704276A external-priority patent/FR2612927B1/fr
Priority claimed from FR8704277A external-priority patent/FR2612928B1/fr
Application filed by Synthelabo filed Critical Synthelabo
Publication of PT87090A publication Critical patent/PT87090A/pt
Publication of PT87090B publication Critical patent/PT87090B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Neurology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Transplantation (AREA)
  • Anesthesiology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PT87090A 1987-03-27 1988-03-25 Processo para a preparacao de derivados de imidazopiridinas e de composicoes farmaceuticas que os contem PT87090B (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8704276A FR2612927B1 (fr) 1987-03-27 1987-03-27 Derives d'imidazopyridines, leur preparation et leur application en therapeutique
FR8704277A FR2612928B1 (fr) 1987-03-27 1987-03-27 Derives hydroxyles d'imidazopyridines, leur preparation et leur application en therapeutique

Publications (2)

Publication Number Publication Date
PT87090A true PT87090A (pt) 1988-04-01
PT87090B PT87090B (pt) 1992-07-31

Family

ID=26225872

Family Applications (1)

Application Number Title Priority Date Filing Date
PT87090A PT87090B (pt) 1987-03-27 1988-03-25 Processo para a preparacao de derivados de imidazopiridinas e de composicoes farmaceuticas que os contem

Country Status (17)

Country Link
US (1) US4847263A (pt)
EP (1) EP0289371B1 (pt)
JP (1) JP2733492B2 (pt)
KR (1) KR880011155A (pt)
AR (1) AR243523A1 (pt)
AU (1) AU597809B2 (pt)
CA (1) CA1324139C (pt)
DE (1) DE3865073D1 (pt)
DK (1) DK167388A (pt)
ES (1) ES2026666T3 (pt)
FI (1) FI881434A (pt)
GR (1) GR3003145T3 (pt)
HU (1) HU198048B (pt)
IL (1) IL85840A (pt)
NO (1) NO881333L (pt)
NZ (1) NZ224032A (pt)
PT (1) PT87090B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4791117A (en) * 1986-09-22 1988-12-13 Ortho Pharmaceutical Corporation 2- or 3-aryl substituted imidazo[1,2-a]pyridines and their use as calcium channel blockers
US5032595A (en) * 1989-11-24 1991-07-16 Fidia-Georgetown Institute For The Neurosciences Method of stimulating steroidogenesis with alpidem
FR2727864B1 (fr) 1994-12-12 1997-04-04 Synthelabo Utilisation des ligands des sites de liaison peripherique pour les benzodiazepines pour la preparation de medicaments utiles dans le traitement des neuropathies peripheriques
AUPP278498A0 (en) 1998-04-03 1998-04-30 Australian Nuclear Science & Technology Organisation Peripheral benzodiazepine receptor binding agents
AU2001249672A1 (en) * 2000-03-31 2001-10-15 Ortho-Mcneil Pharmaceutical, Inc. Method for using 2- or 3-aryl substituted imidazo(1,2-a) pyridines as h3 antagonists
EP1268478B1 (en) 2000-03-31 2007-05-02 Ortho-McNeil Pharmaceutical, Inc. Phenyl-substituted imidazopyridines
DE20122435U1 (de) * 2000-04-24 2005-10-06 Teva Pharmaceutical Industries Ltd. Mikronisiertes Zolpidem-Hemitartrat
EP1475093B1 (en) 2000-04-24 2006-09-06 Teva Pharmaceutical Industries Ltd. Micronized Zolpidem hemitartrate
ATE394398T1 (de) * 2002-07-15 2008-05-15 Scinopharm Taiwan Ltd Verfahren zur herstellung von imidazo(1,2- a)pyridin-3-acetamiden
EP1575952B1 (en) * 2002-12-18 2009-02-18 Mallinckrodt Inc. Synthesis of heteroaryl acetamides
WO2006008636A2 (en) * 2004-07-16 2006-01-26 Ranbaxy Laboratories Limited Processes for the preparation of zolpidem and its hemitartrate

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1442707A (en) * 1973-07-07 1976-07-14 Yoshitomi Pharmaceutical Substituted phenylalkanoic acids and their derivatives and pharma ceutical compositions thereof
US4221796A (en) * 1979-09-19 1980-09-09 E. R. Squibb & Sons, Inc. Substituted imidazolo-pyridines and method
FR2492382A1 (fr) * 1980-10-22 1982-04-23 Synthelabo Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique
FR2568880B1 (fr) * 1984-08-07 1986-12-12 Synthelabo Derives d'acylaminomethyl-3 imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique
EP0234970B1 (fr) * 1986-01-22 1991-04-17 Synthelabo Dérivés d'acylaminométhyl-3 imidazo[1,2-a]pyridines, leur préparation et leur application en thérapeutique
FR2599368B1 (fr) * 1986-06-02 1988-08-05 Synthelabo Derives hydroxyles d'imidazopyridines, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
NO881333L (no) 1988-09-28
JPS63258475A (ja) 1988-10-25
AU1373688A (en) 1988-09-29
DE3865073D1 (de) 1991-10-31
FI881434A0 (fi) 1988-03-25
AU597809B2 (en) 1990-06-07
NO881333D0 (no) 1988-03-25
IL85840A (en) 1992-03-29
EP0289371B1 (fr) 1991-09-25
CA1324139C (en) 1993-11-09
DK167388A (da) 1988-09-28
ES2026666T3 (es) 1992-05-01
KR880011155A (ko) 1988-10-26
HU198048B (en) 1989-07-28
EP0289371A1 (fr) 1988-11-02
NZ224032A (en) 1990-05-28
JP2733492B2 (ja) 1998-03-30
FI881434A (fi) 1988-09-28
PT87090B (pt) 1992-07-31
AR243523A1 (es) 1993-08-31
HUT46692A (en) 1988-11-28
IL85840A0 (en) 1988-09-30
US4847263A (en) 1989-07-11
GR3003145T3 (en) 1993-02-17
DK167388D0 (da) 1988-03-25

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Legal Events

Date Code Title Description
FG3A Patent granted, date of granting

Effective date: 19920110