PT81893B - Processo para a preparacao de derivados de labdano e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de derivados de labdano e de composicoes farmaceuticas que os contem

Info

Publication number
PT81893B
PT81893B PT81893A PT8189386A PT81893B PT 81893 B PT81893 B PT 81893B PT 81893 A PT81893 A PT 81893A PT 8189386 A PT8189386 A PT 8189386A PT 81893 B PT81893 B PT 81893B
Authority
PT
Portugal
Prior art keywords
derivatives
labdano
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
PT81893A
Other languages
English (en)
Other versions
PT81893A (de
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of PT81893A publication Critical patent/PT81893A/pt
Publication of PT81893B publication Critical patent/PT81893B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78Ring systems having three or more relevant rings
    • C07D311/92Naphthopyrans; Hydrogenated naphthopyrans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
PT81893A 1985-01-26 1986-01-23 Processo para a preparacao de derivados de labdano e de composicoes farmaceuticas que os contem PT81893B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19853502686 DE3502686A1 (de) 1985-01-26 1985-01-26 Verfahren zur herstellung von labdan-derivaten und ihre verwendung als arzneimittel

Publications (2)

Publication Number Publication Date
PT81893A PT81893A (de) 1986-02-01
PT81893B true PT81893B (pt) 1988-07-01

Family

ID=6260904

Family Applications (1)

Application Number Title Priority Date Filing Date
PT81893A PT81893B (pt) 1985-01-26 1986-01-23 Processo para a preparacao de derivados de labdano e de composicoes farmaceuticas que os contem

Country Status (9)

Country Link
US (1) US4724238A (pt)
EP (1) EP0192056B1 (pt)
JP (1) JPS61176585A (pt)
AT (1) ATE44874T1 (pt)
DE (2) DE3502686A1 (pt)
ES (1) ES8705874A1 (pt)
GR (1) GR860205B (pt)
IE (1) IE860211L (pt)
PT (1) PT81893B (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4963537A (en) * 1985-03-01 1990-10-16 Hoechst-Roussel Pharmaceuticals Inc. Labdane compounds, pharmaceutical compositions and use
US5247097A (en) * 1986-08-28 1993-09-21 Hoechst-Roussel Pharmaceuticals Incorporated Oxolabdanes
US5130332A (en) * 1986-08-28 1992-07-14 Hoechst Roussel Pharmaceuticals Inc. Oxolabdanes
US4978678A (en) * 1986-11-20 1990-12-18 Hoechst-Roussel Pharmaceuticals Inc. 12-halogenated forskolin derivatives
US5646175A (en) * 1987-12-28 1997-07-08 Hoechst Marion Roussel, Inc. Carbamoyloxylabdane compounds
US4920146A (en) * 1986-12-29 1990-04-24 Hoechst Roussel Pharmaceuticals Inc. Carbamoyloxylabdane compounds useful in reducing intraocular pressure
FR2613935B1 (fr) * 1987-04-15 1989-12-01 Roussel Uclaf Association renfermant a titre de principes actifs, un analgesique central et la forskoline
AT389114B (de) * 1987-10-08 1989-10-25 Hoechst Ag 7-acyloxy-6-aminoacyloxypolyoxylabdane und verfahren zu ihrer herstellung
US4883793A (en) * 1988-05-09 1989-11-28 Hoechst-Roussel Pharmaceuticals Inc. Hydrazinocarbonyloxylabdanes for treating cardiac failure
DE68902811D1 (de) * 1988-11-19 1992-10-15 Hoechst Ag Pharmazeutische zusammensetzungen mit einem gehalt an labdan-di-terpenoid-derivaten und pyrimido(6,1-a)isochinolin-4-on-derivaten und ihre anwendung.
US5177207A (en) * 1989-01-11 1993-01-05 Hoechst-Roussel Pharmaceuticals, Inc. 7-aryl and heteroaryl ethers of desacetylforskolin
US4999351A (en) * 1989-01-11 1991-03-12 Hoechst-Roussel Pharmaceuticals, Inc. 7-aryl and heteroaryl ethers of desacetylforskolin
IL89530A0 (en) * 1989-03-08 1989-09-10 Jeffrey J Feigenbaum Compositions containing forskolin
US5093336A (en) * 1989-07-06 1992-03-03 Hoechat-Roussel Pharmaceuticals, Inc. 6- and 7-deoxyforskolin and derivatives thereof
US5145855A (en) * 1989-07-06 1992-09-08 Hoechst Roussel Pharmaceuticals, Inc. 6- and 7-deoxyforskolin and derivatives thereof
DE10048596A1 (de) * 2000-09-30 2002-04-25 Henkel Kgaa Entzündungshemmende Wirkstoffe
US7240135B2 (en) 2004-03-05 2007-07-03 International Business Machines Corporation Method of balancing work load with prioritized tasks across a multitude of communication ports

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE43545B1 (en) * 1975-09-06 1981-03-25 Hoechst Ag Pharmacologically active substance obtainable from plants
DE2557784C2 (de) * 1975-12-22 1986-04-17 Hoechst Ag, 6230 Frankfurt Forskolin, Verfahren zu dessen Gewinnung und diese Verbindung enthaltende pharmazeutische Präparate
DE2640275A1 (de) * 1976-09-08 1978-03-09 Hoechst Ag Pharmakologisch wirksame substanz aus labiaten
AU2717777A (en) * 1976-07-21 1979-01-25 Hoechst Ag Pharmacologically effective substance from plants belonging to the family of labiatae
DE2654796A1 (de) * 1976-12-03 1978-06-08 Hoechst Ag Polyoxygenierte labdan-derivate
US4517200A (en) * 1982-12-27 1985-05-14 Schering-Plough Corporation Method for treating allergic reactions with forskolin
US4564626A (en) * 1983-04-01 1986-01-14 Schering Corporation Methods of inducing bronchodilation
DE3314999A1 (de) * 1983-04-26 1985-03-14 Behringwerke Ag, 3550 Marburg Verwendung des diterpen-derivates forskolin zur immunstimulation
US4476140A (en) * 1983-05-16 1984-10-09 Yale University Composition and method for treatment of glaucoma
EP0167567A1 (en) * 1983-12-14 1986-01-15 Brown University Research Foundation Treatment of metastasis

Also Published As

Publication number Publication date
US4724238A (en) 1988-02-09
IE860211L (en) 1986-07-26
EP0192056B1 (de) 1989-07-26
GR860205B (en) 1986-05-21
ES8705874A1 (es) 1987-05-16
DE3664562D1 (en) 1989-08-31
JPS61176585A (ja) 1986-08-08
EP0192056A1 (de) 1986-08-27
DE3502686A1 (de) 1986-08-14
ATE44874T1 (de) 1989-08-15
PT81893A (de) 1986-02-01
ES551204A0 (es) 1987-05-16

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Effective date: 19930630